Compile Data Set for Download or QSAR
Report error Found 41 Enz. Inhib. hit(s) with all data for entry = 50016611
TargetSerine/threonine-protein kinase PLK1(Human)
University of South Carolina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50596070BDBM50596070(CHEMBL5180726)
Affinity DataEC50:  820nMAssay Description:Binding affinity to full length PLK1 in human PC-3 cells assessed as stabilized protein incubated for 2 hrs followed by aggregation temperature at 56...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK3(Human)
University of South Carolina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50596069BDBM50596069(CHEMBL5175899)
Affinity DataIC50: 2.00E+3nMAssay Description:Binding affinity to recombinant human N-terminal MBP tagged/C-terminal His-tagged human PLK3-PBD (335 to 646 residue) expressed in Escherichia coli e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
University of South Carolina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50596070BDBM50596070(CHEMBL5180726)
Affinity DataIC50: 2.20E+3nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged PLK1-PBD (367 to 603 end residue) expressed in Escherichia coli using MAGPMQS[pT]PLNGAKK ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
University of South Carolina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50596072BDBM50596072(CHEMBL5209469)
Affinity DataIC50: 4.00E+3nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged PLK1-PBD (367 to 603 end residue) expressed in Escherichia coli using MAGPMQS[pT]PLNGAKK ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
University of South Carolina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50596071BDBM50596071(CHEMBL5179948)
Affinity DataIC50: 5.90E+3nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged PLK1-PBD (367 to 603 end residue) expressed in Escherichia coli using MAGPMQS[pT]PLNGAKK ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
University of South Carolina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50596069BDBM50596069(CHEMBL5175899)
Affinity DataIC50: 6.00E+3nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged PLK1-PBD (367 to 603 end residue) expressed in Escherichia coli using MAGPMQS[pT]PLNGAKK ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
University of South Carolina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50596080BDBM50596080(CHEMBL5182503)
Affinity DataIC50: 6.10E+3nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged PLK1-PBD (367 to 603 end residue) expressed in Escherichia coli using MAGPMQS[pT]PLNGAKK ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK3(Human)
University of South Carolina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50596070BDBM50596070(CHEMBL5180726)
Affinity DataEC50:  6.90E+3nMAssay Description:Binding affinity to full length PLK3 in human PC-3 cells assessed as stabilized protein incubated for 2 hrs followed by aggregation temperature at 48...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK3(Human)
University of South Carolina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50596072BDBM50596072(CHEMBL5209469)
Affinity DataIC50: 7.40E+3nMAssay Description:Binding affinity to recombinant human N-terminal MBP tagged/C-terminal His-tagged human PLK3-PBD (335 to 646 residue) expressed in Escherichia coli e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK3(Human)
University of South Carolina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50596070BDBM50596070(CHEMBL5180726)
Affinity DataIC50: 7.70E+3nMAssay Description:Binding affinity to recombinant human N-terminal MBP tagged/C-terminal His-tagged human PLK3-PBD (335 to 646 residue) expressed in Escherichia coli e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
University of South Carolina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50596082BDBM50596082(CHEMBL5183471)
Affinity DataIC50: 7.90E+3nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged PLK1-PBD (367 to 603 end residue) expressed in Escherichia coli using MAGPMQS[pT]PLNGAKK ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
University of South Carolina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50596086BDBM50596086(CHEMBL5173820)
Affinity DataIC50: 9.80E+3nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged PLK1-PBD (367 to 603 end residue) expressed in Escherichia coli using MAGPMQS[pT]PLNGAKK ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK3(Human)
University of South Carolina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50596080BDBM50596080(CHEMBL5182503)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to recombinant human N-terminal MBP tagged/C-terminal His-tagged human PLK3-PBD (335 to 646 residue) expressed in Escherichia coli e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
University of South Carolina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50596078BDBM50596078(CHEMBL5183088)
Affinity DataIC50: 1.11E+4nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged PLK1-PBD (367 to 603 end residue) expressed in Escherichia coli using MAGPMQS[pT]PLNGAKK ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
University of South Carolina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50596068BDBM50596068(CHEMBL5178208)
Affinity DataIC50: 1.13E+4nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged PLK1-PBD (367 to 603 end residue) expressed in Escherichia coli using MAGPMQS[pT]PLNGAKK ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
University of South Carolina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50596084BDBM50596084(CHEMBL5173392)
Affinity DataIC50: 1.20E+4nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged PLK1-PBD (367 to 603 end residue) expressed in Escherichia coli using MAGPMQS[pT]PLNGAKK ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK3(Human)
University of South Carolina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50596082BDBM50596082(CHEMBL5183471)
Affinity DataIC50: 1.21E+4nMAssay Description:Binding affinity to recombinant human N-terminal MBP tagged/C-terminal His-tagged human PLK3-PBD (335 to 646 residue) expressed in Escherichia coli e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK3(Human)
University of South Carolina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50596078BDBM50596078(CHEMBL5183088)
Affinity DataIC50: 1.32E+4nMAssay Description:Binding affinity to recombinant human N-terminal MBP tagged/C-terminal His-tagged human PLK3-PBD (335 to 646 residue) expressed in Escherichia coli e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK3(Human)
University of South Carolina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50596071BDBM50596071(CHEMBL5179948)
Affinity DataIC50: 1.36E+4nMAssay Description:Binding affinity to recombinant human N-terminal MBP tagged/C-terminal His-tagged human PLK3-PBD (335 to 646 residue) expressed in Escherichia coli e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK3(Human)
University of South Carolina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50596068BDBM50596068(CHEMBL5178208)
Affinity DataIC50: 1.55E+4nMAssay Description:Binding affinity to recombinant human N-terminal MBP tagged/C-terminal His-tagged human PLK3-PBD (335 to 646 residue) expressed in Escherichia coli e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK3(Human)
University of South Carolina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50581994BDBM50581994(CHEMBL5087960)
Affinity DataIC50: 1.80E+4nMAssay Description:Binding affinity to recombinant human N-terminal MBP tagged/C-terminal His-tagged human PLK3-PBD (335 to 646 residue) expressed in Escherichia coli e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
University of South Carolina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50581994BDBM50581994(CHEMBL5087960)
Affinity DataIC50: 1.84E+4nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged PLK1-PBD (367 to 603 end residue) expressed in Escherichia coli using MAGPMQS[pT]PLNGAKK ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
University of South Carolina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50596091BDBM50596091(CHEMBL5195887)
Affinity DataIC50: 1.88E+4nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged PLK1-PBD (367 to 603 end residue) expressed in Escherichia coli using MAGPMQS[pT]PLNGAKK ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
University of South Carolina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50596089BDBM50596089(CHEMBL5196414)
Affinity DataIC50: 2.17E+4nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged PLK1-PBD (367 to 603 end residue) expressed in Escherichia coli using MAGPMQS[pT]PLNGAKK ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK3(Human)
University of South Carolina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50596081BDBM50596081(CHEMBL5204555)
Affinity DataIC50: 2.29E+4nMAssay Description:Binding affinity to recombinant human N-terminal MBP tagged/C-terminal His-tagged human PLK3-PBD (335 to 646 residue) expressed in Escherichia coli e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
University of South Carolina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50596085BDBM50596085(CHEMBL5207741)
Affinity DataIC50: 2.53E+4nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged PLK1-PBD (367 to 603 end residue) expressed in Escherichia coli using MAGPMQS[pT]PLNGAKK ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
University of South Carolina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50596081BDBM50596081(CHEMBL5204555)
Affinity DataIC50: 2.94E+4nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged PLK1-PBD (367 to 603 end residue) expressed in Escherichia coli using MAGPMQS[pT]PLNGAKK ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
University of South Carolina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50596083BDBM50596083(CHEMBL5181122)
Affinity DataIC50: 2.96E+4nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged PLK1-PBD (367 to 603 end residue) expressed in Escherichia coli using MAGPMQS[pT]PLNGAKK ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
University of South Carolina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50596079BDBM50596079(CHEMBL5190849)
Affinity DataIC50: 3.06E+4nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged PLK1-PBD (367 to 603 end residue) expressed in Escherichia coli using MAGPMQS[pT]PLNGAKK ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK3(Human)
University of South Carolina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50596079BDBM50596079(CHEMBL5190849)
Affinity DataIC50: 3.97E+4nMAssay Description:Binding affinity to recombinant human N-terminal MBP tagged/C-terminal His-tagged human PLK3-PBD (335 to 646 residue) expressed in Escherichia coli e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
University of South Carolina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50596077BDBM50596077(CHEMBL5206566)
Affinity DataIC50: 9.83E+4nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged PLK1-PBD (367 to 603 end residue) expressed in Escherichia coli using MAGPMQS[pT]PLNGAKK ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
University of South Carolina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50596090BDBM50596090(CHEMBL5169598)
Affinity DataIC50: 1.18E+5nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged PLK1-PBD (367 to 603 end residue) expressed in Escherichia coli using MAGPMQS[pT]PLNGAKK ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
University of South Carolina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50596067BDBM50596067(CHEMBL4864977)
Affinity DataIC50: 2.24E+5nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged PLK1-PBD (367 to 603 end residue) expressed in Escherichia coli using MAGPMQS[pT]PLNGAKK ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
University of South Carolina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50596076BDBM50596076(CHEMBL5178482)
Affinity DataIC50: 2.59E+5nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged PLK1-PBD (367 to 603 end residue) expressed in Escherichia coli using MAGPMQS[pT]PLNGAKK ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
University of South Carolina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50596088BDBM50596088(CHEMBL5174046)
Affinity DataIC50: 6.00E+5nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged PLK1-PBD (367 to 603 end residue) expressed in Escherichia coli using MAGPMQS[pT]PLNGAKK ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
University of South Carolina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50596087BDBM50596087(CHEMBL5176465)
Affinity DataIC50: 6.00E+5nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged PLK1-PBD (367 to 603 end residue) expressed in Escherichia coli using MAGPMQS[pT]PLNGAKK ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
University of South Carolina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50596074BDBM50596074(CHEMBL5178662)
Affinity DataIC50: 6.00E+5nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged PLK1-PBD (367 to 603 end residue) expressed in Escherichia coli using MAGPMQS[pT]PLNGAKK ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
University of South Carolina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50596073BDBM50596073(CHEMBL5202121)
Affinity DataIC50: 6.00E+5nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged PLK1-PBD (367 to 603 end residue) expressed in Escherichia coli using MAGPMQS[pT]PLNGAKK ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
University of South Carolina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50596092BDBM50596092(CHEMBL5175885)
Affinity DataIC50: 6.00E+5nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged PLK1-PBD (367 to 603 end residue) expressed in Escherichia coli using MAGPMQS[pT]PLNGAKK ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
University of South Carolina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50596075BDBM50596075(CHEMBL5177850)
Affinity DataIC50: 6.00E+5nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged PLK1-PBD (367 to 603 end residue) expressed in Escherichia coli using MAGPMQS[pT]PLNGAKK ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
University of South Carolina

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50596066BDBM50596066(CHEMBL5185527)
Affinity DataIC50: 6.00E+5nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged PLK1-PBD (367 to 603 end residue) expressed in Escherichia coli using MAGPMQS[pT]PLNGAKK ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed