Affinity DataIC50: 22nMAssay Description:Binding affinity to BRD4 bromodomain 1 in human Ramos cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 240nMAssay Description:Induction of BRD4 degradation in human 231MFP cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 470nMAssay Description:Inhibition of RNF114 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 670nMAssay Description:Inhibition of FNIP1 in human HEK293T cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 7.60E+3nMAssay Description:Binding affinity to BRD4 bromodomain 1 in human Ramos cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 150nMAssay Description:Activation of caspase 3/7 in human 22Rv1 cells by Caspase-Glo reagent based analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 2nMAssay Description:Activation of caspase 3/7 in human 22Rv1 cells by Caspase-Glo reagent based analysisMore data for this Ligand-Target Pair
Affinity DataKd: 740nMAssay Description:Binding affinity to BRD4 BD2 (unknown origin) assessed as dissociation constant by isothermal titration calorimetry assayMore data for this Ligand-Target Pair
Affinity DataKd: 180nMAssay Description:Binding affinity to BRD4 BD2 (unknown origin) assessed as dissociation constant by isothermal titration calorimetry assayMore data for this Ligand-Target Pair
Affinity DataKd: 740nMAssay Description:Binding affinity to BRD2 BD1 (unknown origin) assessed as dissociation constant by isothermal titration calorimetry assayMore data for this Ligand-Target Pair
Affinity DataKd: 180nMAssay Description:Binding affinity to BRD2 BD1 (unknown origin) assessed as dissociation constant by isothermal titration calorimetry assayMore data for this Ligand-Target Pair
Affinity DataKd: 66nMAssay Description:Binding affinity to VHL (unknown origin) assessed as dissociation constant by isothermal titration calorimetry assayMore data for this Ligand-Target Pair
Affinity DataKd: 47nMAssay Description:Binding affinity to VHL (unknown origin) assessed as dissociation constant by isothermal titration calorimetry assayMore data for this Ligand-Target Pair
Affinity DataEC50: 90nMAssay Description:Activation of caspase 3/7 in human 22Rv1 cells by Caspase-Glo reagent based analysisMore data for this Ligand-Target Pair
Affinity DataKd: 115nMAssay Description:Binding affinity to BRD4 (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKd: 115nMAssay Description:Binding affinity to BRD3 (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKd: 115nMAssay Description:Binding affinity to BRD2 (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKd: 28nMAssay Description:Binding affinity to BRD4 BD1 in human Burkitts lymphoma cells assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKd: 3.00E+3nMAssay Description:Binding affinity to CRBN in human Burkitts lymphoma cells assessed as dissociation constantMore data for this Ligand-Target Pair