Compile Data Set for Download or QSAR
Report error Found 102 Enz. Inhib. hit(s) with all data for entry = 50015271
TargetKelch-like ECH-associated protein 1(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584857(CHEMBL5089816)
Affinity DataKd:  27nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based direct binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584856(CHEMBL5078020)
Affinity DataKd:  29nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584861(CHEMBL5082511)
Affinity DataKd:  29nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584857(CHEMBL5089816)
Affinity DataKd:  29nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584860(CHEMBL5077539)
Affinity DataKd:  33nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584859(CHEMBL5070465)
Affinity DataKd:  36nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584862(CHEMBL5087851)
Affinity DataKd:  37nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584822(CHEMBL5092602)
Affinity DataKd:  41nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584858(CHEMBL5070545)
Affinity DataKd:  43nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584851(CHEMBL5091126)
Affinity DataKd:  44nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584851(CHEMBL5091126)
Affinity DataKd:  46nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584858(CHEMBL5070545)
Affinity DataKd:  49nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based direct binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584822(CHEMBL5092602)
Affinity DataKd:  68nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584860(CHEMBL5077539)
Affinity DataKd:  85nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based direct binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584856(CHEMBL5078020)
Affinity DataKd:  97nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based direct binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584861(CHEMBL5082511)
Affinity DataKd:  102nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based direct binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584859(CHEMBL5070465)
Affinity DataKd:  132nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based direct binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584862(CHEMBL5087851)
Affinity DataKd:  152nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based direct binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584852(CHEMBL5092330)
Affinity DataKd:  383nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584852(CHEMBL5092330)
Affinity DataKd:  758nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584832(CHEMBL5076271)
Affinity DataKd:  780nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584845(CHEMBL5082765)
Affinity DataKd:  890nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584848(CHEMBL5090388)
Affinity DataKd:  890nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584823(CHEMBL5075717)
Affinity DataKd:  910nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584826(CHEMBL5090939)
Affinity DataKd:  1.00E+3nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584786(CHEMBL5089493)
Affinity DataKd:  1.00E+3nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584845(CHEMBL5082765)
Affinity DataKd:  1.10E+3nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584824(CHEMBL5080665)
Affinity DataKd:  1.40E+3nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetKelch-like ECH-associated protein 1(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584831(CHEMBL5092331)
Affinity DataKd:  1.50E+3nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584788(CHEMBL5094633)
Affinity DataKd:  1.60E+3nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584826(CHEMBL5090939)
Affinity DataKd:  1.70E+3nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584827(CHEMBL5082071)
Affinity DataKd:  2.20E+3nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584823(CHEMBL5075717)
Affinity DataKd:  2.40E+3nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584828(CHEMBL5093123)
Affinity DataKd:  2.60E+3nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584832(CHEMBL5076271)
Affinity DataKd:  2.80E+3nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584848(CHEMBL5090388)
Affinity DataKd:  2.80E+3nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584786(CHEMBL5089493)
Affinity DataKd:  3.00E+3nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584829(CHEMBL5086087)
Affinity DataKd:  3.40E+3nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50556867(CHEMBL4757224)
Affinity DataKd:  3.70E+3nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584788(CHEMBL5094633)
Affinity DataKd:  4.10E+3nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584787(CHEMBL5087800)
Affinity DataKd:  4.10E+3nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50556867(CHEMBL4757224)
Affinity DataKd:  4.10E+3nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584824(CHEMBL5080665)
Affinity DataKd:  4.70E+3nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetKelch-like ECH-associated protein 1(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584834(CHEMBL5075129)
Affinity DataKd:  6.00E+3nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584837(CHEMBL5071662)
Affinity DataKd:  6.40E+3nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584833(CHEMBL5076972)
Affinity DataKd:  7.00E+3nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584840(CHEMBL5078448)
Affinity DataKd:  7.10E+3nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584827(CHEMBL5082071)
Affinity DataKd:  7.30E+3nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584841(CHEMBL5078849)
Affinity DataKd:  7.40E+3nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584838(CHEMBL5079382)
Affinity DataKd:  7.50E+3nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
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