Found 11 Enz. Inhib. hit(s) with all data for entry = 50011497 
Affinity DataEC50: 20nMAssay Description:Agonist activity at rat NTR1 expressed in CHO cells assessed as effect on [3H] phosphoinositide accumulation using neurotensin (1 to 13 residues) as ...More data for this Ligand-Target Pair
TargetMas-related G-protein coupled receptor member X1(Homo sapiens (Human))
University Of Queensland
Curated by ChEMBL
University Of Queensland
Curated by ChEMBL
Affinity DataEC50: 500nMAssay Description:Activation of human MrgprX1 expressed in BAM 8-22 activated-rat KNRK cells by fura2-AM dye based calcium imaging assayMore data for this Ligand-Target Pair
TargetMas-related G-protein coupled receptor member X1(Homo sapiens (Human))
University Of Queensland
Curated by ChEMBL
University Of Queensland
Curated by ChEMBL
Affinity DataEC50: 1.80E+3nMAssay Description:Activation of human MrgprX1 expressed in BAM 8-22 activated-rat KNRK cells by fura2-AM dye based calcium imaging assayMore data for this Ligand-Target Pair
TargetMas-related G-protein coupled receptor member X1(Homo sapiens (Human))
University Of Queensland
Curated by ChEMBL
University Of Queensland
Curated by ChEMBL
Affinity DataEC50: 1.80E+3nMAssay Description:Activation of human MrgprX1 expressed in BAM 8-22 activated-rat KNRK cells by fura2-AM dye based calcium imaging assayMore data for this Ligand-Target Pair
Affinity DataEC50: 3.00E+3nMAssay Description:Modulation of rat ASIC3 expressed in Xenopus laevis oocytes at -70 mV holding potential by two-electrode voltage clamp methodMore data for this Ligand-Target Pair
Affinity DataEC50: 12nMAssay Description:Activation of human IR-B expressed in mouse NIH3T3 cells assessed as increase in Akt phosphorylation at Ser473 residue incubated for 30 mins by HTRF ...More data for this Ligand-Target Pair
Affinity DataEC50: 12nMAssay Description:Activation of human IR-B expressed in mouse NIH3T3 cells assessed as increase in Akt phosphorylation at Ser473 residue incubated for 30 mins by HTRF ...More data for this Ligand-Target Pair
Affinity DataEC50: 12nMAssay Description:Activation of human IR-B expressed in mouse NIH3T3 cells assessed as increase in Akt phosphorylation at Ser473 residue incubated for 30 mins by HTRF ...More data for this Ligand-Target Pair
Affinity DataEC50: 12nMAssay Description:Activation of human IR-B expressed in mouse NIH3T3 cells assessed as increase in Akt phosphorylation at Ser473 residue incubated for 30 mins by HTRF ...More data for this Ligand-Target Pair
Affinity DataEC50: 12nMAssay Description:Activation of human IR-B expressed in mouse NIH3T3 cells assessed as increase in Akt phosphorylation at Ser473 residue incubated for 30 mins by HTRF ...More data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+3nMAssay Description:Agonist activity at human V1bR expressed in African green monkey COS-1 cells assessed as increase in intracellular calcium response by FLIPR assayMore data for this Ligand-Target Pair
