Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50011459
TargetApolipoprotein L1(Human)
Smith, Gambrell & Russell

Curated by ChEMBL
LigandPNGBDBM50547875(CHEMBL4754532 | US20230271945, Compound 1)
Affinity DataIC50: 250nMAssay Description:Inhibition of APOL1 (unknown origin) in HEK293 cells assessed as thallium influx incubated for 30 mins by FLIPR based thallium influx assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetApolipoprotein L1(Human)
Smith, Gambrell & Russell

Curated by ChEMBL
LigandPNGBDBM50547880(CHEMBL4789274 | US20230271945, Compound 121)
Affinity DataIC50: 250nMAssay Description:Inhibition of APOL1 (unknown origin) in HEK293 cells assessed as thallium influx incubated for 30 mins by FLIPR based thallium influx assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetApolipoprotein L1(Human)
Smith, Gambrell & Russell

Curated by ChEMBL
LigandPNGBDBM50547879(CHEMBL4780017 | US20230271945, Compound 82)
Affinity DataIC50: 250nMAssay Description:Inhibition of APOL1 (unknown origin) in HEK293 cells assessed as thallium influx incubated for 30 mins by FLIPR based thallium influx assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetApolipoprotein L1(Human)
Smith, Gambrell & Russell

Curated by ChEMBL
LigandPNGBDBM50547878(CHEMBL4752052 | US20230271945, Compound 61)
Affinity DataIC50: 250nMAssay Description:Inhibition of APOL1 (unknown origin) in HEK293 cells assessed as thallium influx incubated for 30 mins by FLIPR based thallium influx assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetApolipoprotein L1(Human)
Smith, Gambrell & Russell

Curated by ChEMBL
LigandPNGBDBM50547877(CHEMBL4795347 | US20230271945, Compound 42)
Affinity DataIC50: 250nMAssay Description:Inhibition of APOL1 (unknown origin) in HEK293 cells assessed as thallium influx incubated for 30 mins by FLIPR based thallium influx assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetApolipoprotein L1(Human)
Smith, Gambrell & Russell

Curated by ChEMBL
LigandPNGBDBM50547876(CHEMBL4791770 | US20230271945, Compound 20)
Affinity DataIC50: 250nMAssay Description:Inhibition of APOL1 (unknown origin) in HEK293 cells assessed as thallium influx incubated for 30 mins by FLIPR based thallium influx assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed