Report error Found 159 Enz. Inhib. hit(s) with all data for entry = 50017936
TargetRAC-gamma serine/threonine-protein kinase(Human)
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 0.100nMAssay Description:Inhibition of recombinant N-terminal GST tagged AKT2 (108 to 479 end residues) (unknown origin) catalytic domain expressed in Sf21 cells using peptid...More data for this Ligand-Target Pair
TargetRAC-gamma serine/threonine-protein kinase(Human)
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 0.100nMAssay Description:Inhibition of recombinant N-terminal GST tagged AKT2 (108 to 479 end residues) (unknown origin) catalytic domain expressed in Sf21 cells using peptid...More data for this Ligand-Target Pair
TargetRAC-gamma serine/threonine-protein kinase(Human)
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 0.100nMAssay Description:Inhibition of recombinant N-terminal GST tagged AKT2 (108 to 479 end residues) (unknown origin) catalytic domain expressed in Sf21 cells using peptid...More data for this Ligand-Target Pair
TargetRAC-gamma serine/threonine-protein kinase(Human)
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Inhibition of recombinant N-terminal GST tagged AKT2 (108 to 479 end residues) (unknown origin) catalytic domain expressed in Sf21 cells using peptid...More data for this Ligand-Target Pair
TargetRAC-gamma serine/threonine-protein kinase(Human)
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Inhibition of recombinant N-terminal GST tagged AKT2 (108 to 479 end residues) (unknown origin) catalytic domain expressed in Sf21 cells using peptid...More data for this Ligand-Target Pair
TargetRAC-gamma serine/threonine-protein kinase(Human)
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Inhibition of recombinant N-terminal GST tagged AKT2 (108 to 479 end residues) (unknown origin) catalytic domain expressed in Sf21 cells using peptid...More data for this Ligand-Target Pair
TargetRAC-gamma serine/threonine-protein kinase(Human)
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Inhibition of recombinant N-terminal GST tagged AKT2 (108 to 479 end residues) (unknown origin) catalytic domain expressed in Sf21 cells using peptid...More data for this Ligand-Target Pair
TargetRAC-gamma serine/threonine-protein kinase(Human)
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Inhibition of recombinant N-terminal GST tagged AKT2 (108 to 479 end residues) (unknown origin) catalytic domain expressed in Sf21 cells using peptid...More data for this Ligand-Target Pair
TargetRAC-gamma serine/threonine-protein kinase(Human)
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 0.300nMAssay Description:Inhibition of recombinant N-terminal GST tagged AKT2 (108 to 479 end residues) (unknown origin) catalytic domain expressed in Sf21 cells using peptid...More data for this Ligand-Target Pair
TargetRAC-gamma serine/threonine-protein kinase(Human)
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 0.300nMAssay Description:Inhibition of recombinant N-terminal GST tagged AKT2 (108 to 479 end residues) (unknown origin) catalytic domain expressed in Sf21 cells using peptid...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Human)
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 0.400nMAssay Description:Inhibition of recombinant AKT1 (104 to 480 end residues) (unknown origin) catalytic domain expressed in Sf21 cells using peptide substrate incubated ...More data for this Ligand-Target Pair
TargetRAC-gamma serine/threonine-protein kinase(Human)
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 0.400nMAssay Description:Inhibition of recombinant N-terminal GST tagged AKT2 (108 to 479 end residues) (unknown origin) catalytic domain expressed in Sf21 cells using peptid...More data for this Ligand-Target Pair
TargetRAC-gamma serine/threonine-protein kinase(Human)
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 0.400nMAssay Description:Inhibition of recombinant N-terminal GST tagged AKT2 (108 to 479 end residues) (unknown origin) catalytic domain expressed in Sf21 cells using peptid...More data for this Ligand-Target Pair
TargetRAC-gamma serine/threonine-protein kinase(Human)
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:Inhibition of recombinant N-terminal GST tagged AKT2 (108 to 479 end residues) (unknown origin) catalytic domain expressed in Sf21 cells using peptid...More data for this Ligand-Target Pair
TargetRAC-gamma serine/threonine-protein kinase(Human)
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:Inhibition of recombinant N-terminal GST tagged AKT2 (108 to 479 end residues) (unknown origin) catalytic domain expressed in Sf21 cells using peptid...More data for this Ligand-Target Pair
TargetRAC-gamma serine/threonine-protein kinase(Human)
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:Inhibition of recombinant N-terminal GST tagged AKT2 (108 to 479 end residues) (unknown origin) catalytic domain expressed in Sf21 cells using peptid...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Human)
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 0.600nMAssay Description:Inhibition of recombinant AKT1 (104 to 480 end residues) (unknown origin) catalytic domain expressed in Sf21 cells using peptide substrate incubated ...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Human)
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 0.600nMAssay Description:Inhibition of recombinant AKT1 (104 to 480 end residues) (unknown origin) catalytic domain expressed in Sf21 cells using peptide substrate incubated ...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Human)
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 0.700nMAssay Description:Inhibition of recombinant AKT1 (104 to 480 end residues) (unknown origin) catalytic domain expressed in Sf21 cells using peptide substrate incubated ...More data for this Ligand-Target Pair
TargetRAC-gamma serine/threonine-protein kinase(Human)
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 0.700nMAssay Description:Inhibition of recombinant N-terminal GST tagged AKT2 (108 to 479 end residues) (unknown origin) catalytic domain expressed in Sf21 cells using peptid...More data for this Ligand-Target Pair
TargetRAC-gamma serine/threonine-protein kinase(Human)
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of recombinant N-terminal GST tagged AKT2 (108 to 479 end residues) (unknown origin) catalytic domain expressed in Sf21 cells using peptid...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Human)
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 1.10nMAssay Description:Inhibition of recombinant AKT1 (104 to 480 end residues) (unknown origin) catalytic domain expressed in Sf21 cells using peptide substrate incubated ...More data for this Ligand-Target Pair
TargetRAC-beta serine/threonine-protein kinase(Human)
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 1.20nMAssay Description:Inhibition of recombinant AKT2 (120 to 481 end residues) (unknown origin) catalytic domain expressed in Sf21 cells using peptide substrate incubated ...More data for this Ligand-Target Pair
TargetRAC-gamma serine/threonine-protein kinase(Human)
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 1.20nMAssay Description:Inhibition of recombinant N-terminal GST tagged AKT2 (108 to 479 end residues) (unknown origin) catalytic domain expressed in Sf21 cells using peptid...More data for this Ligand-Target Pair
TargetRAC-gamma serine/threonine-protein kinase(Human)
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 1.20nMAssay Description:Inhibition of recombinant N-terminal GST tagged AKT2 (108 to 479 end residues) (unknown origin) catalytic domain expressed in Sf21 cells using peptid...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Human)
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 1.30nMAssay Description:Inhibition of recombinant AKT1 (104 to 480 end residues) (unknown origin) catalytic domain expressed in Sf21 cells using peptide substrate incubated ...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Human)
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 1.5nMAssay Description:Inhibition of recombinant AKT1 (104 to 480 end residues) (unknown origin) catalytic domain expressed in Sf21 cells using peptide substrate incubated ...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Human)
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 1.60nMAssay Description:Inhibition of recombinant AKT1 (104 to 480 end residues) (unknown origin) catalytic domain expressed in Sf21 cells using peptide substrate incubated ...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Human)
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 1.60nMAssay Description:Inhibition of recombinant AKT1 (104 to 480 end residues) (unknown origin) catalytic domain expressed in Sf21 cells using peptide substrate incubated ...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Human)
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 1.60nMAssay Description:Inhibition of recombinant AKT1 (104 to 480 end residues) (unknown origin) catalytic domain expressed in Sf21 cells using peptide substrate incubated ...More data for this Ligand-Target Pair
TargetRAC-gamma serine/threonine-protein kinase(Human)
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 1.60nMAssay Description:Inhibition of recombinant N-terminal GST tagged AKT2 (108 to 479 end residues) (unknown origin) catalytic domain expressed in Sf21 cells using peptid...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Human)
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 1.90nMAssay Description:Inhibition of recombinant AKT1 (104 to 480 end residues) (unknown origin) catalytic domain expressed in Sf21 cells using peptide substrate incubated ...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Human)
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 2.40nMAssay Description:Inhibition of recombinant AKT1 (104 to 480 end residues) (unknown origin) catalytic domain expressed in Sf21 cells using peptide substrate incubated ...More data for this Ligand-Target Pair
TargetRAC-gamma serine/threonine-protein kinase(Human)
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 2.60nMAssay Description:Inhibition of recombinant N-terminal GST tagged AKT2 (108 to 479 end residues) (unknown origin) catalytic domain expressed in Sf21 cells using peptid...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Human)
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 2.80nMAssay Description:Inhibition of recombinant AKT1 (104 to 480 end residues) (unknown origin) catalytic domain expressed in Sf21 cells using peptide substrate incubated ...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Human)
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 3.5nMAssay Description:Inhibition of recombinant AKT1 (104 to 480 end residues) (unknown origin) catalytic domain expressed in Sf21 cells using peptide substrate incubated ...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Human)
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 3.80nMAssay Description:Inhibition of recombinant AKT1 (104 to 480 end residues) (unknown origin) catalytic domain expressed in Sf21 cells using peptide substrate incubated ...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Human)
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 4.10nMAssay Description:Inhibition of recombinant AKT1 (104 to 480 end residues) (unknown origin) catalytic domain expressed in Sf21 cells using peptide substrate incubated ...More data for this Ligand-Target Pair
TargetRAC-gamma serine/threonine-protein kinase(Human)
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 4.40nMAssay Description:Inhibition of recombinant N-terminal GST tagged AKT2 (108 to 479 end residues) (unknown origin) catalytic domain expressed in Sf21 cells using peptid...More data for this Ligand-Target Pair
TargetRAC-beta serine/threonine-protein kinase(Human)
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 4.90nMAssay Description:Inhibition of recombinant AKT2 (120 to 481 end residues) (unknown origin) catalytic domain expressed in Sf21 cells using peptide substrate incubated ...More data for this Ligand-Target Pair
TargetRAC-beta serine/threonine-protein kinase(Human)
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 5.70nMAssay Description:Inhibition of recombinant AKT2 (120 to 481 end residues) (unknown origin) catalytic domain expressed in Sf21 cells using peptide substrate incubated ...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Human)
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Inhibition of recombinant AKT1 (104 to 480 end residues) (unknown origin) catalytic domain expressed in Sf21 cells using peptide substrate incubated ...More data for this Ligand-Target Pair
TargetRAC-beta serine/threonine-protein kinase(Human)
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Inhibition of recombinant AKT2 (120 to 481 end residues) (unknown origin) catalytic domain expressed in Sf21 cells using peptide substrate incubated ...More data for this Ligand-Target Pair
TargetRAC-beta serine/threonine-protein kinase(Human)
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 6.30nMAssay Description:Inhibition of recombinant AKT2 (120 to 481 end residues) (unknown origin) catalytic domain expressed in Sf21 cells using peptide substrate incubated ...More data for this Ligand-Target Pair
TargetRAC-gamma serine/threonine-protein kinase(Human)
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 6.60nMAssay Description:Inhibition of recombinant N-terminal GST tagged AKT2 (108 to 479 end residues) (unknown origin) catalytic domain expressed in Sf21 cells using peptid...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Human)
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 6.80nMAssay Description:Inhibition of recombinant AKT1 (104 to 480 end residues) (unknown origin) catalytic domain expressed in Sf21 cells using peptide substrate incubated ...More data for this Ligand-Target Pair
TargetRAC-beta serine/threonine-protein kinase(Human)
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 6.90nMAssay Description:Inhibition of recombinant AKT2 (120 to 481 end residues) (unknown origin) catalytic domain expressed in Sf21 cells using peptide substrate incubated ...More data for this Ligand-Target Pair
TargetRAC-gamma serine/threonine-protein kinase(Human)
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 7.40nMAssay Description:Inhibition of recombinant N-terminal GST tagged AKT2 (108 to 479 end residues) (unknown origin) catalytic domain expressed in Sf21 cells using peptid...More data for this Ligand-Target Pair
TargetRAC-gamma serine/threonine-protein kinase(Human)
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 7.40nMAssay Description:Inhibition of recombinant N-terminal GST tagged AKT2 (108 to 479 end residues) (unknown origin) catalytic domain expressed in Sf21 cells using peptid...More data for this Ligand-Target Pair
TargetRAC-gamma serine/threonine-protein kinase(Human)
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Nanjing Chia-Tai Tianqing Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 7.5nMAssay Description:Inhibition of recombinant N-terminal GST tagged AKT2 (108 to 479 end residues) (unknown origin) catalytic domain expressed in Sf21 cells using peptid...More data for this Ligand-Target Pair





















3D Structure (crystal)



