Compile Data Set for Download or QSAR
Report error Found 43 Enz. Inhib. hit(s) with all data for entry = 50017733
TargetSerine-protein kinase ATM(Human)
Eberhard Karls Universit£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 245474BDBM245474(US9428503, 1)
Affinity DataIC50: 0.220nMAssay Description:Inhibition of ATM in human A549 cells assessed as reduction in etoposide-stimulated KAP1 phosphorylation by In-Cell-Western assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine-protein kinase ATM(Human)
Eberhard Karls Universit£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50604534BDBM50604534(CHEMBL5191923 | US20230348462, Example 50)
Affinity DataIC50: 0.320nMAssay Description:Inhibition of ATM in human A549 cells assessed as reduction in etoposide-stimulated KAP1 phosphorylation by In-Cell-Western assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine-protein kinase ATM(Human)
Eberhard Karls Universit£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50604528BDBM50604528(CHEMBL5183158 | US20230348462, Example 27)
Affinity DataIC50: 0.650nMAssay Description:Inhibition of ATM in human A549 cells assessed as reduction in etoposide-stimulated KAP1 phosphorylation by In-Cell-Western assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine-protein kinase ATM(Human)
Eberhard Karls Universit£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50604529BDBM50604529(CHEMBL5181829 | US20230348462, Example 28)
Affinity DataIC50: 0.710nMAssay Description:Inhibition of ATM in human A549 cells assessed as reduction in etoposide-stimulated KAP1 phosphorylation by In-Cell-Western assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine-protein kinase ATM(Human)
Eberhard Karls Universit£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50604533BDBM50604533(CHEMBL5170132 | US20230348462, Example 49)
Affinity DataIC50: 0.920nMAssay Description:Inhibition of ATM in human A549 cells assessed as reduction in etoposide-stimulated KAP1 phosphorylation by In-Cell-Western assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine-protein kinase ATM(Human)
Eberhard Karls Universit£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50604528BDBM50604528(CHEMBL5183158 | US20230348462, Example 27)
Affinity DataIC50: 1nMAssay Description:Inhibition of ATM (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine-protein kinase ATM(Human)
Eberhard Karls Universit£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50604529BDBM50604529(CHEMBL5181829 | US20230348462, Example 28)
Affinity DataIC50: 1nMAssay Description:Inhibition of ATM (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine-protein kinase ATM(Human)
Eberhard Karls Universit£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50604534BDBM50604534(CHEMBL5191923 | US20230348462, Example 50)
Affinity DataIC50: 1nMAssay Description:Inhibition of ATM (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine-protein kinase ATM(Human)
Eberhard Karls Universit£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50604502BDBM50604502(CHEMBL5203201 | US20230348462, Example 7)
Affinity DataIC50: 1nMAssay Description:Inhibition of ATM (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine-protein kinase ATM(Human)
Eberhard Karls Universit£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50604533BDBM50604533(CHEMBL5170132 | US20230348462, Example 49)
Affinity DataIC50: 1nMAssay Description:Inhibition of ATM (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine-protein kinase ATM(Human)
Eberhard Karls Universit£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 245474BDBM245474(US9428503, 1)
Affinity DataIC50: 1nMAssay Description:Inhibition of ATM (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine-protein kinase ATM(Human)
Eberhard Karls Universit£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50604504BDBM50604504(CHEMBL5184135 | US20230348462, Example 10)
Affinity DataIC50: 1nMAssay Description:Inhibition of ATM (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine-protein kinase ATM(Human)
Eberhard Karls Universit£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50604535BDBM50604535(CHEMBL5198342 | US20230348462, Example 51)
Affinity DataIC50: 1nMAssay Description:Inhibition of ATM (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine-protein kinase ATM(Human)
Eberhard Karls Universit£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50604506BDBM50604506(CHEMBL5179355 | US20230348462, Example 21)
Affinity DataIC50: 1nMAssay Description:Inhibition of ATM (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine-protein kinase ATM(Human)
Eberhard Karls Universit£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50604505BDBM50604505(CHEMBL5171246 | US20230348462, Example 11)
Affinity DataIC50: 1nMAssay Description:Inhibition of ATM (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine-protein kinase ATM(Human)
Eberhard Karls Universit£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50604508BDBM50604508(CHEMBL5204162 | US20230348462, Example 17)
Affinity DataIC50: 1nMAssay Description:Inhibition of ATM (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine-protein kinase ATM(Human)
Eberhard Karls Universit£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50604507BDBM50604507(CHEMBL5204408 | US20230348462, Example 19)
Affinity DataIC50: 1nMAssay Description:Inhibition of ATM (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine-protein kinase ATM(Human)
Eberhard Karls Universit£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50604510BDBM50604510(CHEMBL5209108 | US20230348462, Example 15)
Affinity DataIC50: 1nMAssay Description:Inhibition of ATM (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine-protein kinase ATM(Human)
Eberhard Karls Universit£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50604512BDBM50604512(CHEMBL5207887)
Affinity DataIC50: 1nMAssay Description:Inhibition of ATM (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine-protein kinase ATM(Human)
Eberhard Karls Universit£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50604511BDBM50604511(CHEMBL5199423 | US20230348462, Example 16)
Affinity DataIC50: 1nMAssay Description:Inhibition of ATM (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine-protein kinase ATM(Human)
Eberhard Karls Universit£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50604513BDBM50604513(CHEMBL5191914)
Affinity DataIC50: 1nMAssay Description:Inhibition of ATM (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine-protein kinase ATM(Human)
Eberhard Karls Universit£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50604513BDBM50604513(CHEMBL5191914)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of ATM in human A549 cells assessed as reduction in etoposide-stimulated KAP1 phosphorylation by In-Cell-Western assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine-protein kinase ATM(Human)
Eberhard Karls Universit£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50604505BDBM50604505(CHEMBL5171246 | US20230348462, Example 11)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of ATM in human A549 cells assessed as reduction in etoposide-stimulated KAP1 phosphorylation by In-Cell-Western assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine-protein kinase ATM(Human)
Eberhard Karls Universit£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50604503BDBM50604503(CHEMBL5201821 | US20230348462, Example 8)
Affinity DataIC50: 2nMAssay Description:Inhibition of ATM (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine-protein kinase ATM(Human)
Eberhard Karls Universit£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50604521BDBM50604521(CHEMBL5195854 | US20230348462, Example 13)
Affinity DataIC50: 2nMAssay Description:Inhibition of ATM (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine-protein kinase ATM(Human)
Eberhard Karls Universit£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50604530BDBM50604530(CHEMBL5179580 | US20230348462, Example 46)
Affinity DataIC50: 3nMAssay Description:Inhibition of ATM (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine-protein kinase ATM(Human)
Eberhard Karls Universit£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50604535BDBM50604535(CHEMBL5198342 | US20230348462, Example 51)
Affinity DataIC50: 3.30nMAssay Description:Inhibition of ATM in human A549 cells assessed as reduction in etoposide-stimulated KAP1 phosphorylation by In-Cell-Western assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine-protein kinase ATM(Human)
Eberhard Karls Universit£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50604518BDBM50604518(CHEMBL5209089 | US20230348462, Example 26)
Affinity DataIC50: 4nMAssay Description:Inhibition of ATM (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine-protein kinase ATM(Human)
Eberhard Karls Universit£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50604509BDBM50604509(CHEMBL5172175 | US20230348462, Example 18)
Affinity DataIC50: 4nMAssay Description:Inhibition of ATM (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine-protein kinase ATM(Human)
Eberhard Karls Universit£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50604519BDBM50604519(CHEMBL5171104 | US20230348462, Example 25)
Affinity DataIC50: 7nMAssay Description:Inhibition of ATM (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine-protein kinase ATM(Human)
Eberhard Karls Universit£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50604522BDBM50604522(CHEMBL5175636)
Affinity DataIC50: 16nMAssay Description:Inhibition of ATM (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine-protein kinase ATM(Human)
Eberhard Karls Universit£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50604515BDBM50604515(CHEMBL5195925)
Affinity DataIC50: 25nMAssay Description:Inhibition of ATM (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine-protein kinase ATM(Human)
Eberhard Karls Universit£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50604531BDBM50604531(CHEMBL5181690)
Affinity DataIC50: 32nMAssay Description:Inhibition of ATM (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine-protein kinase ATM(Human)
Eberhard Karls Universit£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50604532BDBM50604532(CHEMBL5189299)
Affinity DataIC50: 37nMAssay Description:Inhibition of ATM (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine-protein kinase ATM(Human)
Eberhard Karls Universit£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50604514BDBM50604514(CHEMBL5193567)
Affinity DataIC50: 78nMAssay Description:Inhibition of ATM (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine-protein kinase ATM(Human)
Eberhard Karls Universit£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50604523BDBM50604523(CHEMBL5200163)
Affinity DataIC50: 101nMAssay Description:Inhibition of ATM (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine-protein kinase ATM(Human)
Eberhard Karls Universit£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50604517BDBM50604517(CHEMBL5191601)
Affinity DataIC50: 158nMAssay Description:Inhibition of ATM (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine-protein kinase ATM(Human)
Eberhard Karls Universit£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50604516BDBM50604516(CHEMBL5206081)
Affinity DataIC50: 159nMAssay Description:Inhibition of ATM (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine-protein kinase ATM(Human)
Eberhard Karls Universit£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50604525BDBM50604525(CHEMBL5207735)
Affinity DataIC50: 212nMAssay Description:Inhibition of ATM (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine-protein kinase ATM(Human)
Eberhard Karls Universit£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50604524BDBM50604524(CHEMBL5200256)
Affinity DataIC50: 394nMAssay Description:Inhibition of ATM (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine-protein kinase ATM(Human)
Eberhard Karls Universit£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50604526BDBM50604526(CHEMBL5200053)
Affinity DataIC50: 885nMAssay Description:Inhibition of ATM (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine-protein kinase ATM(Human)
Eberhard Karls Universit£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50604520BDBM50604520(CHEMBL5171662)
Affinity DataIC50: 945nMAssay Description:Inhibition of ATM (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine-protein kinase ATM(Human)
Eberhard Karls Universit£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50604527BDBM50604527(CHEMBL5206686)
Affinity DataIC50: 1.58E+3nMAssay Description:Inhibition of ATM (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed