Compile Data Set for Download or QSAR
maximum 50k data
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50002621
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Pacific electric ray)
Stauffer Chemical

Curated by ChEMBL
LigandPNGBDBM50023331((+)-pyrido[3,4-b]homotropane | (+/-)-pyrido[3,4-b]...)
Affinity DataIC50:  0.100nMAssay Description:Inhibition of [3H]-MCC binding to torpedo electroplax membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Pacific electric ray)
Stauffer Chemical

Curated by ChEMBL
LigandPNGBDBM50023330(1-(9-Aza-bicyclo[4.2.1]non-2-en-2-yl)-ethanone | 1...)
Affinity DataIC50:  0.100nMAssay Description:Inhibition of (-)-[3H]-nicotine binding to rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Pacific electric ray)
Stauffer Chemical

Curated by ChEMBL
LigandPNGBDBM50023330(1-(9-Aza-bicyclo[4.2.1]non-2-en-2-yl)-ethanone | 1...)
Affinity DataIC50:  1nMAssay Description:inhibition of (-)-[3H]-nicotine binding to torpedo electroplax membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Pacific electric ray)
Stauffer Chemical

Curated by ChEMBL
LigandPNGBDBM82070(CAS_29790-52-1 | NICOTINE-L (BASE) | Nicotine-D sa...)
Affinity DataIC50:  1nMAssay Description:Inhibition of [3H]-MCC binding to rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Pacific electric ray)
Stauffer Chemical

Curated by ChEMBL
LigandPNGBDBM50023331((+)-pyrido[3,4-b]homotropane | (+/-)-pyrido[3,4-b]...)
Affinity DataIC50:  1nMAssay Description:inhibition of (-)-[3H]-nicotine binding to torpedo electroplax membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Pacific electric ray)
Stauffer Chemical

Curated by ChEMBL
LigandPNGBDBM82070(CAS_29790-52-1 | NICOTINE-L (BASE) | Nicotine-D sa...)
Affinity DataIC50:  4nMAssay Description:Inhibition of (-)-[3H]-nicotine binding to rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Pacific electric ray)
Stauffer Chemical

Curated by ChEMBL
LigandPNGBDBM50023328(3-Pyrrolidin-2-yl-pyridine | CHEMBL1132 | Nornicot...)
Affinity DataIC50:  100nMAssay Description:inhibition of (-)-[3H]-nicotine binding to torpedo electroplax membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Pacific electric ray)
Stauffer Chemical

Curated by ChEMBL
LigandPNGBDBM50023327(3-Methyl-4,13-diaza-tricyclo[8.2.1.0*2,7*]trideca-...)
Affinity DataIC50:  300nMAssay Description:Inhibition of (-)-[3H]-nicotine binding to rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Pacific electric ray)
Stauffer Chemical

Curated by ChEMBL
LigandPNGBDBM50023327(3-Methyl-4,13-diaza-tricyclo[8.2.1.0*2,7*]trideca-...)
Affinity DataIC50:  300nMAssay Description:Inhibition of [3H]-MCC binding to rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Pacific electric ray)
Stauffer Chemical

Curated by ChEMBL
LigandPNGBDBM50023328(3-Pyrrolidin-2-yl-pyridine | CHEMBL1132 | Nornicot...)
Affinity DataIC50:  300nMAssay Description:Inhibition of [3H]-MCC binding to rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Pacific electric ray)
Stauffer Chemical

Curated by ChEMBL
LigandPNGBDBM50023329(13-Methyl-4,13-diaza-tricyclo[8.2.1.0*2,7*]trideca...)
Affinity DataIC50:  800nMAssay Description:Inhibition of (-)-[3H]-nicotine binding to rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Pacific electric ray)
Stauffer Chemical

Curated by ChEMBL
LigandPNGBDBM50023329(13-Methyl-4,13-diaza-tricyclo[8.2.1.0*2,7*]trideca...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of [3H]-MCC binding to rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed