Compile Data Set for Download or QSAR
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Found 13 Enz. Inhib. hit(s) with all data for entry = 50018011
TargetBile acid receptor(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50606957(CHEMBL5218997)
Affinity DataEC50:  570nMAssay Description:Agonist activity at FXR in HEK293T cells assessed as transcriptional activity by measuring fluorescence intensity by luciferase reporter assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBile acid receptor(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50606958(CHEMBL5219921)
Affinity DataEC50:  410nMAssay Description:Agonist activity at FXR in HEK293T cells assessed as transcriptional activity by measuring fluorescence intensity by luciferase reporter assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBile acid receptor(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50606959(CHEMBL5219668)
Affinity DataEC50:  350nMAssay Description:Agonist activity at FXR in HEK293T cells assessed as transcriptional activity by measuring fluorescence intensity by luciferase reporter assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBile acid receptor(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50606960(CHEMBL5218477)
Affinity DataEC50:  2.16E+3nMAssay Description:Agonist activity at FXR in HEK293T cells assessed as transcriptional activity by measuring fluorescence intensity by luciferase reporter assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBile acid receptor(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50606961(CHEMBL5220072)
Affinity DataEC50:  270nMAssay Description:Agonist activity at FXR in HEK293T cells assessed as transcriptional activity by measuring fluorescence intensity by luciferase reporter assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBile acid receptor(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50606962(CHEMBL5219682)
Affinity DataEC50:  310nMAssay Description:Agonist activity at FXR in HEK293T cells assessed as transcriptional activity by measuring fluorescence intensity by luciferase reporter assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBile acid receptor(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM21724(3-[(E)-2-(2-chloro-4-{[3-(2,6-dichlorophenyl)-5-(1...)
Affinity DataEC50:  550nMAssay Description:Agonist activity at FXR in HEK293T cells assessed as transcriptional activity by measuring fluorescence intensity by luciferase reporter assayMore data for this Ligand-Target Pair
TargetBile acid receptor(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50606964(CHEMBL5220726)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at FXR in HEK293T cells assessed as transcriptional activity by measuring fluorescence intensity by luciferase reporter assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBile acid receptor(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50606965(CHEMBL5220601)
Affinity DataEC50:  1.12E+3nMAssay Description:Agonist activity at FXR in HEK293T cells assessed as transcriptional activity by measuring fluorescence intensity by luciferase reporter assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBile acid receptor(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50606966(CHEMBL5220022)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at FXR in HEK293T cells assessed as transcriptional activity by measuring fluorescence intensity by luciferase reporter assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBile acid receptor(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50606967(CHEMBL5219979)
Affinity DataEC50:  510nMAssay Description:Agonist activity at FXR in HEK293T cells assessed as transcriptional activity by measuring fluorescence intensity by luciferase reporter assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBile acid receptor(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50606968(CHEMBL5220935)
Affinity DataEC50:  3.19E+3nMAssay Description:Agonist activity at FXR in HEK293T cells assessed as transcriptional activity by measuring fluorescence intensity by luciferase reporter assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBile acid receptor(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50606963(CHEMBL5220664)
Affinity DataEC50:  1.09E+3nMAssay Description:Agonist activity at FXR in HEK293T cells assessed as transcriptional activity by measuring fluorescence intensity by luciferase reporter assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed