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Found 33 Enz. Inhib. hit(s) with all data for entry = 50015841
TargetCoagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL
LigandPNGBDBM50590085(CHEMBL5187102)
Affinity DataKi:  0.5nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCoagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL
LigandPNGBDBM12400(1-[(4-Chloro-phenylcarbamoyl)-methyl]-1H-indole-2-...)
Affinity DataKi:  3nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
TargetCoagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL
LigandPNGBDBM50590072(CHEMBL3904655)
Affinity DataKi:  3nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCoagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL
LigandPNGBDBM12372(1-{[5-(5-chlorothiophen-2-yl)-1,2-oxazol-3-yl]meth...)
Affinity DataKi:  3nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
TargetCoagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL
LigandPNGBDBM50590086(CHEMBL5192536)
Affinity DataKi:  4nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCoagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL
LigandPNGBDBM50590082(CHEMBL5175184)
Affinity DataKi:  6nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCoagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL
LigandPNGBDBM50590073(CHEMBL5175600)
Affinity DataKi:  7nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCoagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL
LigandPNGBDBM50590087(CHEMBL5179837)
Affinity DataKi:  8nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCoagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL
LigandPNGBDBM50590097(CHEMBL5187449)
Affinity DataKi:  9nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCoagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL
LigandPNGBDBM50590083(CHEMBL5192808)
Affinity DataKi:  11nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCoagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL
LigandPNGBDBM50590078(CHEMBL5175799)
Affinity DataKi:  12nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCoagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL
LigandPNGBDBM50590081(CHEMBL5180386)
Affinity DataKi:  13nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCoagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL
LigandPNGBDBM50590099(CHEMBL5193338)
Affinity DataKi:  37nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCoagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL
LigandPNGBDBM50590075(CHEMBL5190215)
Affinity DataKi:  49nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCoagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL
LigandPNGBDBM50590084(CHEMBL5208176)
Affinity DataKi:  51nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCoagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL
LigandPNGBDBM50590089(CHEMBL5181980)
Affinity DataKi:  52nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCoagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL
LigandPNGBDBM50590080(CHEMBL5185736)
Affinity DataKi:  55nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCoagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL
LigandPNGBDBM50590074(CHEMBL5187415)
Affinity DataKi:  56nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCoagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL
LigandPNGBDBM50590088(CHEMBL5192209)
Affinity DataKi:  57nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCoagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL
LigandPNGBDBM50590071(CHEMBL5178354)
Affinity DataKi:  63nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCoagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL
LigandPNGBDBM50590096(CHEMBL5173515)
Affinity DataKi:  65nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCoagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL
LigandPNGBDBM50590077(CHEMBL5188689)
Affinity DataKi:  70nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCoagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL
LigandPNGBDBM50590076(CHEMBL5204725)
Affinity DataKi:  162nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCoagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL
LigandPNGBDBM50590079(CHEMBL5193560)
Affinity DataKi:  188nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCoagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL
LigandPNGBDBM50590070(CHEMBL5206688)
Affinity DataKi:  204nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCoagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL
LigandPNGBDBM50590093(CHEMBL5186260)
Affinity DataKi:  204nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCoagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL
LigandPNGBDBM50590095(CHEMBL5199539)
Affinity DataKi:  241nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCoagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL
LigandPNGBDBM50590098(CHEMBL5194849)
Affinity DataKi:  1.24E+3nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCoagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL
LigandPNGBDBM50590092(CHEMBL5205467)
Affinity DataKi:  1.74E+3nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCoagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL
LigandPNGBDBM50590091(CHEMBL5202796)
Affinity DataKi:  2.93E+3nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCoagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL
LigandPNGBDBM50590090(CHEMBL5175878)
Affinity DataKi:  5.13E+3nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCoagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL
LigandPNGBDBM50590100(CHEMBL5176283)
Affinity DataKi:  1.48E+4nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCoagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL
LigandPNGBDBM50590094(CHEMBL5205339)
Affinity DataKi:  2.05E+4nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed