Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 50017867
TargetNuclear receptor subfamily 5 group A member 2(Human)
Emory University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50605641(CHEMBL5177743)
Affinity DataKi:  0.150nMAssay Description:Binding affinity to N-terminal 6-His tagged human LRH-1 LBD (299 to 541 residues) expressed in Escherichia coli BL21-(DE3) assessed as inhibition con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
Emory University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50511467(CHEMBL4551205)
Affinity DataKi:  1.30nMAssay Description:Binding affinity to N-terminal 6-His tagged human LRH-1 LBD (299 to 541 residues) expressed in Escherichia coli BL21-(DE3) assessed as inhibition con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
Emory University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50605640(CHEMBL5198453)
Affinity DataKi:  5.30nMAssay Description:Binding affinity to N-terminal 6-His tagged human LRH-1 LBD (299 to 541 residues) expressed in Escherichia coli BL21-(DE3) assessed as inhibition con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
Emory University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50605641(CHEMBL5177743)
Affinity DataEC50:  43nMAssay Description:Agonist activity at LRH-1 (unknown origin) transfected in human HeLa cells measured after 24 hrs by Dual Glo luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
Emory University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50511467(CHEMBL4551205)
Affinity DataEC50:  100nMAssay Description:Agonist activity at LRH-1 (unknown origin) transfected in human HeLa cells measured after 24 hrs by Dual Glo luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
Emory University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50605641(CHEMBL5177743)
Affinity DataKd:  120nMAssay Description:Binding affinity to N-terminal 6-His tagged human LRH-1 LBD (299 to 541 residues) expressed in Escherichia coli BL21-(DE3) assessed as dissociation c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
Emory University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50511467(CHEMBL4551205)
Affinity DataKd:  320nMAssay Description:Binding affinity to N-terminal 6-His tagged human LRH-1 LBD (299 to 541 residues) expressed in Escherichia coli BL21-(DE3) assessed as dissociation c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
Emory University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50605640(CHEMBL5198453)
Affinity DataKd:  340nMAssay Description:Binding affinity to N-terminal 6-His tagged human LRH-1 LBD (299 to 541 residues) expressed in Escherichia coli BL21-(DE3) assessed as dissociation c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
Emory University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50605641(CHEMBL5177743)
Affinity DataKd:  340nMAssay Description:Binding affinity to N-terminal 6-His tagged human LRH-1 LBD (299 to 541 residues) expressed in Escherichia coli BL21-(DE3) assessed as dissociation c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
Emory University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50511467(CHEMBL4551205)
Affinity DataKd:  620nMAssay Description:Binding affinity to N-terminal 6-His tagged human LRH-1 LBD (299 to 541 residues) expressed in Escherichia coli BL21-(DE3) assessed as dissociation c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
Emory University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50605640(CHEMBL5198453)
Affinity DataKd:  720nMAssay Description:Binding affinity to N-terminal 6-His tagged human LRH-1 LBD (299 to 541 residues) expressed in Escherichia coli BL21-(DE3) assessed as dissociation c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
Emory University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50605640(CHEMBL5198453)
Affinity DataEC50:  1.70E+3nMAssay Description:Agonist activity at LRH-1 (unknown origin) transfected in human HeLa cells measured after 24 hrs by Dual Glo luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
Emory University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50605641(CHEMBL5177743)
Affinity DataKd:  1.80E+3nMAssay Description:Binding affinity to N-terminal 6-His tagged human LRH-1 LBD (299 to 541 residues) expressed in Escherichia coli BL21-(DE3) assessed as dissociation c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
Emory University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50511467(CHEMBL4551205)
Affinity DataKd:  2.10E+3nMAssay Description:Binding affinity to N-terminal 6-His tagged human LRH-1 LBD (299 to 541 residues) expressed in Escherichia coli BL21-(DE3) assessed as dissociation c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
Emory University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50605640(CHEMBL5198453)
Affinity DataKd:  2.50E+3nMAssay Description:Binding affinity to N-terminal 6-His tagged human LRH-1 LBD (299 to 541 residues) expressed in Escherichia coli BL21-(DE3) assessed as dissociation c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed