Compile Data Set for Download or QSAR
Report error Found 41 Enz. Inhib. hit(s) with all data for entry = 50013199
TargetProteasome subunit beta type-8(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50563581(CHEMBL4797911)
Affinity DataIC50: 22nMAssay Description:Inhibition of 20S immunoproteasome beta 5 chymotrypsin-like activity in human H226 cell using Suc-LLVY-AMC as substrate for 10 mins by fluorescence b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetProteasome subunit beta type-8(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50563589(CHEMBL4744255)
Affinity DataIC50: 25nMAssay Description:Inhibition of 20S immunoproteasome beta 5 chymotrypsin-like activity in human H226 cell using Suc-LLVY-AMC as substrate for 10 mins by fluorescence b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetProteasome subunit beta type-8(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50563587(CHEMBL4765143)
Affinity DataIC50: 26nMAssay Description:Inhibition of 20S immunoproteasome beta 5 chymotrypsin-like activity in human H226 cell using Suc-LLVY-AMC as substrate for 10 mins by fluorescence b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetProteasome subunit beta type-8(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50563590(CHEMBL4753369)
Affinity DataIC50: 29nMAssay Description:Inhibition of 20S immunoproteasome beta 5 chymotrypsin-like activity in human H226 cell using Suc-LLVY-AMC as substrate for 10 mins by fluorescence b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetProteasome subunit beta type-8(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50563578(CHEMBL4743601)
Affinity DataIC50: 30nMAssay Description:Inhibition of 20S immunoproteasome beta 5 chymotrypsin-like activity in human H226 cell using Suc-LLVY-AMC as substrate for 10 mins by fluorescence b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetProteasome subunit beta type-8(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50563588(CHEMBL4790349)
Affinity DataIC50: 32nMAssay Description:Inhibition of 20S immunoproteasome beta 5 chymotrypsin-like activity in human H226 cell using Suc-LLVY-AMC as substrate for 10 mins by fluorescence b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetProteasome subunit beta type-8(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50563569(CHEMBL4793363)
Affinity DataIC50: 35nMAssay Description:Inhibition of 20S immunoproteasome beta 5 chymotrypsin-like activity in human H226 cell using Suc-LLVY-AMC as substrate for 10 mins by fluorescence b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetProteasome subunit beta type-8(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50563586(CHEMBL4745732)
Affinity DataIC50: 35nMAssay Description:Inhibition of 20S immunoproteasome beta 5 chymotrypsin-like activity in human H226 cell using Suc-LLVY-AMC as substrate for 10 mins by fluorescence b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetProteasome subunit beta type-8(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50563585(CHEMBL4760977)
Affinity DataIC50: 42nMAssay Description:Inhibition of 20S immunoproteasome beta 5 chymotrypsin-like activity in human H226 cell using Suc-LLVY-AMC as substrate for 10 mins by fluorescence b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetProteasome subunit beta type-8(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50563568(CHEMBL4743123)
Affinity DataIC50: 51nMAssay Description:Inhibition of 20S immunoproteasome beta 5 chymotrypsin-like activity in human H226 cell using Suc-LLVY-AMC as substrate for 10 mins by fluorescence b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetProteasome subunit beta type-8(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50007203(CHEMBL3237875)
Affinity DataIC50: 59nMAssay Description:Inhibition of 20S immunoproteasome beta 5 chymotrypsin-like activity in human H226 cell using Suc-LLVY-AMC as substrate for 10 mins by fluorescence b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetProteasome subunit beta type-8(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50563579(CHEMBL4799577)
Affinity DataIC50: 60nMAssay Description:Inhibition of 20S immunoproteasome beta 5 chymotrypsin-like activity in human H226 cell using Suc-LLVY-AMC as substrate for 10 mins by fluorescence b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetProteasome subunit beta type-8(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50563577(CHEMBL4749833)
Affinity DataIC50: 61nMAssay Description:Inhibition of 20S immunoproteasome beta 5 chymotrypsin-like activity in human H226 cell using Suc-LLVY-AMC as substrate for 10 mins by fluorescence b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetProteasome subunit beta type-8(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50563583(CHEMBL4792535)
Affinity DataIC50: 64nMAssay Description:Inhibition of 20S immunoproteasome beta 5 chymotrypsin-like activity in human H226 cell using Suc-LLVY-AMC as substrate for 10 mins by fluorescence b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetProteasome subunit beta type-8(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50563572(CHEMBL4794207)
Affinity DataIC50: 67nMAssay Description:Inhibition of 20S immunoproteasome beta 5 chymotrypsin-like activity in human H226 cell using Suc-LLVY-AMC as substrate for 10 mins by fluorescence b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetProteasome subunit beta type-8(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50563582(CHEMBL4746065)
Affinity DataIC50: 100nMAssay Description:Inhibition of 20S immunoproteasome beta 5 chymotrypsin-like activity in human H226 cell using Suc-LLVY-AMC as substrate for 10 mins by fluorescence b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetProteasome subunit beta type-2(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50563589(CHEMBL4744255)
Affinity DataIC50: 133nMAssay Description:Inhibition of 20S immunoproteasome beta 2 trypsin-like activity in human H226 cell using Z-LRR-aminoluciferin as substrate for 10 mins by fluorescenc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetProteasome subunit beta type-8(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50563567(CHEMBL4748545)
Affinity DataIC50: 134nMAssay Description:Inhibition of 20S immunoproteasome beta 5 chymotrypsin-like activity in human H226 cell using Suc-LLVY-AMC as substrate for 10 mins by fluorescence b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetProteasome subunit beta type-8(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50563570(CHEMBL4798244)
Affinity DataIC50: 156nMAssay Description:Inhibition of 20S immunoproteasome beta 5 chymotrypsin-like activity in human H226 cell using Suc-LLVY-AMC as substrate for 10 mins by fluorescence b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetProteasome subunit beta type-8(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50563580(CHEMBL4743273)
Affinity DataIC50: 165nMAssay Description:Inhibition of 20S immunoproteasome beta 5 chymotrypsin-like activity in human H226 cell using Suc-LLVY-AMC as substrate for 10 mins by fluorescence b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetProteasome subunit beta type-2(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50563587(CHEMBL4765143)
Affinity DataIC50: 168nMAssay Description:Inhibition of 20S immunoproteasome beta 2 trypsin-like activity in human H226 cell using Z-LRR-aminoluciferin as substrate for 10 mins by fluorescenc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetProteasome subunit beta type-8(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50563573(CHEMBL4742723)
Affinity DataIC50: 231nMAssay Description:Inhibition of 20S immunoproteasome beta 5 chymotrypsin-like activity in human H226 cell using Suc-LLVY-AMC as substrate for 10 mins by fluorescence b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetProteasome subunit beta type-8(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50563562(CHEMBL4756789)
Affinity DataIC50: 234nMAssay Description:Inhibition of 20S immunoproteasome beta 5 chymotrypsin-like activity in human H226 cell using Suc-LLVY-AMC as substrate for 10 mins by fluorescence b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetProteasome subunit beta type-8(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50563575(CHEMBL4787300)
Affinity DataIC50: 243nMAssay Description:Inhibition of 20S immunoproteasome beta 5 chymotrypsin-like activity in human H226 cell using Suc-LLVY-AMC as substrate for 10 mins by fluorescence b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetProteasome subunit beta type-8(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50563566(CHEMBL4799548)
Affinity DataIC50: 311nMAssay Description:Inhibition of 20S immunoproteasome beta 5 chymotrypsin-like activity in human H226 cell using Suc-LLVY-AMC as substrate for 10 mins by fluorescence b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetProteasome subunit beta type-1(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50563587(CHEMBL4765143)
Affinity DataIC50: 361nMAssay Description:Inhibition of 20S immunoproteasome beta 1 caspase-like activity in human H226 cell using Z-nLPnLD-aminoluciferin as substrate for 10 mins by fluoresc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetProteasome subunit beta type-8(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50563591(CHEMBL4758922)
Affinity DataIC50: 365nMAssay Description:Inhibition of 20S immunoproteasome beta 5 chymotrypsin-like activity in human H226 cell using Suc-LLVY-AMC as substrate for 10 mins by fluorescence b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetProteasome subunit beta type-2(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50563569(CHEMBL4793363)
Affinity DataIC50: 381nMAssay Description:Inhibition of 20S immunoproteasome beta 2 trypsin-like activity in human H226 cell using Z-LRR-aminoluciferin as substrate for 10 mins by fluorescenc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetProteasome subunit beta type-8(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50563576(CHEMBL4785143)
Affinity DataIC50: 386nMAssay Description:Inhibition of 20S immunoproteasome beta 5 chymotrypsin-like activity in human H226 cell using Suc-LLVY-AMC as substrate for 10 mins by fluorescence b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetProteasome subunit beta type-1(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50563589(CHEMBL4744255)
Affinity DataIC50: 418nMAssay Description:Inhibition of 20S immunoproteasome beta 1 caspase-like activity in human H226 cell using Z-nLPnLD-aminoluciferin as substrate for 10 mins by fluoresc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetProteasome subunit beta type-8(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50563560(CHEMBL4758923)
Affinity DataIC50: 419nMAssay Description:Inhibition of 20S immunoproteasome beta 5 chymotrypsin-like activity in human H226 cell using Suc-LLVY-AMC as substrate for 10 mins by fluorescence b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetProteasome subunit beta type-2(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50563578(CHEMBL4743601)
Affinity DataIC50: 469nMAssay Description:Inhibition of 20S immunoproteasome beta 2 trypsin-like activity in human H226 cell using Z-LRR-aminoluciferin as substrate for 10 mins by fluorescenc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetProteasome subunit beta type-8(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50563574(CHEMBL4788993)
Affinity DataIC50: 603nMAssay Description:Inhibition of 20S immunoproteasome beta 5 chymotrypsin-like activity in human H226 cell using Suc-LLVY-AMC as substrate for 10 mins by fluorescence b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetProteasome subunit beta type-1(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50563569(CHEMBL4793363)
Affinity DataIC50: 611nMAssay Description:Inhibition of 20S immunoproteasome beta 1 caspase-like activity in human H226 cell using Z-nLPnLD-aminoluciferin as substrate for 10 mins by fluoresc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetProteasome subunit beta type-8(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50563565(CHEMBL4747174)
Affinity DataIC50: 717nMAssay Description:Inhibition of 20S immunoproteasome beta 5 chymotrypsin-like activity in human H226 cell using Suc-LLVY-AMC as substrate for 10 mins by fluorescence b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetProteasome subunit beta type-8(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50563561(CHEMBL4739929)
Affinity DataIC50: 1.03E+3nMAssay Description:Inhibition of 20S immunoproteasome beta 5 chymotrypsin-like activity in human H226 cell using Suc-LLVY-AMC as substrate for 10 mins by fluorescence b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetProteasome subunit beta type-1(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50563578(CHEMBL4743601)
Affinity DataIC50: 1.21E+3nMAssay Description:Inhibition of 20S immunoproteasome beta 1 caspase-like activity in human H226 cell using Z-nLPnLD-aminoluciferin as substrate for 10 mins by fluoresc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetProteasome subunit beta type-8(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50563564(CHEMBL4786861)
Affinity DataIC50: 1.36E+3nMAssay Description:Inhibition of 20S immunoproteasome beta 5 chymotrypsin-like activity in human H226 cell using Suc-LLVY-AMC as substrate for 10 mins by fluorescence b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetProteasome subunit beta type-8(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50563563(CHEMBL4780187)
Affinity DataIC50: 1.75E+3nMAssay Description:Inhibition of 20S immunoproteasome beta 5 chymotrypsin-like activity in human H226 cell using Suc-LLVY-AMC as substrate for 10 mins by fluorescence b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetProteasome subunit beta type-8(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50563571(CHEMBL4762071)
Affinity DataIC50: 2.01E+3nMAssay Description:Inhibition of 20S immunoproteasome beta 5 chymotrypsin-like activity in human H226 cell using Suc-LLVY-AMC as substrate for 10 mins by fluorescence b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetProteasome subunit beta type-8(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50563584(CHEMBL4758374)
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of 20S immunoproteasome beta 5 chymotrypsin-like activity in human H226 cell using Suc-LLVY-AMC as substrate for 10 mins by fluorescence b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed