Compile Data Set for Download or QSAR
Report error Found 29 Enz. Inhib. hit(s) with all data for entry = 50012403
TargetHeat shock protein HSP 90-alpha(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50557372(CHEMBL4741221)
Affinity DataKd:  63nMAssay Description:Binding affinity to HSP90-alpha (unknown origin) expressed in Escherichia coli BL21 by SPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50557372(CHEMBL4741221)
Affinity DataIC50: 160nMAssay Description:Inhibition of HSP90-alpha (unknown origin) expressed in Escherichia coli BL21 assessed as reduction in ATPase activity in presence of PEP, NADH and A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-beta(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50557372(CHEMBL4741221)
Affinity DataIC50: 180nMAssay Description:Inhibition of HSP90-beta (unknown origin) expressed in Escherichia coli BL21 assessed as reduction in ATPase activity in presence of PEP, NADH and AT...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-beta(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50008057(CHEBI:64153 | BMS-722782 | TANESPIMYCIN)
Affinity DataIC50: 810nMAssay Description:Inhibition of HSP90-beta (unknown origin) expressed in Escherichia coli BL21 assessed as reduction in ATPase activity in presence of PEP, NADH and AT...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50008057(CHEBI:64153 | BMS-722782 | TANESPIMYCIN)
Affinity DataIC50: 850nMAssay Description:Inhibition of HSP90-alpha (unknown origin) expressed in Escherichia coli BL21 assessed as reduction in ATPase activity in presence of PEP, NADH and A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50008057(CHEBI:64153 | BMS-722782 | TANESPIMYCIN)
Affinity DataKd:  900nMAssay Description:Binding affinity to HSP90-alpha (unknown origin) expressed in Escherichia coli BL21 by SPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-beta(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50008057(CHEBI:64153 | BMS-722782 | TANESPIMYCIN)
Affinity DataKd:  900nMAssay Description:Binding affinity to HSP90-beta (unknown origin) expressed in Escherichia coli BL21 by SPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50557373(CHEMBL4777111)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of HSP90-alpha (unknown origin) expressed in Escherichia coli BL21 assessed as reduction in ATPase activity in presence of PEP, NADH and A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50557376(CHEMBL4748845)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of HSP90-alpha (unknown origin) expressed in Escherichia coli BL21 assessed as reduction in ATPase activity in presence of PEP, NADH and A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-beta(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50557376(CHEMBL4748845)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of HSP90-beta (unknown origin) expressed in Escherichia coli BL21 assessed as reduction in ATPase activity in presence of PEP, NADH and AT...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-beta(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50557373(CHEMBL4777111)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of HSP90-beta (unknown origin) expressed in Escherichia coli BL21 assessed as reduction in ATPase activity in presence of PEP, NADH and AT...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-beta(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50557379(CHEMBL4759116)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of HSP90-beta (unknown origin) expressed in Escherichia coli BL21 assessed as reduction in ATPase activity in presence of PEP, NADH and AT...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50557379(CHEMBL4759116)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of HSP90-alpha (unknown origin) expressed in Escherichia coli BL21 assessed as reduction in ATPase activity in presence of PEP, NADH and A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50557371(CHEMBL4778213)
Affinity DataKd:  3.10E+3nMAssay Description:Binding affinity to HSP90-alpha (unknown origin) expressed in Escherichia coli BL21 by SPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-beta(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50557370(CHEMBL4777557)
Affinity DataKd:  4.80E+3nMAssay Description:Binding affinity to HSP90-beta (unknown origin) expressed in Escherichia coli BL21 by SPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50557370(CHEMBL4777557)
Affinity DataKd:  4.80E+3nMAssay Description:Binding affinity to HSP90-alpha (unknown origin) expressed in Escherichia coli BL21 by SPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50557378(CHEMBL4777925)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of HSP90-alpha (unknown origin) expressed in Escherichia coli BL21 assessed as reduction in ATPase activity in presence of PEP, NADH and A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-beta(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50557378(CHEMBL4777925)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of HSP90-beta (unknown origin) expressed in Escherichia coli BL21 assessed as reduction in ATPase activity in presence of PEP, NADH and AT...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50557370(CHEMBL4777557)
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of HSP90-alpha (unknown origin) expressed in Escherichia coli BL21 assessed as reduction in ATPase activity in presence of PEP, NADH and A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-beta(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50557370(CHEMBL4777557)
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of HSP90-beta (unknown origin) expressed in Escherichia coli BL21 assessed as reduction in ATPase activity in presence of PEP, NADH and AT...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50557371(CHEMBL4778213)
Affinity DataIC50: 6.20E+3nMAssay Description:Inhibition of HSP90-alpha (unknown origin) expressed in Escherichia coli BL21 assessed as reduction in ATPase activity in presence of PEP, NADH and A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-beta(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50557371(CHEMBL4778213)
Affinity DataKd:  7.00E+3nMAssay Description:Binding affinity to HSP90-beta (unknown origin) expressed in Escherichia coli BL21 by SPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-beta(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50557371(CHEMBL4778213)
Affinity DataIC50: 9.80E+3nMAssay Description:Inhibition of HSP90-beta (unknown origin) expressed in Escherichia coli BL21 assessed as reduction in ATPase activity in presence of PEP, NADH and AT...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50557377(CHEMBL4745924)
Affinity DataIC50: 1.37E+4nMAssay Description:Inhibition of HSP90-alpha (unknown origin) expressed in Escherichia coli BL21 assessed as reduction in ATPase activity in presence of PEP, NADH and A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-beta(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50557377(CHEMBL4745924)
Affinity DataIC50: 1.46E+4nMAssay Description:Inhibition of HSP90-beta (unknown origin) expressed in Escherichia coli BL21 assessed as reduction in ATPase activity in presence of PEP, NADH and AT...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50557375(CHEMBL4760861)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of HSP90-alpha (unknown origin) expressed in Escherichia coli BL21 assessed as reduction in ATPase activity in presence of PEP, NADH and A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50557374(CHEMBL4746322)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of HSP90-alpha (unknown origin) expressed in Escherichia coli BL21 assessed as reduction in ATPase activity in presence of PEP, NADH and A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-beta(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50557375(CHEMBL4760861)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of HSP90-beta (unknown origin) expressed in Escherichia coli BL21 assessed as reduction in ATPase activity in presence of PEP, NADH and AT...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-beta(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50557374(CHEMBL4746322)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of HSP90-beta (unknown origin) expressed in Escherichia coli BL21 assessed as reduction in ATPase activity in presence of PEP, NADH and AT...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed