Compile Data Set for Download or QSAR
Report error Found 132 Enz. Inhib. hit(s) with all data for entry = 50014724
TargetStanniocalcin-1(Mouse)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 201239BDBM201239(US9187424, 6-2)
Affinity DataIC50: 0.580nMAssay Description:Inhibition of mouse STC1 in cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
TargetStanniocalcin-1(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 201239BDBM201239(US9187424, 6-2)
Affinity DataIC50: 0.630nMAssay Description:Inhibition of human STC1 in cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50579517BDBM50579517(CHEMBL4847167)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of human recombinant MGAT2 expressed in Sf9 cell membrane using 2-monooleglycerol and [H3]-oleoyl-CoA as substrates incubated for 20 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50579517BDBM50579517(CHEMBL4847167)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of mouse recombinant MGAT2 expressed in Sf9 cell membrane using 2-oleoylglycerol and oleoyl-CoA as substrates incubated for 10 mins by LCM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 201239BDBM201239(US9187424, 6-2)
Affinity DataIC50: 2.30nMAssay Description:Inhibition of human recombinant MGAT2 expressed in Sf9 cell membrane using 2-monooleglycerol and [H3]-oleoyl-CoA as substrates incubated for 20 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 201301BDBM201301(US9187424, 77 | US9187424, 65)
Affinity DataIC50: 2.5nMAssay Description:Inhibition of human recombinant MGAT2 expressed in Sf9 cell membrane using 2-monooleglycerol and [H3]-oleoyl-CoA as substrates incubated for 20 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50579522BDBM50579522(CHEMBL4863471)
Affinity DataIC50: 2.60nMAssay Description:Inhibition of human recombinant MGAT2 expressed in Sf9 cell membrane using 2-monooleglycerol and [H3]-oleoyl-CoA as substrates incubated for 20 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50579531BDBM50579531(CHEMBL4869563)
Affinity DataIC50: 2.60nMAssay Description:Inhibition of human recombinant MGAT2 expressed in Sf9 cell membrane using 2-monooleglycerol and [H3]-oleoyl-CoA as substrates incubated for 20 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 201239BDBM201239(US9187424, 6-2)
Affinity DataIC50: 3.10nMAssay Description:Inhibition of rat recombinant MGAT2 expressed in Sf9 cell membrane using 2-oleoylglycerol and oleoyl-CoA as substrates incubated for 10 mins by LCMS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 201316BDBM201316(US9187424, 145 | US9187424, 80)
Affinity DataIC50: 3.40nMAssay Description:Inhibition of mouse recombinant MGAT2 expressed in Sf9 cell membrane using 2-oleoylglycerol and oleoyl-CoA as substrates incubated for 10 mins by LCM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 201295BDBM201295(US9187424, 59)
Affinity DataIC50: 4nMAssay Description:Inhibition of human recombinant MGAT2 expressed in Sf9 cell membrane using 2-monooleglycerol and [H3]-oleoyl-CoA as substrates incubated for 20 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50579508BDBM50579508(CHEMBL4868038)
Affinity DataIC50: 4.20nMAssay Description:Inhibition of human recombinant MGAT2 expressed in Sf9 cell membrane using 2-monooleglycerol and [H3]-oleoyl-CoA as substrates incubated for 20 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50579511BDBM50579511(CHEMBL4872250)
Affinity DataIC50: 5nMAssay Description:Inhibition of mouse recombinant MGAT2 expressed in Sf9 cell membrane using 2-oleoylglycerol and oleoyl-CoA as substrates incubated for 10 mins by LCM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50579511BDBM50579511(CHEMBL4872250)
Affinity DataIC50: 5nMAssay Description:Inhibition of human recombinant MGAT2 expressed in Sf9 cell membrane using 2-monooleglycerol and [H3]-oleoyl-CoA as substrates incubated for 20 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50579529BDBM50579529(CHEMBL4875367)
Affinity DataIC50: 5nMAssay Description:Inhibition of human recombinant MGAT2 expressed in Sf9 cell membrane using 2-monooleglycerol and [H3]-oleoyl-CoA as substrates incubated for 20 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50579522BDBM50579522(CHEMBL4863471)
Affinity DataIC50: 5.10nMAssay Description:Inhibition of mouse recombinant MGAT2 expressed in Sf9 cell membrane using 2-oleoylglycerol and oleoyl-CoA as substrates incubated for 10 mins by LCM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50579514BDBM50579514(CHEMBL4863703)
Affinity DataIC50: 5.20nMAssay Description:Inhibition of human recombinant MGAT2 expressed in Sf9 cell membrane using 2-monooleglycerol and [H3]-oleoyl-CoA as substrates incubated for 20 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 201316BDBM201316(US9187424, 145 | US9187424, 80)
Affinity DataIC50: 5.30nMAssay Description:Inhibition of human recombinant MGAT2 expressed in Sf9 cell membrane using 2-monooleglycerol and [H3]-oleoyl-CoA as substrates incubated for 20 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50579520BDBM50579520(CHEMBL4851952)
Affinity DataIC50: 5.5nMAssay Description:Inhibition of human recombinant MGAT2 expressed in Sf9 cell membrane using 2-monooleglycerol and [H3]-oleoyl-CoA as substrates incubated for 20 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50579509BDBM50579509(CHEMBL4872517)
Affinity DataIC50: 6nMAssay Description:Inhibition of mouse recombinant MGAT2 expressed in Sf9 cell membrane using 2-oleoylglycerol and oleoyl-CoA as substrates incubated for 10 mins by LCM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50579526BDBM50579526(CHEMBL4878564)
Affinity DataIC50: 6.10nMAssay Description:Inhibition of human recombinant MGAT2 expressed in Sf9 cell membrane using 2-monooleglycerol and [H3]-oleoyl-CoA as substrates incubated for 20 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50579531BDBM50579531(CHEMBL4869563)
Affinity DataIC50: 6.20nMAssay Description:Inhibition of mouse recombinant MGAT2 expressed in Sf9 cell membrane using 2-oleoylglycerol and oleoyl-CoA as substrates incubated for 10 mins by LCM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50442178BDBM50442178(CHEMBL2441600 | US9187424, 124)
Affinity DataIC50: 6.70nMAssay Description:Inhibition of human recombinant MGAT2 expressed in Sf9 cell membrane using 2-monooleglycerol and [H3]-oleoyl-CoA as substrates incubated for 20 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50579519BDBM50579519(CHEMBL3912712)
Affinity DataIC50: 7.10nMAssay Description:Inhibition of human recombinant MGAT2 expressed in Sf9 cell membrane using 2-monooleglycerol and [H3]-oleoyl-CoA as substrates incubated for 20 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50579510BDBM50579510(CHEMBL4865613)
Affinity DataIC50: 7.10nMAssay Description:Inhibition of human recombinant MGAT2 expressed in Sf9 cell membrane using 2-monooleglycerol and [H3]-oleoyl-CoA as substrates incubated for 20 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 201239BDBM201239(US9187424, 6-2)
Affinity DataIC50: 7.20nMAssay Description:Inhibition of mouse recombinant MGAT2 expressed in Sf9 cell membrane using 2-oleoylglycerol and oleoyl-CoA as substrates incubated for 10 mins by LCM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50579516BDBM50579516(CHEMBL4854178)
Affinity DataIC50: 7.30nMAssay Description:Inhibition of human recombinant MGAT2 expressed in Sf9 cell membrane using 2-monooleglycerol and [H3]-oleoyl-CoA as substrates incubated for 20 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50579526BDBM50579526(CHEMBL4878564)
Affinity DataIC50: 8.60nMAssay Description:Inhibition of rat recombinant MGAT2 expressed in Sf9 cell membrane using 2-oleoylglycerol and oleoyl-CoA as substrates incubated for 10 mins by LCMS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 201314BDBM201314(US9187424, 144 | US9187424, 78)
Affinity DataIC50: 9.90nMAssay Description:Inhibition of mouse recombinant MGAT2 expressed in Sf9 cell membrane using 2-oleoylglycerol and oleoyl-CoA as substrates incubated for 10 mins by LCM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50579509BDBM50579509(CHEMBL4872517)
Affinity DataIC50: 10nMAssay Description:Inhibition of human recombinant MGAT2 expressed in Sf9 cell membrane using 2-monooleglycerol and [H3]-oleoyl-CoA as substrates incubated for 20 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50579519BDBM50579519(CHEMBL3912712)
Affinity DataIC50: 10nMAssay Description:Inhibition of rat recombinant MGAT2 expressed in Sf9 cell membrane using 2-oleoylglycerol and oleoyl-CoA as substrates incubated for 10 mins by LCMS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50579528BDBM50579528(CHEMBL4872367)
Affinity DataIC50: 10nMAssay Description:Inhibition of human recombinant MGAT2 expressed in Sf9 cell membrane using 2-monooleglycerol and [H3]-oleoyl-CoA as substrates incubated for 20 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 201269BDBM201269(US9187424, 76 | US9187424, 269 | US9187424, 53 | U...)
Affinity DataIC50: 12nMAssay Description:Inhibition of human recombinant MGAT2 expressed in Sf9 cell membrane using 2-monooleglycerol and [H3]-oleoyl-CoA as substrates incubated for 20 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50579508BDBM50579508(CHEMBL4868038)
Affinity DataIC50: 12nMAssay Description:Inhibition of mouse recombinant MGAT2 expressed in Sf9 cell membrane using 2-oleoylglycerol and oleoyl-CoA as substrates incubated for 10 mins by LCM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50579526BDBM50579526(CHEMBL4878564)
Affinity DataIC50: 12nMAssay Description:Inhibition of mouse recombinant MGAT2 expressed in Sf9 cell membrane using 2-oleoylglycerol and oleoyl-CoA as substrates incubated for 10 mins by LCM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 201271BDBM201271(US9187424, 35)
Affinity DataIC50: 13nMAssay Description:Inhibition of human recombinant MGAT2 expressed in Sf9 cell membrane using 2-monooleglycerol and [H3]-oleoyl-CoA as substrates incubated for 20 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
TargetStanniocalcin-1(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50579526BDBM50579526(CHEMBL4878564)
Affinity DataIC50: 13nMAssay Description:Inhibition of human STC1 in cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 201314BDBM201314(US9187424, 144 | US9187424, 78)
Affinity DataIC50: 14nMAssay Description:Inhibition of human recombinant MGAT2 expressed in Sf9 cell membrane using 2-monooleglycerol and [H3]-oleoyl-CoA as substrates incubated for 20 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 201273BDBM201273(US9187424, 37)
Affinity DataIC50: 15nMAssay Description:Inhibition of human recombinant MGAT2 expressed in Sf9 cell membrane using 2-monooleglycerol and [H3]-oleoyl-CoA as substrates incubated for 20 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 201293BDBM201293(US9187424, 57)
Affinity DataIC50: 16nMAssay Description:Inhibition of human recombinant MGAT2 expressed in Sf9 cell membrane using 2-monooleglycerol and [H3]-oleoyl-CoA as substrates incubated for 20 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50442178BDBM50442178(CHEMBL2441600 | US9187424, 124)
Affinity DataIC50: 17nMAssay Description:Inhibition of mouse recombinant MGAT2 expressed in Sf9 cell membrane using 2-oleoylglycerol and oleoyl-CoA as substrates incubated for 10 mins by LCM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50579529BDBM50579529(CHEMBL4875367)
Affinity DataIC50: 18nMAssay Description:Inhibition of mouse recombinant MGAT2 expressed in Sf9 cell membrane using 2-oleoylglycerol and oleoyl-CoA as substrates incubated for 10 mins by LCM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50579519BDBM50579519(CHEMBL3912712)
Affinity DataIC50: 18nMAssay Description:Inhibition of mouse recombinant MGAT2 expressed in Sf9 cell membrane using 2-oleoylglycerol and oleoyl-CoA as substrates incubated for 10 mins by LCM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 201307BDBM201307(US9187424, 71)
Affinity DataIC50: 18nMAssay Description:Inhibition of mouse recombinant MGAT2 expressed in Sf9 cell membrane using 2-oleoylglycerol and oleoyl-CoA as substrates incubated for 10 mins by LCM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 201301BDBM201301(US9187424, 77 | US9187424, 65)
Affinity DataIC50: 20nMAssay Description:Inhibition of mouse recombinant MGAT2 expressed in Sf9 cell membrane using 2-oleoylglycerol and oleoyl-CoA as substrates incubated for 10 mins by LCM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
TargetStanniocalcin-1(Mouse)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50579526BDBM50579526(CHEMBL4878564)
Affinity DataIC50: 20nMAssay Description:Inhibition of mouse STC1 in cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 201237BDBM201237(US9187424, 5)
Affinity DataIC50: 21nMAssay Description:Inhibition of human recombinant MGAT2 expressed in Sf9 cell membrane using 2-monooleglycerol and [H3]-oleoyl-CoA as substrates incubated for 20 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50579515BDBM50579515(CHEMBL4865861)
Affinity DataIC50: 21nMAssay Description:Inhibition of human recombinant MGAT2 expressed in Sf9 cell membrane using 2-monooleglycerol and [H3]-oleoyl-CoA as substrates incubated for 20 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50579528BDBM50579528(CHEMBL4872367)
Affinity DataIC50: 22nMAssay Description:Inhibition of mouse recombinant MGAT2 expressed in Sf9 cell membrane using 2-oleoylglycerol and oleoyl-CoA as substrates incubated for 10 mins by LCM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50579521BDBM50579521(CHEMBL4862212)
Affinity DataIC50: 23nMAssay Description:Inhibition of mouse recombinant MGAT2 expressed in Sf9 cell membrane using 2-oleoylglycerol and oleoyl-CoA as substrates incubated for 10 mins by LCM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
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