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Found 12 Enz. Inhib. hit(s) with all data for entry = 50017346
TargetYTH domain-containing protein 1(Homo sapiens)
University Of Zurich

Curated by ChEMBL
LigandPNGBDBM50601383(CHEMBL5177286)
Affinity DataIC50:  3.90E+4nMAssay Description:Binding affinity to GST-tagged YTHDC1 m6A-reader domain (unknown origin) using RRACH-containing methylated oligoRNA incubated for 3 hrs by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetYTH domain-containing protein 1(Homo sapiens)
University Of Zurich

Curated by ChEMBL
LigandPNGBDBM50601384(CHEMBL5205586)
Affinity DataIC50:  1.42E+5nMAssay Description:Binding affinity to GST-tagged YTHDC1 m6A-reader domain (unknown origin) using RRACH-containing methylated oligoRNA incubated for 3 hrs by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails PubMed
TargetYTH domain-containing family protein 2(Homo sapiens)
University Of Zurich

Curated by ChEMBL
LigandPNGBDBM50601384(CHEMBL5205586)
Affinity DataIC50:  1.61E+5nMAssay Description:Binding affinity to GST-tagged YTHDF2 m6A-reader domain (unknown origin) using RRACH-containing methylated oligoRNA incubated for 3 hrs by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetYTH domain-containing family protein 2(Homo sapiens)
University Of Zurich

Curated by ChEMBL
LigandPNGBDBM50601385(CHEMBL5192478)
Affinity DataIC50:  1.74E+5nMAssay Description:Binding affinity to GST-tagged YTHDF2 m6A-reader domain (unknown origin) using RRACH-containing methylated oligoRNA incubated for 3 hrs by HTRF assayMore data for this Ligand-Target Pair
TargetYTH domain-containing family protein 3(Homo sapiens)
University Of Zurich

Curated by ChEMBL
LigandPNGBDBM50601385(CHEMBL5192478)
Affinity DataIC50:  2.18E+5nMAssay Description:Binding affinity to GST-tagged YTHDF3 m6A-reader domain (unknown origin) using RRACH-containing methylated oligoRNA incubated for 3 hrs by HTRF assayMore data for this Ligand-Target Pair
TargetYTH domain-containing protein 1(Homo sapiens)
University Of Zurich

Curated by ChEMBL
LigandPNGBDBM50601388(CHEMBL5170722)
Affinity DataIC50:  2.94E+5nMAssay Description:Binding affinity to GST-tagged YTHDC1 m6A-reader domain (unknown origin) using RRACH-containing methylated oligoRNA incubated for 3 hrs by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetYTH domain-containing protein 1(Homo sapiens)
University Of Zurich

Curated by ChEMBL
LigandPNGBDBM50601387(CHEMBL5179548)
Affinity DataIC50:  3.06E+5nMAssay Description:Binding affinity to GST-tagged YTHDC1 m6A-reader domain (unknown origin) using RRACH-containing methylated oligoRNA incubated for 3 hrs by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetYTH domain-containing family protein 1(Homo sapiens)
University Of Zurich

Curated by ChEMBL
LigandPNGBDBM50601385(CHEMBL5192478)
Affinity DataIC50:  3.79E+5nMAssay Description:Binding affinity to GST-tagged YTHDF1 m6A-reader domain (unknown origin) using RRACH-containing methylated oligoRNA incubated for 3 hrs by HTRF assayMore data for this Ligand-Target Pair
TargetYTH domain-containing family protein 2(Homo sapiens)
University Of Zurich

Curated by ChEMBL
LigandPNGBDBM50601383(CHEMBL5177286)
Affinity DataIC50:  4.10E+5nMAssay Description:Binding affinity to GST-tagged YTHDF2 m6A-reader domain (unknown origin) using RRACH-containing methylated oligoRNA incubated for 3 hrs by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetYTH domain-containing family protein 2(Homo sapiens)
University Of Zurich

Curated by ChEMBL
LigandPNGBDBM50601386(CHEMBL5201513)
Affinity DataIC50:  4.91E+5nMAssay Description:Binding affinity to GST-tagged YTHDF2 m6A-reader domain (unknown origin) using RRACH-containing methylated oligoRNA incubated for 3 hrs by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetYTH domain-containing protein 1(Homo sapiens)
University Of Zurich

Curated by ChEMBL
LigandPNGBDBM50163023((2R,3S,4R,5R)-2-Hydroxymethyl-5-(6-methylamino-pur...)
Affinity DataIC50:  5.04E+5nMAssay Description:Binding affinity to GST-tagged YTHDC1 m6A-reader domain (unknown origin) using RRACH-containing methylated oligoRNA incubated for 3 hrs by HTRF assayMore data for this Ligand-Target Pair
TargetYTH domain-containing protein 1(Homo sapiens)
University Of Zurich

Curated by ChEMBL
LigandPNGBDBM50601385(CHEMBL5192478)
Affinity DataIC50: >1.00E+6nMAssay Description:Binding affinity to GST-tagged YTHDC1 m6A-reader domain (unknown origin) using RRACH-containing methylated oligoRNA incubated for 3 hrs by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails PubMed