Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50016505
TargetNAD-dependent protein deacetylase sirtuin-2(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50595366(CHEMBL5207210)
Affinity DataIC50: 1.18E+5nMAssay Description:Inhibition of human SIRT2 using fluorogenic ZMAL as substrate incubated for 4 hrs in the presence of beta-NAD+ as cofactor by fluorescence based micr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50595367(CHEMBL5172985)
Affinity DataIC50: 1.51E+5nMAssay Description:Inhibition of human SIRT2 using fluorogenic ZMAL as substrate incubated for 4 hrs in the presence of beta-NAD+ as cofactor by fluorescence based micr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50595365(CHEMBL5208366)
Affinity DataIC50: 1.53E+5nMAssay Description:Inhibition of human SIRT2 using fluorogenic ZMAL as substrate incubated for 4 hrs in the presence of beta-NAD+ as cofactor by fluorescence based micr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetNAD-dependent protein deacetylase sirtuin-1(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50595365(CHEMBL5208366)
Affinity DataIC50: 1.76E+5nMAssay Description:Inhibition of human SIRT1 using fluorogenic ZMAL as substrate incubated for 4 hrs in the presence of beta-NAD+ as cofactor by fluorescence based micr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed