Compile Data Set for Download or QSAR
Report error Found 30 Enz. Inhib. hit(s) with all data for entry = 50014236
TargetNucleosome-remodeling factor subunit BPTF(Human)
Fujian Medical University

Curated by ChEMBL
LigandPNGBDBM50573840(CHEMBL4860578)
Affinity DataIC50: 16nMAssay Description:Inhibition of N-terminal GST-tagged human BPTF (2914 to 3037 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Fujian Medical University

Curated by ChEMBL
LigandPNGBDBM50573844(CHEMBL4873042)
Affinity DataIC50: 27nMAssay Description:Inhibition of N-terminal GST-tagged human BPTF (2914 to 3037 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Fujian Medical University

Curated by ChEMBL
LigandPNGBDBM50573839(CHEMBL4870170)
Affinity DataIC50: 29nMAssay Description:Inhibition of N-terminal GST-tagged human BPTF (2914 to 3037 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Fujian Medical University

Curated by ChEMBL
LigandPNGBDBM50573837(CHEMBL4867072)
Affinity DataIC50: 33nMAssay Description:Inhibition of N-terminal GST-tagged human BPTF (2914 to 3037 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Fujian Medical University

Curated by ChEMBL
LigandPNGBDBM50573838(CHEMBL4868713)
Affinity DataIC50: 37nMAssay Description:Inhibition of N-terminal GST-tagged human BPTF (2914 to 3037 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Fujian Medical University

Curated by ChEMBL
LigandPNGBDBM50573845(CHEMBL4851594)
Affinity DataIC50: 59nMAssay Description:Inhibition of N-terminal GST-tagged human BPTF (2914 to 3037 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Fujian Medical University

Curated by ChEMBL
LigandPNGBDBM50573849(CHEMBL4866637)
Affinity DataIC50: 59nMAssay Description:Inhibition of N-terminal GST-tagged human BPTF (2914 to 3037 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Fujian Medical University

Curated by ChEMBL
LigandPNGBDBM50573848(CHEMBL4862619)
Affinity DataIC50: 64nMAssay Description:Inhibition of N-terminal GST-tagged human BPTF (2914 to 3037 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Fujian Medical University

Curated by ChEMBL
LigandPNGBDBM50573852(CHEMBL4780673)
Affinity DataKd:  71nMAssay Description:Binding affinity to BPTF (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetNucleosome-remodeling factor subunit BPTF(Human)
Fujian Medical University

Curated by ChEMBL
LigandPNGBDBM50573841(CHEMBL4852588)
Affinity DataIC50: 114nMAssay Description:Inhibition of N-terminal GST-tagged human BPTF (2914 to 3037 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Fujian Medical University

Curated by ChEMBL
LigandPNGBDBM50573844(CHEMBL4873042)
Affinity DataEC50:  120nMAssay Description:Displacement of Halo-tagged histone H4 from NanoLuc-tagged BPTF (unknown origin) expressed in HEK293 cells by NanoBRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Fujian Medical University

Curated by ChEMBL
LigandPNGBDBM50514899(CHEMBL4461619)
Affinity DataKd:  120nMAssay Description:Binding affinity to BPTF (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Fujian Medical University

Curated by ChEMBL
LigandPNGBDBM50573846(CHEMBL4853486)
Affinity DataIC50: 145nMAssay Description:Inhibition of N-terminal GST-tagged human BPTF (2914 to 3037 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Fujian Medical University

Curated by ChEMBL
LigandPNGBDBM50573850(CHEMBL4861221)
Affinity DataIC50: 157nMAssay Description:Inhibition of N-terminal GST-tagged human BPTF (2914 to 3037 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Fujian Medical University

Curated by ChEMBL
LigandPNGBDBM50514899(CHEMBL4461619)
Affinity DataKd:  200nMAssay Description:Binding affinity to BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Fujian Medical University

Curated by ChEMBL
LigandPNGBDBM50573842(CHEMBL4863921)
Affinity DataIC50: 288nMAssay Description:Inhibition of N-terminal GST-tagged human BPTF (2914 to 3037 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Fujian Medical University

Curated by ChEMBL
LigandPNGBDBM50573836(CHEMBL4861375)
Affinity DataIC50: 698nMAssay Description:Inhibition of N-terminal GST-tagged human BPTF (2914 to 3037 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Fujian Medical University

Curated by ChEMBL
LigandPNGBDBM50573835(CHEMBL4872350)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of N-terminal GST-tagged human BPTF (2914 to 3037 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Fujian Medical University

Curated by ChEMBL
LigandPNGBDBM50234923(CHEMBL4069412)
Affinity DataKd:  1.70E+3nMAssay Description:Binding affinity to BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetNucleosome-remodeling factor subunit BPTF(Human)
Fujian Medical University

Curated by ChEMBL
LigandPNGBDBM50573851(CHEMBL4872422)
Affinity DataKd:  1.80E+3nMAssay Description:Binding affinity to human BPTF by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Fujian Medical University

Curated by ChEMBL
LigandPNGBDBM50573847(CHEMBL4872974)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of N-terminal GST-tagged human BPTF (2914 to 3037 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Fujian Medical University

Curated by ChEMBL
LigandPNGBDBM50157526(TCMDC-133606 | CHEMBL586426 | D3RKN_107)
Affinity DataKd:  2.80E+3nMAssay Description:Binding affinity to 5FW-labelled BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells by 19F-NMR spectraMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Fujian Medical University

Curated by ChEMBL
LigandPNGBDBM50573836(CHEMBL4861375)
Affinity DataKd:  2.81E+3nMAssay Description:Binding affinity to N-terminal GST-tagged human BPTF (2914 to 3037 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells by SPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Fujian Medical University

Curated by ChEMBL
LigandPNGBDBM50573183(CHEMBL4867912)
Affinity DataKd:  6.00E+3nMAssay Description:Binding affinity to BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetNucleosome-remodeling factor subunit BPTF(Human)
Fujian Medical University

Curated by ChEMBL
LigandPNGBDBM50573834(CHEMBL4863800)
Affinity DataIC50: 7.80E+3nMAssay Description:Inhibition of N-terminal GST-tagged human BPTF (2914 to 3037 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Fujian Medical University

Curated by ChEMBL
LigandPNGBDBM50573843(CHEMBL4875586)
Affinity DataIC50: 1.47E+4nMAssay Description:Inhibition of N-terminal GST-tagged human BPTF (2914 to 3037 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Fujian Medical University

Curated by ChEMBL
LigandPNGBDBM50571298(CHEMBL4846726)
Affinity DataKd:  1.79E+4nMAssay Description:Binding affinity to BPTF (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Fujian Medical University

Curated by ChEMBL
LigandPNGBDBM50573844(CHEMBL4873042)
Affinity DataKd:  2.07E+4nMAssay Description:Binding affinity to N-terminal GST-tagged human BPTF (2914 to 3037 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells by SPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Fujian Medical University

Curated by ChEMBL
LigandPNGBDBM25121(4-{[(7R)-8-cyclopentyl-7-ethyl-5-methyl-6-oxo-5,6,...)
Affinity DataKd:  3.70E+4nMAssay Description:Binding affinity to 5FW-labelled BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells by 19F-NMR spectraMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Fujian Medical University

Curated by ChEMBL
LigandPNGBDBM50573840(CHEMBL4860578)
Affinity DataKd:  4.96E+4nMAssay Description:Binding affinity to N-terminal GST-tagged human BPTF (2914 to 3037 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells by SPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed