Compile Data Set for Download or QSAR
maximum 50k data
Found 16 Enz. Inhib. hit(s) with all data for entry = 50048774
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50227275(PD-117558)
Affinity DataIC50:  3.57E+3nMAssay Description:50% inhibitory concentration against DNA-gyraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50227280(CHEMBL15247)
Affinity DataIC50:  6.64E+3nMAssay Description:50% inhibitory concentration against DNA-gyraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50227274(CHEMBL15186)
Affinity DataIC50:  7.13E+3nMAssay Description:50% inhibitory concentration against DNA-gyraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50227279(CHEMBL47028)
Affinity DataIC50:  7.40E+3nMAssay Description:50% inhibitory concentration against DNA-gyraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50227282(CHEMBL275174)
Affinity DataIC50:  7.64E+3nMAssay Description:50% inhibitory concentration against DNA-gyraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50227273(CHEMBL15391)
Affinity DataIC50:  7.66E+3nMAssay Description:50% inhibitory concentration against DNA-gyraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50227283(CHEMBL274469)
Affinity DataIC50:  7.68E+3nMAssay Description:50% inhibitory concentration against DNA-gyraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50227277(CHEMBL15549)
Affinity DataIC50:  8.01E+3nMAssay Description:50% inhibitory concentration against DNA-gyraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM21690(1-cyclopropyl-6-fluoro-4-oxo-7-(piperazin-1-yl)-1,...)
Affinity DataIC50:  1.59E+4nMAssay Description:50% inhibitory concentration against DNA-gyraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045004(9-fluoro-3-methyl-10-(4-methylpiperazin-1-yl)-7-ox...)
Affinity DataIC50:  2.07E+4nMAssay Description:50% inhibitory concentration against DNA-gyraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50227281(CHEMBL359193)
Affinity DataIC50:  3.32E+4nMAssay Description:50% inhibitory concentration against DNA-gyraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50227285(CHEMBL149425)
Affinity DataIC50:  3.70E+4nMAssay Description:50% inhibitory concentration against DNA-gyraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50227278(CHEMBL146339)
Affinity DataIC50:  6.90E+4nMAssay Description:50% inhibitory concentration against DNA-gyraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50227276(CHEMBL356984)
Affinity DataIC50: >2.22E+5nMAssay Description:50% inhibitory concentration against DNA-gyraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50227272(CHEMBL422131)
Affinity DataIC50: >2.46E+5nMAssay Description:50% inhibitory concentration against DNA-gyraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50227284(CHEMBL42299)
Affinity DataIC50: >4.92E+5nMAssay Description:50% inhibitory concentration against DNA-gyraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed