Compile Data Set for Download or QSAR
Report error Found 29 Enz. Inhib. hit(s) with all data for entry = 50011947
TargetGlycogen synthase kinase-3 beta(Human)
Charles University

Curated by ChEMBL
LigandPNGBDBM50325983(6-(2-(4-(2,4-dichlorophenyl)-5-(4-methyl-1H-imidaz...)
Affinity DataIC50: 9.90nMAssay Description:Inhibition of human recombinant GSK3beta using GSK3 peptide as substrate preincubated for 15 mins followed by ATP addition and measured after 90 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCathepsin K(Human)
Charles University

Curated by ChEMBL
LigandPNGBDBM50552626(CHEMBL4762594)
Affinity DataIC50: 2.63E+3nMAssay Description:Inhibition of recombinant human Cathepsin K expressed in Pichia pastoris X-33 using Z-Gly-Pro-Arg-AMC as substrate preincubated for 10 mins followed ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetCathepsin K(Human)
Charles University

Curated by ChEMBL
LigandPNGBDBM50552627(CHEMBL4797349)
Affinity DataIC50: 6.34E+3nMAssay Description:Inhibition of recombinant human Cathepsin K expressed in Pichia pastoris X-33 using Z-Gly-Pro-Arg-AMC as substrate preincubated for 10 mins followed ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetCathepsin K(Human)
Charles University

Curated by ChEMBL
LigandPNGBDBM50552629(CHEMBL4740934)
Affinity DataIC50: 9.25E+3nMAssay Description:Inhibition of recombinant human Cathepsin K expressed in Pichia pastoris X-33 using Z-Gly-Pro-Arg-AMC as substrate preincubated for 10 mins followed ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Charles University

Curated by ChEMBL
LigandPNGBDBM50552631(CHEMBL4752567)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant GSK3beta using GSK3 peptide as substrate preincubated for 15 mins followed by ATP addition and measured after 90 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Charles University

Curated by ChEMBL
LigandPNGBDBM50552630(CHEMBL4791863)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant GSK3beta using GSK3 peptide as substrate preincubated for 15 mins followed by ATP addition and measured after 90 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Charles University

Curated by ChEMBL
LigandPNGBDBM50552629(CHEMBL4740934)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant GSK3beta using GSK3 peptide as substrate preincubated for 15 mins followed by ATP addition and measured after 90 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Charles University

Curated by ChEMBL
LigandPNGBDBM50552628(CHEMBL4741923)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant GSK3beta using GSK3 peptide as substrate preincubated for 15 mins followed by ATP addition and measured after 90 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Charles University

Curated by ChEMBL
LigandPNGBDBM50552627(CHEMBL4797349)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant GSK3beta using GSK3 peptide as substrate preincubated for 15 mins followed by ATP addition and measured after 90 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Charles University

Curated by ChEMBL
LigandPNGBDBM50552626(CHEMBL4762594)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant GSK3beta using GSK3 peptide as substrate preincubated for 15 mins followed by ATP addition and measured after 90 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Charles University

Curated by ChEMBL
LigandPNGBDBM50166940(NP-031112 | NP-12 | Tideglusib | med.21724, Compou...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant GSK3beta using GSK3 peptide as substrate preincubated for 15 mins followed by ATP addition and measured after 90 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Charles University

Curated by ChEMBL
LigandPNGBDBM50552645(CHEMBL4763526)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant GSK3beta using GSK3 peptide as substrate preincubated for 15 mins followed by ATP addition and measured after 90 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Charles University

Curated by ChEMBL
LigandPNGBDBM50552644(CHEMBL4793802)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant GSK3beta using GSK3 peptide as substrate preincubated for 15 mins followed by ATP addition and measured after 90 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Charles University

Curated by ChEMBL
LigandPNGBDBM50552643(CHEMBL4741856)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant GSK3beta using GSK3 peptide as substrate preincubated for 15 mins followed by ATP addition and measured after 90 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Charles University

Curated by ChEMBL
LigandPNGBDBM50552642(CHEMBL4779756)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant GSK3beta using GSK3 peptide as substrate preincubated for 15 mins followed by ATP addition and measured after 90 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Charles University

Curated by ChEMBL
LigandPNGBDBM50552641(CHEMBL4747111)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant GSK3beta using GSK3 peptide as substrate preincubated for 15 mins followed by ATP addition and measured after 90 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Charles University

Curated by ChEMBL
LigandPNGBDBM50552640(CHEMBL4756684)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant GSK3beta using GSK3 peptide as substrate preincubated for 15 mins followed by ATP addition and measured after 90 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Charles University

Curated by ChEMBL
LigandPNGBDBM50552639(CHEMBL4778188)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant GSK3beta using GSK3 peptide as substrate preincubated for 15 mins followed by ATP addition and measured after 90 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Charles University

Curated by ChEMBL
LigandPNGBDBM60185(N-(3-hydroxy-1,2,4-thiadiazol-5-yl)benzenecarboxam...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant GSK3beta using GSK3 peptide as substrate preincubated for 15 mins followed by ATP addition and measured after 90 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Charles University

Curated by ChEMBL
LigandPNGBDBM50552638(CHEMBL4759710)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant GSK3beta using GSK3 peptide as substrate preincubated for 15 mins followed by ATP addition and measured after 90 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Charles University

Curated by ChEMBL
LigandPNGBDBM50552637(CHEMBL4778558)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant GSK3beta using GSK3 peptide as substrate preincubated for 15 mins followed by ATP addition and measured after 90 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Charles University

Curated by ChEMBL
LigandPNGBDBM50552636(CHEMBL4762316)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant GSK3beta using GSK3 peptide as substrate preincubated for 15 mins followed by ATP addition and measured after 90 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Charles University

Curated by ChEMBL
LigandPNGBDBM50552635(CHEMBL4782522)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant GSK3beta using GSK3 peptide as substrate preincubated for 15 mins followed by ATP addition and measured after 90 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Charles University

Curated by ChEMBL
LigandPNGBDBM50552634(CHEMBL4753880)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant GSK3beta using GSK3 peptide as substrate preincubated for 15 mins followed by ATP addition and measured after 90 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Charles University

Curated by ChEMBL
LigandPNGBDBM50552633(CHEMBL4790689)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant GSK3beta using GSK3 peptide as substrate preincubated for 15 mins followed by ATP addition and measured after 90 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Charles University

Curated by ChEMBL
LigandPNGBDBM50552632(CHEMBL4777309)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant GSK3beta using GSK3 peptide as substrate preincubated for 15 mins followed by ATP addition and measured after 90 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetCathepsin K(Human)
Charles University

Curated by ChEMBL
LigandPNGBDBM50552628(CHEMBL4741923)
Affinity DataIC50: 1.01E+4nMAssay Description:Inhibition of recombinant human Cathepsin K expressed in Pichia pastoris X-33 using Z-Gly-Pro-Arg-AMC as substrate preincubated for 10 mins followed ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetCathepsin K(Human)
Charles University

Curated by ChEMBL
LigandPNGBDBM50552631(CHEMBL4752567)
Affinity DataIC50: 1.02E+4nMAssay Description:Inhibition of recombinant human Cathepsin K expressed in Pichia pastoris X-33 using Z-Gly-Pro-Arg-AMC as substrate preincubated for 10 mins followed ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetCathepsin K(Human)
Charles University

Curated by ChEMBL
LigandPNGBDBM50552630(CHEMBL4791863)
Affinity DataIC50: 1.49E+4nMAssay Description:Inhibition of recombinant human Cathepsin K expressed in Pichia pastoris X-33 using Z-Gly-Pro-Arg-AMC as substrate preincubated for 10 mins followed ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed