Compile Data Set for Download or QSAR
Report error Found 28 Enz. Inhib. hit(s) with all data for entry = 50014650
TargetCysteine proteinase falcipain 2a(malaria parasite P. falciparum)
India

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50578419BDBM50578419(CHEMBL4857262)
Affinity DataKi:  2.49E+3nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15 assessed as reduction in free AMC release using Z-FR-AM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 2a(malaria parasite P. falciparum)
India

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50578421BDBM50578421(CHEMBL4850572)
Affinity DataKi:  2.60E+3nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15 assessed as reduction in free AMC release using Z-FR-AM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 2a(malaria parasite P. falciparum)
India

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50578417BDBM50578417(CHEMBL4868442)
Affinity DataKi:  2.78E+3nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15 assessed as reduction in free AMC release using Z-FR-AM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 2a(malaria parasite P. falciparum)
India

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50578406BDBM50578406(CHEMBL4869807)
Affinity DataKi:  3.32E+3nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15 assessed as reduction in free AMC release using Z-FR-AM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 2a(malaria parasite P. falciparum)
India

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50578419BDBM50578419(CHEMBL4857262)
Affinity DataIC50: 3.38E+3nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15 assessed as reduction in free AMC release using Z-FR-AM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 2a(malaria parasite P. falciparum)
India

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50578405BDBM50578405(CHEMBL4856045)
Affinity DataKi:  3.49E+3nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15 assessed as reduction in free AMC release using Z-FR-AM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 2a(malaria parasite P. falciparum)
India

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50578421BDBM50578421(CHEMBL4850572)
Affinity DataIC50: 3.53E+3nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15 assessed as reduction in free AMC release using Z-FR-AM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 2a(malaria parasite P. falciparum)
India

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50578417BDBM50578417(CHEMBL4868442)
Affinity DataIC50: 3.78E+3nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15 assessed as reduction in free AMC release using Z-FR-AM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 2a(malaria parasite P. falciparum)
India

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50578408BDBM50578408(CHEMBL4857754)
Affinity DataKi:  4.54E+3nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15 assessed as reduction in free AMC release using Z-FR-AM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 2a(malaria parasite P. falciparum)
India

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50578406BDBM50578406(CHEMBL4869807)
Affinity DataIC50: 5.62E+3nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15 assessed as reduction in free AMC release using Z-FR-AM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 2a(malaria parasite P. falciparum)
India

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50578405BDBM50578405(CHEMBL4856045)
Affinity DataIC50: 5.90E+3nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15 assessed as reduction in free AMC release using Z-FR-AM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 2a(malaria parasite P. falciparum)
India

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50578420BDBM50578420(CHEMBL4853187)
Affinity DataKi:  6.91E+3nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15 assessed as reduction in free AMC release using Z-FR-AM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 2a(malaria parasite P. falciparum)
India

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50578408BDBM50578408(CHEMBL4857754)
Affinity DataIC50: 7.67E+3nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15 assessed as reduction in free AMC release using Z-FR-AM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 2a(malaria parasite P. falciparum)
India

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50578420BDBM50578420(CHEMBL4853187)
Affinity DataIC50: 9.38E+3nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15 assessed as reduction in free AMC release using Z-FR-AM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 2a(malaria parasite P. falciparum)
India

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50578418BDBM50578418(CHEMBL4871791)
Affinity DataKi:  9.92E+3nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15 assessed as reduction in free AMC release using Z-FR-AM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 2a(malaria parasite P. falciparum)
India

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50578422BDBM50578422(CHEMBL4845812)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15 assessed as reduction in free AMC release using Z-FR-AM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 2a(malaria parasite P. falciparum)
India

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50578418BDBM50578418(CHEMBL4871791)
Affinity DataIC50: 1.35E+4nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15 assessed as reduction in free AMC release using Z-FR-AM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 2a(malaria parasite P. falciparum)
India

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50578410BDBM50578410(CHEMBL4859406)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15 assessed as reduction in free AMC release using Z-FR-AM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 2a(malaria parasite P. falciparum)
India

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50578411BDBM50578411(CHEMBL4858403)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15 assessed as reduction in free AMC release using Z-FR-AM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 2a(malaria parasite P. falciparum)
India

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50578412BDBM50578412(CHEMBL4854350)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15 assessed as reduction in free AMC release using Z-FR-AM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 2a(malaria parasite P. falciparum)
India

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50578413BDBM50578413(CHEMBL4860649)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15 assessed as reduction in free AMC release using Z-FR-AM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 2a(malaria parasite P. falciparum)
India

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50578414BDBM50578414(CHEMBL4863049)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15 assessed as reduction in free AMC release using Z-FR-AM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 2a(malaria parasite P. falciparum)
India

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50578415BDBM50578415(CHEMBL4859035)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15 assessed as reduction in free AMC release using Z-FR-AM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 2a(malaria parasite P. falciparum)
India

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50578416BDBM50578416(CHEMBL4870203)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15 assessed as reduction in free AMC release using Z-FR-AM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 2a(malaria parasite P. falciparum)
India

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50578403BDBM50578403(CHEMBL4870974)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15 assessed as reduction in free AMC release using Z-FR-AM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 2a(malaria parasite P. falciparum)
India

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50578404BDBM50578404(CHEMBL4864385)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15 assessed as reduction in free AMC release using Z-FR-AM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 2a(malaria parasite P. falciparum)
India

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50578407BDBM50578407(CHEMBL4861198)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15 assessed as reduction in free AMC release using Z-FR-AM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 2a(malaria parasite P. falciparum)
India

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50578409BDBM50578409(CHEMBL307261)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15 assessed as reduction in free AMC release using Z-FR-AM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed