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Found 5 Enz. Inhib. hit(s) with all data for entry = 50018045
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Tongji University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50140257(5,7-Dihydroxy-8-methoxy-2-phenyl-chromen-4-one | 5...)
Affinity DataIC50:  190nMAssay Description:Inhibition of CDK9 (unknown origin) using [33-p]-ATP as substrate incubated for 40 mins by Western blot analysisMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetE3 ubiquitin-protein ligase RNF114(Homo sapiens)
Tongji University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50607224(CHEMBL5218793)
Affinity DataIC50:  240nMAssay Description:Inhibition of RNF114 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Homo sapiens (Human))
Tongji University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50607226(CHEMBL5220731)
Affinity DataIC50:  250nMAssay Description:Inhibition of HMGCR (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Tongji University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50607227(CHEMBL4530229)
Affinity DataIC50:  523nMAssay Description:Inhibition of CDK9 (unknown origin) incubated for 1 hr by fluorescent polarisation based assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Homo sapiens (Human))
Tongji University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50607225(CHEMBL5218794)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of HMGCR (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed