Compile Data Set for Download or QSAR
Report error Found 73 Enz. Inhib. hit(s) with all data for entry = 50013141
TargetNeurotensin receptor type 2(Human)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50563034(CHEMBL4742223)
Affinity DataKi: >1nMAssay Description:Binding affinity to NTS2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Human)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50562998(CHEMBL4786574)
Affinity DataKi:  1.80nMAssay Description:Displacement of [125I]Tyr3-neurotensin from human recombinant NTS1 stably expressed in CHO-K1 cell membranes incubated for 60 mins by gamma counter a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Human)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50562995(CHEMBL4799695)
Affinity DataKi:  2nMAssay Description:Displacement of [125I]Tyr3-neurotensin from human recombinant NTS1 stably expressed in CHO-K1 cell membranes incubated for 60 mins by gamma counter a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Human)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50562996(CHEMBL4751221)
Affinity DataKi:  2.40nMAssay Description:Displacement of [125I]Tyr3-neurotensin from human recombinant NTS1 stably expressed in CHO-K1 cell membranes incubated for 60 mins by gamma counter a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Human)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50562999(CHEMBL4794420)
Affinity DataKi:  2.40nMAssay Description:Displacement of [125I]Tyr3-neurotensin from human recombinant NTS1 stably expressed in CHO-K1 cell membranes incubated for 60 mins by gamma counter a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50562998(CHEMBL4786574)
Affinity DataKi:  2.70nMAssay Description:Displacement of [125I]Tyr3-neurotensin from human recombinant NTS2 stably expressed in human 1321N1 cell membranes incubated for 60 mins by gamma cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Human)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50562997(CHEMBL4799000)
Affinity DataKi:  2.80nMAssay Description:Displacement of [125I]Tyr3-neurotensin from human recombinant NTS1 stably expressed in CHO-K1 cell membranes incubated for 60 mins by gamma counter a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Human)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50563001(CHEMBL4756326)
Affinity DataKi:  2.90nMAssay Description:Displacement of [125I]Tyr3-neurotensin from human recombinant NTS1 stably expressed in CHO-K1 cell membranes incubated for 60 mins by gamma counter a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Human)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50130880(pGlu-Leu-Tyr-Glu-Asn-Lys-Pro-Arg-Arg-Pro-Tyr-Ile-L...)
Affinity DataKi:  3.30nMAssay Description:Displacement of [125I]Tyr3-neurotensin from human recombinant NTS1 stably expressed in CHO-K1 cell membranes incubated for 60 mins by gamma counter a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50130880(pGlu-Leu-Tyr-Glu-Asn-Lys-Pro-Arg-Arg-Pro-Tyr-Ile-L...)
Affinity DataKi:  4.10nMAssay Description:Displacement of [125I]Tyr3-neurotensin from human recombinant NTS2 stably expressed in human 1321N1 cell membranes incubated for 60 mins by gamma cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50563033(CHEMBL4789911)
Affinity DataKi:  4.5nMAssay Description:Binding affinity to NTS2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50563001(CHEMBL4756326)
Affinity DataKi:  4.60nMAssay Description:Displacement of [125I]Tyr3-neurotensin from human recombinant NTS2 stably expressed in human 1321N1 cell membranes incubated for 60 mins by gamma cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Human)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50563000(CHEMBL4787611)
Affinity DataKi:  6nMAssay Description:Displacement of [125I]Tyr3-neurotensin from human recombinant NTS1 stably expressed in CHO-K1 cell membranes incubated for 60 mins by gamma counter a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50562996(CHEMBL4751221)
Affinity DataKi:  6.80nMAssay Description:Displacement of [125I]Tyr3-neurotensin from human recombinant NTS2 stably expressed in human 1321N1 cell membranes incubated for 60 mins by gamma cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50562997(CHEMBL4799000)
Affinity DataKi:  8.70nMAssay Description:Displacement of [125I]Tyr3-neurotensin from human recombinant NTS2 stably expressed in human 1321N1 cell membranes incubated for 60 mins by gamma cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50562995(CHEMBL4799695)
Affinity DataKi:  8.70nMAssay Description:Displacement of [125I]Tyr3-neurotensin from human recombinant NTS2 stably expressed in human 1321N1 cell membranes incubated for 60 mins by gamma cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50562999(CHEMBL4794420)
Affinity DataKi:  8.80nMAssay Description:Displacement of [125I]Tyr3-neurotensin from human recombinant NTS2 stably expressed in human 1321N1 cell membranes incubated for 60 mins by gamma cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50563000(CHEMBL4787611)
Affinity DataKi:  9.30nMAssay Description:Displacement of [125I]Tyr3-neurotensin from human recombinant NTS2 stably expressed in human 1321N1 cell membranes incubated for 60 mins by gamma cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50563003(CHEMBL267714)
Affinity DataKi:  10nMAssay Description:Displacement of [125I]Tyr3-neurotensin from human recombinant NTS2 stably expressed in human 1321N1 cell membranes incubated for 60 mins by gamma cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50563004(CHEMBL4763222)
Affinity DataKi:  16nMAssay Description:Displacement of [125I]Tyr3-neurotensin from human recombinant NTS2 stably expressed in human 1321N1 cell membranes incubated for 60 mins by gamma cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Mouse)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50563026(CHEMBL4748559)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]-neurotensin from NTS1 in mouse brain membrane incubated for 30 mins by liquid scintillation counter analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50563032(CHEMBL4787727)
Affinity DataKi:  24nMAssay Description:Binding affinity to NTS2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50563008(CHEMBL4742361)
Affinity DataKi:  36nMAssay Description:Displacement of [125I]Tyr3-neurotensin from human recombinant NTS2 stably expressed in human 1321N1 cell membranes incubated for 60 mins by gamma cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Human)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50563008(CHEMBL4742361)
Affinity DataKi:  43nMAssay Description:Displacement of [125I]Tyr3-neurotensin from human recombinant NTS1 stably expressed in CHO-K1 cell membranes incubated for 60 mins by gamma counter a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50563014(CHEMBL4788991)
Affinity DataKi:  50nMAssay Description:Displacement of [125I]Tyr3-neurotensin from human recombinant NTS2 stably expressed in human 1321N1 cell membranes incubated for 60 mins by gamma cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Human)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50563002(CHEMBL4753810)
Affinity DataKi:  75nMAssay Description:Displacement of [125I]Tyr3-neurotensin from human recombinant NTS1 stably expressed in CHO-K1 cell membranes incubated for 60 mins by gamma counter a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Mouse)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50563028(CHEMBL4786197)
Affinity DataKi:  83nMAssay Description:Displacement of [3H]-neurotensin from NTS1 in mouse brain membrane incubated for 30 mins by liquid scintillation counter analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50563023(CHEMBL4796587)
Affinity DataKi:  90nMAssay Description:Displacement of [125I]Tyr3-neurotensin from human recombinant NTS2 stably expressed in human 1321N1 cell membranes incubated for 60 mins by gamma cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50563002(CHEMBL4753810)
Affinity DataKi:  95nMAssay Description:Displacement of [125I]Tyr3-neurotensin from human recombinant NTS2 stably expressed in human 1321N1 cell membranes incubated for 60 mins by gamma cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50563021(CHEMBL4740987)
Affinity DataKi:  100nMAssay Description:Displacement of [125I]Tyr3-neurotensin from human recombinant NTS2 stably expressed in human 1321N1 cell membranes incubated for 60 mins by gamma cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Human)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50563004(CHEMBL4763222)
Affinity DataKi:  161nMAssay Description:Displacement of [125I]Tyr3-neurotensin from human recombinant NTS1 stably expressed in CHO-K1 cell membranes incubated for 60 mins by gamma counter a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Human)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50563003(CHEMBL267714)
Affinity DataKi:  174nMAssay Description:Displacement of [125I]Tyr3-neurotensin from human recombinant NTS1 stably expressed in CHO-K1 cell membranes incubated for 60 mins by gamma counter a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50563018(CHEMBL4764437)
Affinity DataKi:  200nMAssay Description:Displacement of [125I]Tyr3-neurotensin from human recombinant NTS2 stably expressed in human 1321N1 cell membranes incubated for 60 mins by gamma cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Human)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50563006(CHEMBL4759247)
Affinity DataKi:  210nMAssay Description:Displacement of [125I]Tyr3-neurotensin from human recombinant NTS1 stably expressed in CHO-K1 cell membranes incubated for 60 mins by gamma counter a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Human)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50458824(CHEMBL4207932)
Affinity DataKi:  300nMAssay Description:Binding affinity to NTS1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50563010(CHEMBL4787163)
Affinity DataKi:  391nMAssay Description:Displacement of [125I]Tyr3-neurotensin from human recombinant NTS2 stably expressed in human 1321N1 cell membranes incubated for 60 mins by gamma cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Mouse)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50563025(CHEMBL4750764)
Affinity DataKi:  410nMAssay Description:Displacement of [3H]-neurotensin from NTS1 in mouse brain membrane incubated for 30 mins by liquid scintillation counter analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Human)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50563030(CHEMBL4779035)
Affinity DataKi:  450nMAssay Description:Displacement of [125I]Tyr3-neurotensin from human recombinant NTS1 stably expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50563005(CHEMBL408057)
Affinity DataKi:  590nMAssay Description:Displacement of [125I]Tyr3-neurotensin from human recombinant NTS2 stably expressed in human 1321N1 cell membranes incubated for 60 mins by gamma cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50563009(CHEMBL4786965)
Affinity DataKi:  620nMAssay Description:Displacement of [125I]Tyr3-neurotensin from human recombinant NTS2 stably expressed in human 1321N1 cell membranes incubated for 60 mins by gamma cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50563007(CHEMBL4749690)
Affinity DataKi:  655nMAssay Description:Displacement of [125I]Tyr3-neurotensin from human recombinant NTS2 stably expressed in human 1321N1 cell membranes incubated for 60 mins by gamma cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50563006(CHEMBL4759247)
Affinity DataKi:  740nMAssay Description:Displacement of [125I]Tyr3-neurotensin from human recombinant NTS2 stably expressed in human 1321N1 cell membranes incubated for 60 mins by gamma cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Mouse)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50563027(CHEMBL4796388)
Affinity DataKi:  770nMAssay Description:Displacement of [3H]-neurotensin from NTS1 in mouse brain membrane incubated for 30 mins by liquid scintillation counter analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50563020(CHEMBL4787256)
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of [125I]Tyr3-neurotensin from human recombinant NTS2 stably expressed in human 1321N1 cell membranes incubated for 60 mins by gamma cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50563016(CHEMBL4760222)
Affinity DataKi:  1.30E+3nMAssay Description:Displacement of [125I]Tyr3-neurotensin from human recombinant NTS2 stably expressed in human 1321N1 cell membranes incubated for 60 mins by gamma cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50563024(CHEMBL4782113)
Affinity DataKi:  1.50E+3nMAssay Description:Displacement of [125I]Tyr3-neurotensin from human recombinant NTS2 stably expressed in human 1321N1 cell membranes incubated for 60 mins by gamma cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50563022(CHEMBL4752398)
Affinity DataKi:  2.20E+3nMAssay Description:Displacement of [125I]Tyr3-neurotensin from human recombinant NTS2 stably expressed in human 1321N1 cell membranes incubated for 60 mins by gamma cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50563019(CHEMBL4758998)
Affinity DataKi:  2.50E+3nMAssay Description:Displacement of [125I]Tyr3-neurotensin from human recombinant NTS2 stably expressed in human 1321N1 cell membranes incubated for 60 mins by gamma cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Human)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50563029(CHEMBL4762781)
Affinity DataKi:  3.50E+3nMAssay Description:Displacement of [3H]-neurotensin from NTS1 in human HT-29 cell membrane incubated for 20 mins by liquid scintillation counter analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50563017(CHEMBL4794489)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]Tyr3-neurotensin from human recombinant NTS2 stably expressed in human 1321N1 cell membranes incubated for 60 mins by gamma cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
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