Affinity DataIC50: 1.30nMAssay Description:Inhibition of GSK3 (unknown origin)More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Zunyi Medical University
Curated by ChEMBL
Zunyi Medical University
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of FLT3 (unknown origin)More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Homo sapiens (Human))
Zunyi Medical University
Curated by ChEMBL
Zunyi Medical University
Curated by ChEMBL
Affinity DataIC50: 4.40nMAssay Description:Inhibition of RET (unknown origin)More data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta/[Tau protein] kinase(Sus scrofa)
Zunyi Medical University
Curated by ChEMBL
Zunyi Medical University
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of porcine brain GSK-3alpha/beta incubated for 30 mins in presence of [33p]-gamma ATP by scintillation counter analysisMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Zunyi Medical University
Curated by ChEMBL
Zunyi Medical University
Curated by ChEMBL
Affinity DataIC50: 5.5nMAssay Description:Inhibition of GSK3beta (unknown origin)More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Zunyi Medical University
Curated by ChEMBL
Zunyi Medical University
Curated by ChEMBL
Affinity DataIC50: 7.90nMAssay Description:Inhibition of FLT3 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibition of recombinant Lyn (unknown origin)More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Zunyi Medical University
Curated by ChEMBL
Zunyi Medical University
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of recombinant c-Src (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibition of recombinant JAK2 (unknown origin)More data for this Ligand-Target Pair
TargetNon-receptor tyrosine-protein kinase TYK2(Homo sapiens (Human))
Zunyi Medical University
Curated by ChEMBL
Zunyi Medical University
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of recombinant Tyk2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibition of recombinant Hck (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibition of recombinant JAK1 (unknown origin)More data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta/[Tau protein] kinase(Sus scrofa)
Zunyi Medical University
Curated by ChEMBL
Zunyi Medical University
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of porcine brain GSK-3alpha/beta incubated for 30 mins in presence of [33p]-gamma ATP by scintillation counter analysisMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Zunyi Medical University
Curated by ChEMBL
Zunyi Medical University
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of GSK3beta (unknown origin) assessed as decrease in tau phosphorylation at Ser214 residue incubated for 30 mins by Western blot assayMore data for this Ligand-Target Pair
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Zunyi Medical University
Curated by ChEMBL
Zunyi Medical University
Curated by ChEMBL
Affinity DataIC50: 35nMAssay Description:Inhibition of CDK2/cyclin A (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Zunyi Medical University
Curated by ChEMBL
Zunyi Medical University
Curated by ChEMBL
Affinity DataIC50: 65nMAssay Description:Inhibition of CDK5/p35 (unknown origin)More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Zunyi Medical University
Curated by ChEMBL
Zunyi Medical University
Curated by ChEMBL
Affinity DataIC50: 79nMAssay Description:Inhibition of recombinant FLT3 (unknown origin) in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Zunyi Medical University
Curated by ChEMBL
Zunyi Medical University
Curated by ChEMBL
Affinity DataIC50: 83nMAssay Description:Inhibition of GST-fused CDK5/p25 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Zunyi Medical University
Curated by ChEMBL
Zunyi Medical University
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of CDK5/p35 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of Aurora C (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of Aurora C (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Zunyi Medical University
Curated by ChEMBL
Zunyi Medical University
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of GST-fused CDK5/p25 (unknown origin)More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Zunyi Medical University
Curated by ChEMBL
Zunyi Medical University
Curated by ChEMBL
Affinity DataIC50: 101nMAssay Description:Inhibition of recombinant FLT3 D835Y mutant (unknown origin) in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Zunyi Medical University
Curated by ChEMBL
Zunyi Medical University
Curated by ChEMBL
Affinity DataIC50: 101nMAssay Description:Inhibition of FLT3 (unknown origin)More data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Zunyi Medical University
Curated by ChEMBL
Zunyi Medical University
Curated by ChEMBL
Affinity DataIC50: 190nMAssay Description:Inhibition of GSK3beta (unknown origin) in presence of ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 222nMAssay Description:Inhibition of Aurora A (unknown origin)More data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Zunyi Medical University
Curated by ChEMBL
Zunyi Medical University
Curated by ChEMBL
Affinity DataIC50: 239nMAssay Description:Inhibition of c-met (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Zunyi Medical University
Curated by ChEMBL
Zunyi Medical University
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of CDK4/cyclin D1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibition of LCK (unknown origin) in presence of ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 370nMAssay Description:Inhibition of Aurora A (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))
Zunyi Medical University
Curated by ChEMBL
Zunyi Medical University
Curated by ChEMBL
Affinity DataIC50: 380nMAssay Description:Inhibition of SGK (unknown origin) in presence of ATPMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Zunyi Medical University
Curated by ChEMBL
Zunyi Medical University
Curated by ChEMBL
Affinity DataIC50: 430nMAssay Description:Inhibition of recombinant c-Src (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Zunyi Medical University
Curated by ChEMBL
Zunyi Medical University
Curated by ChEMBL
Affinity DataIC50: 440nMAssay Description:Inhibition of CDK2/cyclin A (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 523nMAssay Description:Inhibition of recombinant JAK2 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Zunyi Medical University
Curated by ChEMBL
Zunyi Medical University
Curated by ChEMBL
Affinity DataIC50: 590nMAssay Description:Inhibition of GST-fused human CDK2/cyclin A expressed in Escherichia coli using histone H1 as substrate in presence of [33p]-gamma ATP and MgATPMore data for this Ligand-Target Pair
Affinity DataIC50: 690nMAssay Description:Inhibition of JAK3 (unknown origin)More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Zunyi Medical University
Curated by ChEMBL
Zunyi Medical University
Curated by ChEMBL
Affinity DataIC50: 950nMAssay Description:Inhibition of VEGFR2 (unknown origin)More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Zunyi Medical University
Curated by ChEMBL
Zunyi Medical University
Curated by ChEMBL
Affinity DataIC50: 950nMAssay Description:Inhibition of c-SRC in human MDA-MB-468 cells in presence of [gamma-32P]ATP and ATP by immunoprecipitation methodMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta/[Tau protein] kinase(Sus scrofa)
Zunyi Medical University
Curated by ChEMBL
Zunyi Medical University
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of porcine brain GSK-3alpha/beta incubated for 30 mins in presence of [33p]-gamma ATP by scintillation counter analysisMore data for this Ligand-Target Pair
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Zunyi Medical University
Curated by ChEMBL
Zunyi Medical University
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of CDK2/cyclin A (unknown origin)More data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Homo sapiens (Human))
Zunyi Medical University
Curated by ChEMBL
Zunyi Medical University
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of human recombinant GST-fused PDK1 expressed in Sf9 cells incubated for 30 mins in presence of [gamma-33P]ATP by scintillation counter an...More data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of Aurora A (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Zunyi Medical University
Curated by ChEMBL
Zunyi Medical University
Curated by ChEMBL
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of CDK2/cyclin A (unknown origin)More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Zunyi Medical University
Curated by ChEMBL
Zunyi Medical University
Curated by ChEMBL
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of FGFR1 (unknown origin)More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Zunyi Medical University
Curated by ChEMBL
Zunyi Medical University
Curated by ChEMBL
Affinity DataIC50: 3.19E+3nMAssay Description:Inhibition of recombinant FLT3 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Zunyi Medical University
Curated by ChEMBL
Zunyi Medical University
Curated by ChEMBL
Affinity DataIC50: 3.33E+3nMAssay Description:Inhibition of CDK4/cyclin D1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibition of Aurora B (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Zunyi Medical University
Curated by ChEMBL
Zunyi Medical University
Curated by ChEMBL
Affinity DataIC50: 5.50E+3nMAssay Description:Inhibition of CDK5/p35 (unknown origin)More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Zunyi Medical University
Curated by ChEMBL
Zunyi Medical University
Curated by ChEMBL
Affinity DataIC50: 7.89E+3nMAssay Description:Inhibition of recombinant FLT3 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of Aurora B (unknown origin)More data for this Ligand-Target Pair