Compile Data Set for Download or QSAR
maximum 50k data
Found 64 Enz. Inhib. hit(s) with all data for entry = 50017275
TargetApelin receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50600613(CHEMBL5028970)
Affinity DataEC50:  162nMAssay Description:Agonist activity at human APJ receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50600627(CHEMBL5191719)
Affinity DataEC50:  463nMAssay Description:Agonist activity at human AGTRL1 expressed in CHO-K1 cells assessed as induction of beta-arrestin 2 recruitment incubated for 90 mins by PathHunter a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50600615(CHEMBL5187822)
Affinity DataEC50:  7nMAssay Description:Agonist activity at human APJ receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50600616(CHEMBL5171394)
Affinity DataEC50:  4.30nMAssay Description:Agonist activity at human APJ receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50600617(CHEMBL5199407)
Affinity DataEC50:  6.40nMAssay Description:Agonist activity at human APJ receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50600618(CHEMBL5200689)
Affinity DataEC50:  2.40nMAssay Description:Agonist activity at human APJ receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50600619(CHEMBL5180761)
Affinity DataEC50:  28nMAssay Description:Agonist activity at human APJ receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50600620(CHEMBL5169966)
Affinity DataEC50:  6nMAssay Description:Agonist activity at human APJ receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50600621(CHEMBL5204722)
Affinity DataEC50:  3.40nMAssay Description:Agonist activity at human APJ receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50600622(CHEMBL5169875)
Affinity DataEC50:  2nMAssay Description:Agonist activity at human APJ receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50600623(CHEMBL5178250)
Affinity DataEC50:  0.350nMAssay Description:Agonist activity at human APJ receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50600624(CHEMBL5182575)
Affinity DataEC50:  4nMAssay Description:Agonist activity at human APJ receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50600625(CHEMBL5191542)
Affinity DataEC50:  15nMAssay Description:Agonist activity at human APJ receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50600626(CHEMBL5195332)
Affinity DataEC50:  54nMAssay Description:Agonist activity at human APJ receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50600627(CHEMBL5191719)
Affinity DataEC50:  6.5nMAssay Description:Agonist activity at human APJ receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50600613(CHEMBL5028970)
Affinity DataEC50:  136nMAssay Description:Agonist activity at human APJ receptor expressed in CHO cells co-expressing Galphaq16 assessed as stimulation of Ca2+ mobilization measured at 1 sec ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50600628(CHEMBL5202746)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human APJ receptor expressed in CHO cells co-expressing Galphaq16 assessed as stimulation of Ca2+ mobilization measured at 1 sec ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50600629(CHEMBL5173117)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human APJ receptor expressed in CHO cells co-expressing Galphaq16 assessed as stimulation of Ca2+ mobilization measured at 1 sec ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50600630(CHEMBL5193953)
Affinity DataEC50:  3.84E+3nMAssay Description:Agonist activity at human APJ receptor expressed in CHO cells co-expressing Galphaq16 assessed as stimulation of Ca2+ mobilization measured at 1 sec ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50600614(CHEMBL5169699)
Affinity DataEC50:  90nMAssay Description:Agonist activity at human APJ receptor expressed in CHO cells co-expressing Galphaq16 assessed as stimulation of Ca2+ mobilization measured at 1 sec ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50600631(CHEMBL5204058)
Affinity DataEC50:  265nMAssay Description:Agonist activity at human APJ receptor expressed in CHO cells co-expressing Galphaq16 assessed as stimulation of Ca2+ mobilization measured at 1 sec ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50600632(CHEMBL5196764)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human APJ receptor expressed in CHO cells co-expressing Galphaq16 assessed as stimulation of Ca2+ mobilization measured at 1 sec ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50600633(CHEMBL5170758)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human APJ receptor expressed in CHO cells co-expressing Galphaq16 assessed as stimulation of Ca2+ mobilization measured at 1 sec ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50600634(CHEMBL5173155)
Affinity DataEC50:  5.09E+3nMAssay Description:Agonist activity at human APJ receptor expressed in CHO cells co-expressing Galphaq16 assessed as stimulation of Ca2+ mobilization measured at 1 sec ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50600635(CHEMBL5198207)
Affinity DataEC50:  234nMAssay Description:Agonist activity at human APJ receptor expressed in CHO cells co-expressing Galphaq16 assessed as stimulation of Ca2+ mobilization measured at 1 sec ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50600615(CHEMBL5187822)
Affinity DataEC50:  44nMAssay Description:Agonist activity at human APJ receptor expressed in CHO cells co-expressing Galphaq16 assessed as stimulation of Ca2+ mobilization measured at 1 sec ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50600636(CHEMBL5203748)
Affinity DataEC50:  377nMAssay Description:Agonist activity at human APJ receptor expressed in CHO cells co-expressing Galphaq16 assessed as stimulation of Ca2+ mobilization measured at 1 sec ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50600637(CHEMBL5171244)
Affinity DataEC50:  2.97E+3nMAssay Description:Agonist activity at human APJ receptor expressed in CHO cells co-expressing Galphaq16 assessed as stimulation of Ca2+ mobilization measured at 1 sec ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50600616(CHEMBL5171394)
Affinity DataEC50:  46nMAssay Description:Agonist activity at human APJ receptor expressed in CHO cells co-expressing Galphaq16 assessed as stimulation of Ca2+ mobilization measured at 1 sec ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50600638(CHEMBL5206392)
Affinity DataEC50:  140nMAssay Description:Agonist activity at human APJ receptor expressed in CHO cells co-expressing Galphaq16 assessed as stimulation of Ca2+ mobilization measured at 1 sec ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50600617(CHEMBL5199407)
Affinity DataEC50:  49nMAssay Description:Agonist activity at human APJ receptor expressed in CHO cells co-expressing Galphaq16 assessed as stimulation of Ca2+ mobilization measured at 1 sec ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50600639(CHEMBL5208205)
Affinity DataEC50:  267nMAssay Description:Agonist activity at human APJ receptor expressed in CHO cells co-expressing Galphaq16 assessed as stimulation of Ca2+ mobilization measured at 1 sec ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50600640(CHEMBL5183735)
Affinity DataEC50:  272nMAssay Description:Agonist activity at human APJ receptor expressed in CHO cells co-expressing Galphaq16 assessed as stimulation of Ca2+ mobilization measured at 1 sec ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50600641(CHEMBL5206038)
Affinity DataEC50:  163nMAssay Description:Agonist activity at human APJ receptor expressed in CHO cells co-expressing Galphaq16 assessed as stimulation of Ca2+ mobilization measured at 1 sec ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50600618(CHEMBL5200689)
Affinity DataEC50:  64nMAssay Description:Agonist activity at human APJ receptor expressed in CHO cells co-expressing Galphaq16 assessed as stimulation of Ca2+ mobilization measured at 1 sec ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50600642(CHEMBL5188344)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human APJ receptor expressed in CHO cells co-expressing Galphaq16 assessed as stimulation of Ca2+ mobilization measured at 1 sec ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50600643(CHEMBL5171549)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human APJ receptor expressed in CHO cells co-expressing Galphaq16 assessed as stimulation of Ca2+ mobilization measured at 1 sec ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50600644(CHEMBL5178820)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human APJ receptor expressed in CHO cells co-expressing Galphaq16 assessed as stimulation of Ca2+ mobilization measured at 1 sec ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50600645(CHEMBL5207599)
Affinity DataEC50:  5.86E+3nMAssay Description:Agonist activity at human APJ receptor expressed in CHO cells co-expressing Galphaq16 assessed as stimulation of Ca2+ mobilization measured at 1 sec ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50600646(CHEMBL5198051)
Affinity DataEC50:  538nMAssay Description:Agonist activity at human APJ receptor expressed in CHO cells co-expressing Galphaq16 assessed as stimulation of Ca2+ mobilization measured at 1 sec ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50600647(CHEMBL5189487)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human APJ receptor expressed in CHO cells co-expressing Galphaq16 assessed as stimulation of Ca2+ mobilization measured at 1 sec ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50600648(CHEMBL5198518)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human APJ receptor expressed in CHO cells co-expressing Galphaq16 assessed as stimulation of Ca2+ mobilization measured at 1 sec ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50600619(CHEMBL5180761)
Affinity DataEC50:  69nMAssay Description:Agonist activity at human APJ receptor expressed in CHO cells co-expressing Galphaq16 assessed as stimulation of Ca2+ mobilization measured at 1 sec ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50600649(CHEMBL5180988)
Affinity DataEC50:  100nMAssay Description:Agonist activity at human APJ receptor expressed in CHO cells co-expressing Galphaq16 assessed as stimulation of Ca2+ mobilization measured at 1 sec ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50600620(CHEMBL5169966)
Affinity DataEC50:  31nMAssay Description:Agonist activity at human APJ receptor expressed in CHO cells co-expressing Galphaq16 assessed as stimulation of Ca2+ mobilization measured at 1 sec ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50600621(CHEMBL5204722)
Affinity DataEC50:  11nMAssay Description:Agonist activity at human APJ receptor expressed in CHO cells co-expressing Galphaq16 assessed as stimulation of Ca2+ mobilization measured at 1 sec ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50600650(CHEMBL5204090)
Affinity DataEC50:  162nMAssay Description:Agonist activity at human APJ receptor expressed in CHO cells co-expressing Galphaq16 assessed as stimulation of Ca2+ mobilization measured at 1 sec ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50600622(CHEMBL5169875)
Affinity DataEC50:  14nMAssay Description:Agonist activity at human APJ receptor expressed in CHO cells co-expressing Galphaq16 assessed as stimulation of Ca2+ mobilization measured at 1 sec ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50600623(CHEMBL5178250)
Affinity DataEC50:  24nMAssay Description:Agonist activity at human APJ receptor expressed in CHO cells co-expressing Galphaq16 assessed as stimulation of Ca2+ mobilization measured at 1 sec ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50600651(CHEMBL5176533)
Affinity DataEC50:  834nMAssay Description:Agonist activity at human APJ receptor expressed in CHO cells co-expressing Galphaq16 assessed as stimulation of Ca2+ mobilization measured at 1 sec ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
Displayed 1 to 50 (of 64 total ) | Next | Last >>
Jump to: