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Found 79 Enz. Inhib. hit(s) with all data for entry = 50016073
TargetAurora kinase A(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50004205(MK-045 | MK-0457 | TOZASERTIB | US9249124, VX680 |...)
Affinity DataKi:  0.650nMAssay Description:Inhibition of Aurora A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAurora kinase B(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50004205(MK-045 | MK-0457 | TOZASERTIB | US9249124, VX680 |...)
Affinity DataKi:  3.40nMAssay Description:Inhibition of Aurora B (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAurora kinase C(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50004205(MK-045 | MK-0457 | TOZASERTIB | US9249124, VX680 |...)
Affinity DataKi:  4.60nMAssay Description:Inhibition of Aurora C (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50004205(MK-045 | MK-0457 | TOZASERTIB | US9249124, VX680 |...)
Affinity DataKi:  7.70nMAssay Description:Inhibition of PLK4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50591934(CHEMBL5209160)
Affinity DataIC50:  0.100nMAssay Description:Inhibition of recombinant human PLK4 incubated for 60 mins by Lanthascreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50591949(CHEMBL5185001)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of recombinant human PLK4 incubated for 60 mins by Lanthascreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50591932(CHEMBL5171469)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of recombinant human PLK4 incubated for 60 mins by Lanthascreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50591954(CHEMBL5183346)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of recombinant human PLK4 incubated for 60 mins by Lanthascreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50591926(CHEMBL5171233)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of recombinant human PLK4 incubated for 60 mins by Lanthascreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50591948(CHEMBL5188129)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of recombinant human PLK4 incubated for 60 mins by Lanthascreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50591931(CHEMBL5200865)
Affinity DataIC50:  0.800nMAssay Description:Inhibition of recombinant human PLK4 incubated for 60 mins by Lanthascreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50591925(CHEMBL5185324)
Affinity DataIC50:  1nMAssay Description:Inhibition of recombinant human PLK4 incubated for 60 mins by Lanthascreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50591953(CHEMBL5194020)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of recombinant human PLK4 incubated for 60 mins by Lanthascreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50437841(CHEMBL2407900)
Affinity DataIC50:  1.60nMAssay Description:Inhibition of PLK4 (unknown origin) by Lanthascreen Eu Kinase binding assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50591955(CHEMBL5191641)
Affinity DataIC50:  1.80nMAssay Description:Inhibition of recombinant human PLK4 incubated for 60 mins by Lanthascreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50591939(CHEMBL5185225)
Affinity DataIC50:  2.70nMAssay Description:Inhibition of PLK4 (unknown origin) by Lanthascreen Eu Kinase binding assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50591950(CHEMBL5176789)
Affinity DataIC50:  2.70nMAssay Description:Inhibition of recombinant human PLK4 incubated for 60 mins by Lanthascreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50591939(CHEMBL5185225)
Affinity DataIC50:  3nMAssay Description:Inhibition of recombinant human PLK4 incubated for 60 mins by Lanthascreen Eu kinase binding assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50591947(CHEMBL5190548)
Affinity DataIC50:  3.70nMAssay Description:Inhibition of recombinant human PLK4 incubated for 60 mins by Lanthascreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50591942(CHEMBL5207473)
Affinity DataIC50:  3.80nMAssay Description:Inhibition of recombinant human PLK4 incubated for 60 mins by Lanthascreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50591941(CHEMBL5201909)
Affinity DataIC50:  4nMAssay Description:Inhibition of recombinant human PLK4 incubated for 60 mins by Lanthascreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50073587(CHEMBL3408947 | US10358436, Example A185 | US20230...)
Affinity DataIC50:  4.90nMAssay Description:Inhibition of PLK4 (unknown origin) by Lanthascreen Eu Kinase binding assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50591929(CHEMBL5175294)
Affinity DataIC50:  5.5nMAssay Description:Inhibition of recombinant human PLK4 incubated for 60 mins by Lanthascreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50591933(CHEMBL5187941)
Affinity DataIC50:  5.60nMAssay Description:Inhibition of recombinant human PLK4 incubated for 60 mins by Lanthascreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase PAK 4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50591962(CHEMBL5175418)
Affinity DataIC50:  5.90nMAssay Description:Inhibition of PAK4 (unknown origin) using S2 as substrate incubated for 60 mins in the presence of ATP by time-resolved HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50591938(CHEMBL5198607)
Affinity DataIC50:  6.5nMAssay Description:Inhibition of recombinant human PLK4 incubated for 60 mins by Lanthascreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50591940(CHEMBL5200125)
Affinity DataIC50:  7nMAssay Description:Inhibition of recombinant human PLK4 incubated for 60 mins by Lanthascreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50426474(CHEMBL1980391)
Affinity DataIC50:  7nMAssay Description:Inhibition of PLK4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50591951(CHEMBL5180759)
Affinity DataIC50:  7.90nMAssay Description:Inhibition of recombinant human PLK4 incubated for 60 mins by Lanthascreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50591927(CHEMBL5208535)
Affinity DataIC50:  8.70nMAssay Description:Inhibition of recombinant human PLK4 incubated for 60 mins by Lanthascreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50426474(CHEMBL1980391)
Affinity DataIC50:  10nMAssay Description:Inhibition of VEGFR2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50591937(CHEMBL5175172)
Affinity DataIC50:  11nMAssay Description:Inhibition of recombinant human PLK4 incubated for 60 mins by Lanthascreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50591928(CHEMBL5199896)
Affinity DataIC50:  15nMAssay Description:Inhibition of recombinant human PLK4 incubated for 60 mins by Lanthascreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50591952(CHEMBL5169342)
Affinity DataIC50:  18nMAssay Description:Inhibition of recombinant human PLK4 incubated for 60 mins by Lanthascreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50591946(CHEMBL5183478)
Affinity DataIC50:  20nMAssay Description:Inhibition of recombinant human PLK4 incubated for 60 mins by Lanthascreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50591924(CHEMBL5179518)
Affinity DataIC50:  21nMAssay Description:Inhibition of recombinant human PLK4 incubated for 60 mins by Lanthascreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50591961(CHEMBL5200812)
Affinity DataIC50:  21nMAssay Description:Inhibition of recombinant human PLK4 incubated for 60 mins by Lanthascreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50591935(CHEMBL5198928)
Affinity DataIC50:  22nMAssay Description:Inhibition of recombinant human PLK4 incubated for 60 mins by Lanthascreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50591963(CHEMBL5173724)
Affinity DataIC50:  22nMAssay Description:Inhibition of PLK4 (unknown origin) in the presence of ATP at Km concentrationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50591930(CHEMBL5181286)
Affinity DataIC50:  23nMAssay Description:Inhibition of recombinant human PLK4 incubated for 60 mins by Lanthascreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50426474(CHEMBL1980391)
Affinity DataIC50:  24nMAssay Description:Inhibition of CHK2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50591945(CHEMBL5192169)
Affinity DataIC50:  48nMAssay Description:Inhibition of recombinant human PLK4 incubated for 60 mins by Lanthascreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAurora kinase A(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50426474(CHEMBL1980391)
Affinity DataIC50:  58nMAssay Description:Inhibition of Aurora A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50591936(CHEMBL5187903)
Affinity DataIC50:  79nMAssay Description:Inhibition of recombinant human PLK4 incubated for 60 mins by Lanthascreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase PAK 4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50591934(CHEMBL5209160)
Affinity DataIC50:  96nMAssay Description:Inhibition of PAK4 (unknown origin) incubated for 60 mins by time-resolved HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAurora kinase A(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50591939(CHEMBL5185225)
Affinity DataIC50:  108nMAssay Description:Inhibition of Aurora A (unknown origin) by Z'-LYTE kinase assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50591943(CHEMBL5190474)
Affinity DataIC50:  118nMAssay Description:Inhibition of recombinant human PLK4 incubated for 60 mins by Lanthascreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50591923(CHEMBL5192817)
Affinity DataIC50:  206nMAssay Description:Inhibition of recombinant human PLK4 incubated for 60 mins by Lanthascreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase PAK 4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50591948(CHEMBL5188129)
Affinity DataIC50:  231nMAssay Description:Inhibition of PAK4 (unknown origin) incubated for 60 mins by time-resolved HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50591944(CHEMBL5181116)
Affinity DataIC50:  241nMAssay Description:Inhibition of recombinant human PLK4 incubated for 60 mins by Lanthascreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
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