Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50015921
Target5-hydroxytryptamine receptor 6(Human)
Hec Research and Development Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 394084BDBM394084(US9974785, Example 3)
Affinity DataKi:  0.430nMAssay Description:Displacement of [3H]-LSD from human 5HT6 receptor expressed in CHO cells assessed as inhibition constant incubated for 120 mins by liquid scintillati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Hec Research and Development Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 394083BDBM394083(US9974785, Example 2)
Affinity DataKi:  0.460nMAssay Description:Displacement of [3H]-LSD from human 5HT6 receptor expressed in CHO cells assessed as inhibition constant incubated for 120 mins by liquid scintillati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Hec Research and Development Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50590516BDBM50590516(CHEMBL5196479)
Affinity DataKi:  0.510nMAssay Description:Displacement of [3H]-LSD from human 5HT6 receptor expressed in CHO cells assessed as inhibition constant incubated for 120 mins by liquid scintillati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Hec Research and Development Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 394086BDBM394086(US9974785, Example 5)
Affinity DataKi:  0.520nMAssay Description:Displacement of [3H]-LSD from human 5HT6 receptor expressed in CHO cells assessed as inhibition constant incubated for 120 mins by liquid scintillati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Hec Research and Development Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 394087BDBM394087(US9974785, Example 6)
Affinity DataKi:  0.680nMAssay Description:Displacement of [3H]-LSD from human 5HT6 receptor expressed in CHO cells assessed as inhibition constant incubated for 120 mins by liquid scintillati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Hec Research and Development Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50019754BDBM50019754(LU-AE58054 | IDALOPIRDINE)
Affinity DataKi:  0.830nMAssay Description:Displacement of [3H]-LSD from human 5HT6 receptor expressed in CHO cells assessed as inhibition constant incubated for 120 mins by liquid scintillati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Hec Research and Development Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 394085BDBM394085(US9974785, Example 4)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]-LSD from human 5HT6 receptor expressed in CHO cells assessed as inhibition constant incubated for 120 mins by liquid scintillati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Hec Research and Development Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 394082BDBM394082(US9974785, Example 1)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]-LSD from human 5HT6 receptor expressed in CHO cells assessed as inhibition constant incubated for 120 mins by liquid scintillati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Hec Research and Development Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 394088BDBM394088(US9974785, Example 7)
Affinity DataKi:  6.40nMAssay Description:Displacement of [3H]-LSD from human 5HT6 receptor expressed in CHO cells assessed as inhibition constant incubated for 120 mins by liquid scintillati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Hec Research and Development Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 394091BDBM394091(US9974785, Example 11)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]-LSD from human 5HT6 receptor expressed in CHO cells assessed as inhibition constant incubated for 120 mins by liquid scintillati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Hec Research and Development Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 394089BDBM394089(US9974785, Example 8)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]-LSD from human 5HT6 receptor expressed in CHO cells assessed as inhibition constant incubated for 120 mins by liquid scintillati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Hec Research and Development Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 394093BDBM394093(US9974785, Example 13)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]-LSD from human 5HT6 receptor expressed in CHO cells assessed as inhibition constant incubated for 120 mins by liquid scintillati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Hec Research and Development Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 394097BDBM394097(US9974785, Example 17)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]-LSD from human 5HT6 receptor expressed in CHO cells assessed as inhibition constant incubated for 120 mins by liquid scintillati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Hec Research and Development Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 394099BDBM394099(US9974785, Example 19)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]-LSD from human 5HT6 receptor expressed in CHO cells assessed as inhibition constant incubated for 120 mins by liquid scintillati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Hec Research and Development Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 394098BDBM394098(US9974785, Example 18)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]-LSD from human 5HT6 receptor expressed in CHO cells assessed as inhibition constant incubated for 120 mins by liquid scintillati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Hec Research and Development Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 394095BDBM394095(US9974785, Example 15)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]-LSD from human 5HT6 receptor expressed in CHO cells assessed as inhibition constant incubated for 120 mins by liquid scintillati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Hec Research and Development Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 394094BDBM394094(US9974785, Example 14)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]-LSD from human 5HT6 receptor expressed in CHO cells assessed as inhibition constant incubated for 120 mins by liquid scintillati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Hec Research and Development Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 394092BDBM394092(US9974785, Example 12)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]-LSD from human 5HT6 receptor expressed in CHO cells assessed as inhibition constant incubated for 120 mins by liquid scintillati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Hec Research and Development Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 394100BDBM394100(US9974785, Example 20)
Affinity DataKi:  44nMAssay Description:Displacement of [3H]-LSD from human 5HT6 receptor expressed in CHO cells assessed as inhibition constant incubated for 120 mins by liquid scintillati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Hec Research and Development Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 394096BDBM394096(US9974785, Example 16)
Affinity DataKi:  67nMAssay Description:Displacement of [3H]-LSD from human 5HT6 receptor expressed in CHO cells assessed as inhibition constant incubated for 120 mins by liquid scintillati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed