Compile Data Set for Download or QSAR
Report error Found 75 Enz. Inhib. hit(s) with all data for entry = 50013143
TargetP2X purinoceptor 3(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50257829(Ro-51 | 2-(4-amino-5-(5-iodo-2-isopropyl-4-methoxy...)
Affinity DataIC50: 6.30nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetP2X purinoceptor 3(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM183138(US9688643, I-291 | US9718790, I-0291 | US9150546, ...)
Affinity DataIC50: 9.10nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetP2X purinoceptor 3(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM183166(US9688643, I-326 | US9718790, I-0326 | US9150546, ...)
Affinity DataIC50: 11nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetP2X purinoceptor 3(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM183191(US9688643, I-355 | US9718790, I-0355 | US9150546, ...)
Affinity DataIC50: 13nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetP2X purinoceptor 3(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM183184(US9688643, I-348 | US9718790, I-0348 | US9150546, ...)
Affinity DataIC50: 13nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetP2X purinoceptor 3(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM183132(US9688643, I-285 | US9718790, I-0285 | US9150546, ...)
Affinity DataIC50: 14nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetP2X purinoceptor 3(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50563052(CHEMBL4748113)
Affinity DataIC50: 16nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetP2X purinoceptor 3(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM183201(US9688643, I-365 | US9718790, I-0365 | US9150546, ...)
Affinity DataIC50: 18nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetP2X purinoceptor 3(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM183266(US9688643, I-434 | US9718790, I-0443 | US9150546, ...)
Affinity DataIC50: 20nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetP2X purinoceptor 3(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM183145(US9688643, I-298 | US9718790, I-0298 | US9150546, ...)
Affinity DataIC50: 27nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetP2X purinoceptor 3(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM183200(US9688643, I-364 | US9718790, I-0364 | US9150546, ...)
Affinity DataIC50: 30nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetP2X purinoceptor 3(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM183097(US9688643, I-228 | US9718790, I-0228 | US9150546, ...)
Affinity DataIC50: 31nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetP2X purinoceptor 3(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50563048(CHEMBL4789094)
Affinity DataIC50: 34nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetP2X purinoceptor 3(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM183139(US9688643, I-292 | US9718790, I-0292 | US9150546, ...)
Affinity DataIC50: 34nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetP2X purinoceptor 3(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM183125(US9688643, I-277 | US9718790, I-0277 | US9150546, ...)
Affinity DataIC50: 38nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetP2X purinoceptor 3(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM183121(US9688643, I-273 | US9718790, I-0273 | US9150546, ...)
Affinity DataIC50: 38nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetP2X purinoceptor 2/3(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50257829(Ro-51 | 2-(4-amino-5-(5-iodo-2-isopropyl-4-methoxy...)
Affinity DataIC50: 45nMAssay Description:Antagonist activity at human P2X2/3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetP2X purinoceptor 3(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM183107(US9688643, I-244 | US9718790, I-0244 | US9150546, ...)
Affinity DataIC50: 45nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetP2X purinoceptor 3(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM183146(US9688643, I-299 | US9718790, I-0299 | US9150546, ...)
Affinity DataIC50: 46nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetP2X purinoceptor 3(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM183148(US9688643, I-301 | US9718790, I-0301 | US9150546, ...)
Affinity DataIC50: 48nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetP2X purinoceptor 3(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM183136(US9688643, I-289 | US9718790, I-0289 | US9150546, ...)
Affinity DataIC50: 66nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetP2X purinoceptor 3(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM183199(US9688643, I-363 | US9718790, I-0363 | US9150546, ...)
Affinity DataIC50: 78nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetP2X purinoceptor 3(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM183160(US9688643, I-320 | US9718790, I-0320 | US9150546, ...)
Affinity DataIC50: 83nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetP2X purinoceptor 3(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM183135(US9688643, I-288 | US9718790, I-0288 | US9150546, ...)
Affinity DataIC50: 93nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetP2X purinoceptor 3(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM183089(US9688643, I-200 | US9718790, I-0200 | US9150546, ...)
Affinity DataIC50: 128nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetP2X purinoceptor 3(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50413382(CHEMBL494833)
Affinity DataIC50: 136nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetP2X purinoceptor 3(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50563041(CHEMBL4746334)
Affinity DataIC50: 144nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetP2X purinoceptor 3(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50563036(CHEMBL4787960)
Affinity DataIC50: 149nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetP2X purinoceptor 3(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50563049(CHEMBL4752152)
Affinity DataIC50: 152nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetP2X purinoceptor 3(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM183143(US9688643, I-296 | US9718790, I-0296 | US9150546, ...)
Affinity DataIC50: 176nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetP2X purinoceptor 3(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50563050(CHEMBL4796811)
Affinity DataIC50: 219nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetP2X purinoceptor 3(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM183070(US9688643, I-020 | US9718790, I-0020 | US9150546, ...)
Affinity DataIC50: 389nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetP2X purinoceptor 3(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM183117(US9688643, I-269 | US9718790, I-0269 | US9150546, ...)
Affinity DataIC50: 415nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetP2X purinoceptor 3(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM183110(US9688643, I-248 | US9718790, I-0248 | US9150546, ...)
Affinity DataIC50: 420nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetP2X purinoceptor 3(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM183106(US9688643, I-243 | US9718790, I-0243 | US9150546, ...)
Affinity DataIC50: 450nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetP2X purinoceptor 3(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM183112(US9688643, I-255 | US9718790, I-0255 | US9150546, ...)
Affinity DataIC50: 520nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetP2X purinoceptor 3(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50563051(CHEMBL4788581)
Affinity DataIC50: 614nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetP2X purinoceptor 3(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM183131(US9688643, I-284 | US9718790, I-0284 | US9150546, ...)
Affinity DataIC50: 629nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetP2X purinoceptor 3(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM183103(US9688643, I-240 | US9150546, I-240)
Affinity DataIC50: 953nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetP2X purinoceptor 3(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50563035(CHEMBL4778429)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetP2X purinoceptor 3(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50563037(CHEMBL4797969)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetP2X purinoceptor 3(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50563053(CHEMBL4749540)
Affinity DataIC50: 1.20E+3nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetP2X purinoceptor 2/3(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM183200(US9688643, I-364 | US9718790, I-0364 | US9150546, ...)
Affinity DataIC50: 2.37E+3nMAssay Description:Antagonist activity at human P2X2/3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetP2X purinoceptor 2/3(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50563052(CHEMBL4748113)
Affinity DataIC50: 2.93E+3nMAssay Description:Antagonist activity at human P2X2/3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetP2X purinoceptor 3(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50563043(CHEMBL4759101)
Affinity DataIC50: 3.00E+3nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetP2X purinoceptor 3(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50563044(CHEMBL4743578)
Affinity DataIC50: 3.00E+3nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetP2X purinoceptor 3(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50563045(CHEMBL4797152)
Affinity DataIC50: 3.00E+3nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetP2X purinoceptor 3(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50563046(CHEMBL4750072)
Affinity DataIC50: 3.00E+3nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetP2X purinoceptor 3(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50563047(CHEMBL4750833)
Affinity DataIC50: 3.00E+3nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetP2X purinoceptor 3(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50563038(CHEMBL4753465)
Affinity DataIC50: 3.00E+3nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
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