Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50013887
TargetEpidermal growth factor receptor(Human)
Misr International University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50307940BDBM50307940(N-(4-(3-Bromoanilino)quinazolin-6-yl)-2-(3-oxoisot...)
Affinity DataIC50: 0.360nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Misr International University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50570519BDBM50570519(CHEMBL4858583)
Affinity DataIC50: 0.390nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Misr International University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 112499BDBM112499(DACOMITINIB | US8623883, No. 2 | WO2022090481, Exa...)
Affinity DataIC50: 6nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEpidermal growth factor receptor(Human)
Misr International University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50322823BDBM50322823((S)-N-(4-(3-chloro-4-fluorophenylamino)-7-(tetrahy...)
Affinity DataIC50: 10nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEpidermal growth factor receptor(Human)
Misr International University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50029668BDBM50029668(AZD-9291 | Osimertinib | US10085983, Compound AZD-...)
Affinity DataIC50: 13nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Misr International University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50222435BDBM50222435(6,7-dimethoxy-4-(4-phenylbut-1-ynyl)quinazoline | ...)
Affinity DataIC50: 14nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Misr International University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50570521BDBM50570521(CHEMBL4856453)
Affinity DataIC50: 33nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Misr International University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 5446BDBM5446(Erlotinib | OSI-774 | N-(3-ethynylphenyl)-6,7-bis(...)
Affinity DataIC50: 54nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEpidermal growth factor receptor(Human)
Misr International University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50570526BDBM50570526(CHEMBL4866476)
Affinity DataIC50: 66nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Misr International University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50570520BDBM50570520(CHEMBL4857477)
Affinity DataIC50: 81nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Misr International University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50570523BDBM50570523(CHEMBL1988225)
Affinity DataIC50: 81nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Misr International University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50570524BDBM50570524(CHEMBL4849859)
Affinity DataIC50: 136nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Misr International University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50570522BDBM50570522(CHEMBL4859473)
Affinity DataIC50: 143nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Misr International University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 5447BDBM5447(ZD1839 | N-(3-chloro-4-fluorophenyl)-7-methoxy-6-[...)
Affinity DataIC50: 166nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEpidermal growth factor receptor(Human)
Misr International University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50570525BDBM50570525(CHEMBL4877452)
Affinity DataIC50: 178nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Misr International University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50188458BDBM50188458(1-(2-chloroethyl)-1-nitroso-3-methyl-3-{[4-(3-chlo...)
Affinity DataIC50: 204nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed