TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Homo sapiens (Human))
Pmc Isochem
Curated by ChEMBL
Pmc Isochem
Curated by ChEMBL
Affinity DataEC50: <5.00E+3nMAssay Description:Modulation of human Sirt3 (118 to 399 residues) deacetylation activity under non-steady state assessed as substrate deacetylation at low enzyme conce...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Homo sapiens (Human))
Pmc Isochem
Curated by ChEMBL
Pmc Isochem
Curated by ChEMBL
Affinity DataKd: 1.01E+3nMAssay Description:Binding affinity to human Sirt3 (118 to 399 residues) assessed as dissociation constant by microscale thermophoresis analysisMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Homo sapiens (Human))
Pmc Isochem
Curated by ChEMBL
Pmc Isochem
Curated by ChEMBL
Affinity DataKd: 970nMAssay Description:Binding affinity to human Sirt3 (118 to 399 residues) assessed as dissociation constant using acetylated MnSOD peptide as substrate by microscale the...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Homo sapiens (Human))
Pmc Isochem
Curated by ChEMBL
Pmc Isochem
Curated by ChEMBL
Affinity DataKd: 7.30E+3nMAssay Description:Binding affinity to human Sirt3 (118 to 399 residues) assessed as dissociation constant using acetylated MnSOD peptide as substrate by microscale the...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Homo sapiens (Human))
Pmc Isochem
Curated by ChEMBL
Pmc Isochem
Curated by ChEMBL
Affinity DataKd: 6.60E+3nMAssay Description:Binding affinity to human Sirt3 (118 to 399 residues) assessed as dissociation constant using acetylated MnSOD peptide as substrate in presence of ho...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Homo sapiens (Human))
Pmc Isochem
Curated by ChEMBL
Pmc Isochem
Curated by ChEMBL
Affinity DataKd: 290nMAssay Description:Binding affinity to human Sirt3 (118 to 399 residues) assessed as dissociation constant of ternary complex using acetylated MnSOD peptide as substrat...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Homo sapiens (Human))
Pmc Isochem
Curated by ChEMBL
Pmc Isochem
Curated by ChEMBL
Affinity DataKd: 2.99E+3nMAssay Description:Binding affinity to human Sirt3 (118 to 399 residues) assessed as dissociation constant using 625nM acetylated MnSOD peptide as substrate by microsca...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Homo sapiens (Human))
Pmc Isochem
Curated by ChEMBL
Pmc Isochem
Curated by ChEMBL
Affinity DataKon: 0.220M-1s-1Assay Description:Binding affinity to human Sirt3 (118 to 399 residues) assessed as dissociation constant (Koff) by short DNA nano levers based switchSENSE microfluid ...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Homo sapiens (Human))
Pmc Isochem
Curated by ChEMBL
Pmc Isochem
Curated by ChEMBL
Affinity DataKd: 4.60E+3nMAssay Description:Binding affinity to human Sirt3 (118 to 399 residues) assessed as dissociation constant by short DNA nano levers based switchSENSE microfluid bio-chi...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Homo sapiens (Human))
Pmc Isochem
Curated by ChEMBL
Pmc Isochem
Curated by ChEMBL
Affinity DataKoff: 70.9s-1Assay Description:Binding affinity to human Sirt3 (118 to 399 residues) assessed as dissociation constant (Kon) of ternary complex using acetylated MnSOD peptide as su...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Homo sapiens (Human))
Pmc Isochem
Curated by ChEMBL
Pmc Isochem
Curated by ChEMBL
Affinity DataKon: 0.162M-1s-1Assay Description:Binding affinity to human Sirt3 (118 to 399 residues) assessed as dissociation constant (Koff) of ternary complex using acetylated MnSOD peptide as s...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Homo sapiens (Human))
Pmc Isochem
Curated by ChEMBL
Pmc Isochem
Curated by ChEMBL
Affinity DataKd: 1.26E+4nMAssay Description:Binding affinity to human Sirt3 (118 to 399 residues) assessed as dissociation constant of ternary complex using acetylated MnSOD peptide as substrat...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Homo sapiens (Human))
Pmc Isochem
Curated by ChEMBL
Pmc Isochem
Curated by ChEMBL
Affinity DataKoff: 20.1s-1Assay Description:Binding affinity to human Sirt3 (118 to 399 residues) assessed as dissociation constant (Kon) by short DNA nano levers based switchSENSE microfluid b...More data for this Ligand-Target Pair