Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50019800
TargetGonadotropin-releasing hormone receptor(Human)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50623129(CHEMBL5419365 | US20250000864, Compound 7)
Affinity DataIC50: 0.220nMAssay Description:Displacement of [1251][D-Trp6]-LH-RH from human GnRH-R expressed in Chem-1 cells incubated for 60 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50623125(CHEMBL5398152)
Affinity DataIC50: 0.230nMAssay Description:Displacement of [1251][D-Trp6]-LH-RH from human GnRH-R expressed in Chem-1 cells incubated for 60 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50347982(CHEMBL1800159 | US20250000864, Compound Relugolix)
Affinity DataIC50: 0.25nMAssay Description:Displacement of [1251][D-Trp6]-LH-RH from human GnRH-R expressed in Chem-1 cells incubated for 60 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50623120(CHEMBL5434324 | US20250000864, Compound 3)
Affinity DataIC50: 0.260nMAssay Description:Displacement of [1251][D-Trp6]-LH-RH from human GnRH-R expressed in Chem-1 cells incubated for 60 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50623123(CHEMBL5400302)
Affinity DataIC50: 0.260nMAssay Description:Displacement of [1251][D-Trp6]-LH-RH from human GnRH-R expressed in Chem-1 cells incubated for 60 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50623127(CHEMBL5433025)
Affinity DataIC50: 0.280nMAssay Description:Displacement of [1251][D-Trp6]-LH-RH from human GnRH-R expressed in Chem-1 cells incubated for 60 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50623122(CHEMBL5419489)
Affinity DataIC50: 0.320nMAssay Description:Displacement of [1251][D-Trp6]-LH-RH from human GnRH-R expressed in Chem-1 cells incubated for 60 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50623124(CHEMBL5425604)
Affinity DataIC50: 0.350nMAssay Description:Displacement of [1251][D-Trp6]-LH-RH from human GnRH-R expressed in Chem-1 cells incubated for 60 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50623121(CHEMBL5427278 | US20250000864, Compound 5)
Affinity DataIC50: 0.380nMAssay Description:Displacement of [1251][D-Trp6]-LH-RH from human GnRH-R expressed in Chem-1 cells incubated for 60 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50623126(CHEMBL5413078 | US20250000864, Compound 6)
Affinity DataIC50: 0.550nMAssay Description:Displacement of [1251][D-Trp6]-LH-RH from human GnRH-R expressed in Chem-1 cells incubated for 60 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50623128(CHEMBL5420128)
Affinity DataIC50: 0.570nMAssay Description:Displacement of [1251][D-Trp6]-LH-RH from human GnRH-R expressed in Chem-1 cells incubated for 60 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed