Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50018504
TargetBromodomain-containing protein 4(Human)
Institut De Recherches Cliniques De Montreal (IRCM)

Curated by ChEMBL
LigandPNGBDBM220447(US9296741, 36 | US10633379, Compound X)
Affinity DataIC50: 3nMAssay Description:Inhibition of BRD4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Institut De Recherches Cliniques De Montreal (IRCM)

Curated by ChEMBL
LigandPNGBDBM50260093(CHEMBL4078100)
Affinity DataIC50: 5nMAssay Description:Inhibition of BRD4 BD1 (unknown origin) by chromatin/BRD4 displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetBromodomain-containing protein 4(Human)
Institut De Recherches Cliniques De Montreal (IRCM)

Curated by ChEMBL
LigandPNGBDBM50260093(CHEMBL4078100)
Affinity DataIC50: 5nMAssay Description:Inhibition of BRD4 BD2 (unknown origin) by chromatin/BRD4 displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetBromodomain-containing protein 4(Human)
Institut De Recherches Cliniques De Montreal (IRCM)

Curated by ChEMBL
LigandPNGBDBM50260093(CHEMBL4078100)
Affinity DataIC50: 5nMAssay Description:Inhibition of BRD4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetBromodomain-containing protein 4(Human)
Institut De Recherches Cliniques De Montreal (IRCM)

Curated by ChEMBL
LigandPNGBDBM50365463(CHEMBL1232461)
Affinity DataIC50: 30nMAssay Description:Inhibition of BRD4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Institut De Recherches Cliniques De Montreal (IRCM)

Curated by ChEMBL
LigandPNGBDBM50510872(CHEMBL4303404)
Affinity DataIC50: 39nMAssay Description:Inhibition of BRD4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Institut De Recherches Cliniques De Montreal (IRCM)

Curated by ChEMBL
LigandPNGBDBM50103503(CHEMBL2393130 | US11117865, Compound RVX-208 | US2...)
Affinity DataKd:  135nMAssay Description:Binding affinity to BRD4 BD2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetBromodomain-containing protein 4(Human)
Institut De Recherches Cliniques De Montreal (IRCM)

Curated by ChEMBL
LigandPNGBDBM50045000(CHEMBL9 | (norfloxacin)1-Ethyl-6-fluoro-4-oxo-7-pi...)
Affinity DataIC50: 980nMAssay Description:Inhibition of BRD4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Institut De Recherches Cliniques De Montreal (IRCM)

Curated by ChEMBL
LigandPNGBDBM76305(MLS002695956 | cid_2817 | 5-chloro-8-quinolinol | ...)
Affinity DataIC50: 6.47E+3nMAssay Description:Inhibition of BRD4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed