Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50015614
TargetFree fatty acid receptor 1(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50587790(CHEMBL5169614)
Affinity DataEC50:  19nMAssay Description:Agonist activity at FFAR1 (unknown origin) expressed in CHO cells assessed as increase in calcium efflux by Fluo-4AM dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetFree fatty acid receptor 1(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50531655(CHEMBL4579901)
Affinity DataEC50:  67nMAssay Description:Agonist activity at FFAR1 (unknown origin) expressed in CHO cells assessed as increase in calcium efflux by Fluo-4AM dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetFree fatty acid receptor 1(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50587791(CHEMBL5175525)
Affinity DataEC50:  110nMAssay Description:Agonist activity at FFAR1 (unknown origin) expressed in CHO cells assessed as increase in calcium efflux by Fluo-4AM dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetFree fatty acid receptor 1(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50587792(CHEMBL5196447)
Affinity DataEC50:  4nMAssay Description:Agonist activity at FFAR1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetFree fatty acid receptor 1(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50543987(CHEMBL4638956)
Affinity DataEC50:  47nMAssay Description:Agonist activity at FFAR1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetFree fatty acid receptor 1(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50386790(CHEMBL1829174 | CHEMBL2047159 | TAK-875 | US119052...)
Affinity DataEC50:  53nMAssay Description:Agonist activity at FFAR1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetFree fatty acid receptor 1(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50587793(CHEMBL5190303)
Affinity DataEC50:  650nMAssay Description:Agonist activity at human FFAR1 expressed in CHO cells assessed as increase in calcium efflux by Fluo-8AM dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetFree fatty acid receptor 1(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50587794(CHEMBL5188313)
Affinity DataEC50:  750nMAssay Description:Agonist activity at human FFAR1 expressed in CHO cells assessed as increase in calcium efflux by Fluo-8AM dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetFree fatty acid receptor 1(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50587795(CHEMBL459548 | S-Phenylmercaptoacetic Acid)
Affinity DataEC50:  6nMAssay Description:Agonist activity at FFAR1 (unknown origin) expressed in CHO cells by FLIPR calcium assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50531655(CHEMBL4579901)
Affinity DataEC50:  470nMAssay Description:Agonist activity at Gal4-fused PPARgamma LBD (unknown origin) expressed in HepG2 cells incubated for 18 hrs by dual luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50587791(CHEMBL5175525)
Affinity DataEC50:  660nMAssay Description:Agonist activity at Gal4-fused PPARgamma LBD (unknown origin) expressed in HepG2 cells incubated for 18 hrs by dual luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed