Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50014736
TargetArginase-1(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50579614BDBM50579614(CHEMBL4871970)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of ARG1 (unknown origin) assessed as reduction in thio-ornithine production using thioarginine as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
TargetArginase-1(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50579610BDBM50579610(CHEMBL4873520)
Affinity DataIC50: 2.20nMAssay Description:Inhibition of ARG1 (unknown origin) assessed as reduction in thio-ornithine production using thioarginine as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
TargetArginase-1(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50579616BDBM50579616(CHEMBL4845730)
Affinity DataIC50: 3.20nMAssay Description:Inhibition of ARG1 (unknown origin) assessed as reduction in thio-ornithine production using thioarginine as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
TargetArginase-1(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50579611BDBM50579611(CHEMBL4871097)
Affinity DataIC50: 3.90nMAssay Description:Inhibition of ARG1 (unknown origin) assessed as reduction in thio-ornithine production using thioarginine as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
TargetArginase-1(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50579615BDBM50579615(CHEMBL4865209)
Affinity DataIC50: 5nMAssay Description:Inhibition of ARG1 (unknown origin) assessed as reduction in thio-ornithine production using thioarginine as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
TargetArginase-1(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50577458BDBM50577458(CHEMBL4858437)
Affinity DataIC50: 16nMAssay Description:Inhibition of ARG1 (unknown origin) assessed as reduction in thio-ornithine production using thioarginine as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
TargetArginase-1(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50579613BDBM50579613(CHEMBL4850423)
Affinity DataIC50: 25nMAssay Description:Inhibition of ARG1 (unknown origin) assessed as reduction in thio-ornithine production using thioarginine as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
TargetArginase-1(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50579609BDBM50579609(CHEMBL4872874)
Affinity DataIC50: 46nMAssay Description:Inhibition of ARG1 (unknown origin) assessed as reduction in thio-ornithine production using thioarginine as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
TargetArginase-1(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50579618BDBM50579618(CHEMBL4871090)
Affinity DataIC50: 67nMAssay Description:Inhibition of ARG1 (unknown origin) assessed as reduction in thio-ornithine production using thioarginine as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
TargetArginase-1(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50579612BDBM50579612(CHEMBL4847500)
Affinity DataIC50: 104nMAssay Description:Inhibition of ARG1 (unknown origin) assessed as reduction in thio-ornithine production using thioarginine as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
TargetArginase-1(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50579608BDBM50579608(CHEMBL4849969)
Affinity DataIC50: 370nMAssay Description:Inhibition of ARG1 (unknown origin) assessed as reduction in thio-ornithine production using thioarginine as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
TargetArginase-1(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50579617BDBM50579617(CHEMBL4863411)
Affinity DataIC50: 5.74E+3nMAssay Description:Inhibition of ARG1 (unknown origin) assessed as reduction in thio-ornithine production using thioarginine as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
TargetArginase-1(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50579607BDBM50579607(CHEMBL4865167)
Affinity DataIC50: 8.78E+3nMAssay Description:Inhibition of ARG1 (unknown origin) assessed as reduction in thio-ornithine production using thioarginine as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
TargetArginase-1(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50579606BDBM50579606(CHEMBL4851004)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of ARG1 (unknown origin) assessed as reduction in thio-ornithine production using thioarginine as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed