Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50012955
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2(Human)
California Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50561797(CHEMBL4757992)
Affinity DataEC50:  9.00E+3nMAssay Description:Positive allosteric modulator activity at human alpha1beta2S GABA-A receptor expressed in Xenopus laevis oocytes assessed as change in GABA EC50 at 4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2(Human)
California Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50561796(CHEMBL4744964)
Affinity DataEC50:  1.30E+4nMAssay Description:Positive allosteric modulator activity at human alpha1beta2S GABA-A receptor expressed in Xenopus laevis oocytes assessed as change in GABA EC50 at 4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2(Human)
California Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50561798(CHEMBL4797104)
Affinity DataEC50:  1.60E+4nMAssay Description:Positive allosteric modulator activity at human alpha1beta2S GABA-A receptor expressed in Xenopus laevis oocytes assessed as change in GABA EC50 at 4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2(Human)
California Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50561799(CHEMBL4783212)
Affinity DataEC50:  1.60E+4nMAssay Description:Positive allosteric modulator activity at human alpha1beta2S GABA-A receptor expressed in Xenopus laevis oocytes assessed as change in GABA EC50 at 4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Human)
California Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50561796(CHEMBL4744964)
Affinity DataEC50:  1.10E+5nMAssay Description:Positive allosteric modulator activity at human alpha1beta2Sgamma2S GABA-A receptor expressed in Xenopus laevis oocytes in presence of EC5 GABA by tw...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed