Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) with all data for entry = 50014784
TargetNuclear receptor subfamily 4 group A member 2(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50580049(CHEMBL5086921)
Affinity DataEC50:  24nMAssay Description:Agonist activity at full length NURR1 (unknown origin) expressed in mouse MND9 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetNuclear receptor subfamily 4 group A member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50071058(CHEMBL301982 | cid_4274774 | (2R,4aS,6aS,12bR,14aS...)
Affinity DataKd:  290nMAssay Description:Binding affinity to Nur77 LBD (unknown origin) expressed in Escherichia coli incubated for 3 hrs by circular dichroism analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed