TargetP2X purinoceptor 7(Homo sapiens (Human))
Takasaki University Of Health And Welfare
Curated by ChEMBL
Takasaki University Of Health And Welfare
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Antagonist activity at P2X7 receptor in human RPMI-8226 cells assessed as inhibition of ATP-induced Ca2+ influx by fura-2 staining based assayMore data for this Ligand-Target Pair
TargetP2X purinoceptor 7(Homo sapiens (Human))
Takasaki University Of Health And Welfare
Curated by ChEMBL
Takasaki University Of Health And Welfare
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Antagonist activity at P2X7 receptor in human RPMI-8226 cells assessed as inhibition of ATP-induced Ca2+ influx by fura-2 staining based assayMore data for this Ligand-Target Pair
TargetP2X purinoceptor 7(Homo sapiens (Human))
Takasaki University Of Health And Welfare
Curated by ChEMBL
Takasaki University Of Health And Welfare
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Antagonist activity at P2X7 receptor in human RPMI-8226 cells assessed as inhibition of ATP-induced Ca2+ influx by fura-2 staining based assayMore data for this Ligand-Target Pair
TargetP2X purinoceptor 7(Homo sapiens (Human))
Takasaki University Of Health And Welfare
Curated by ChEMBL
Takasaki University Of Health And Welfare
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Antagonist activity at P2X7 receptor in human RPMI-8226 cells assessed as inhibition of ATP-induced Ca2+ influx by fura-2 staining based assayMore data for this Ligand-Target Pair
TargetP2X purinoceptor 7(Homo sapiens (Human))
Takasaki University Of Health And Welfare
Curated by ChEMBL
Takasaki University Of Health And Welfare
Curated by ChEMBL
Affinity DataIC50: 150nMAssay Description:Antagonist activity at P2X7 receptor in human RPMI-8226 cells assessed as inhibition of ATP-induced Ca2+ influx by fura-2 staining based assayMore data for this Ligand-Target Pair
TargetP2X purinoceptor 7(Homo sapiens (Human))
Takasaki University Of Health And Welfare
Curated by ChEMBL
Takasaki University Of Health And Welfare
Curated by ChEMBL
Affinity DataIC50: 180nMAssay Description:Antagonist activity at P2X7 receptor in human RPMI-8226 cells assessed as inhibition of ATP-induced Ca2+ influx by fura-2 staining based assayMore data for this Ligand-Target Pair
TargetP2X purinoceptor 7(Homo sapiens (Human))
Takasaki University Of Health And Welfare
Curated by ChEMBL
Takasaki University Of Health And Welfare
Curated by ChEMBL
Affinity DataIC50: 180nMAssay Description:Antagonist activity at P2X7 receptor in human RPMI-8226 cells assessed as inhibition of ATP-induced Ca2+ influx by fura-2 staining based assayMore data for this Ligand-Target Pair
TargetP2X purinoceptor 7(Homo sapiens (Human))
Takasaki University Of Health And Welfare
Curated by ChEMBL
Takasaki University Of Health And Welfare
Curated by ChEMBL
Affinity DataIC50: 180nMAssay Description:Antagonist activity at P2X7 receptor in human RPMI-8226 cells assessed as inhibition of ATP-induced Ca2+ influx by fura-2 staining based assayMore data for this Ligand-Target Pair
TargetP2X purinoceptor 7(Homo sapiens (Human))
Takasaki University Of Health And Welfare
Curated by ChEMBL
Takasaki University Of Health And Welfare
Curated by ChEMBL
Affinity DataIC50: 190nMAssay Description:Antagonist activity at P2X7 receptor in human RPMI-8226 cells assessed as inhibition of ATP-induced Ca2+ influx by fura-2 staining based assayMore data for this Ligand-Target Pair
TargetP2X purinoceptor 7(Homo sapiens (Human))
Takasaki University Of Health And Welfare
Curated by ChEMBL
Takasaki University Of Health And Welfare
Curated by ChEMBL
Affinity DataIC50: 240nMAssay Description:Antagonist activity at P2X7 receptor in human RPMI-8226 cells assessed as inhibition of ATP-induced Ca2+ influx by fura-2 staining based assayMore data for this Ligand-Target Pair
TargetP2X purinoceptor 7(Homo sapiens (Human))
Takasaki University Of Health And Welfare
Curated by ChEMBL
Takasaki University Of Health And Welfare
Curated by ChEMBL
Affinity DataIC50: 320nMAssay Description:Antagonist activity at P2X7 receptor in human RPMI-8226 cells assessed as inhibition of ATP-induced Ca2+ influx by fura-2 staining based assayMore data for this Ligand-Target Pair
TargetP2X purinoceptor 7(Homo sapiens (Human))
Takasaki University Of Health And Welfare
Curated by ChEMBL
Takasaki University Of Health And Welfare
Curated by ChEMBL
Affinity DataIC50: 460nMAssay Description:Antagonist activity at P2X7 receptor in human RPMI-8226 cells assessed as inhibition of ATP-induced Ca2+ influx by fura-2 staining based assayMore data for this Ligand-Target Pair
TargetP2X purinoceptor 7(Homo sapiens (Human))
Takasaki University Of Health And Welfare
Curated by ChEMBL
Takasaki University Of Health And Welfare
Curated by ChEMBL
Affinity DataIC50: 480nMAssay Description:Antagonist activity at P2X7 receptor in human RPMI-8226 cells assessed as inhibition of ATP-induced Ca2+ influx by fura-2 staining based assayMore data for this Ligand-Target Pair
TargetP2X purinoceptor 7(Homo sapiens (Human))
Takasaki University Of Health And Welfare
Curated by ChEMBL
Takasaki University Of Health And Welfare
Curated by ChEMBL
Affinity DataIC50: 560nMAssay Description:Antagonist activity at P2X7 receptor in human RPMI-8226 cells assessed as inhibition of ATP-induced Ca2+ influx by fura-2 staining based assayMore data for this Ligand-Target Pair
TargetP2X purinoceptor 7(Homo sapiens (Human))
Takasaki University Of Health And Welfare
Curated by ChEMBL
Takasaki University Of Health And Welfare
Curated by ChEMBL
Affinity DataIC50: 770nMAssay Description:Antagonist activity at P2X7 receptor in human RPMI-8226 cells assessed as inhibition of ATP-induced Ca2+ influx by fura-2 staining based assayMore data for this Ligand-Target Pair
TargetP2X purinoceptor 7(Homo sapiens (Human))
Takasaki University Of Health And Welfare
Curated by ChEMBL
Takasaki University Of Health And Welfare
Curated by ChEMBL
Affinity DataIC50: 830nMAssay Description:Antagonist activity at P2X7 receptor in human RPMI-8226 cells assessed as inhibition of ATP-induced Ca2+ influx by fura-2 staining based assayMore data for this Ligand-Target Pair
TargetP2X purinoceptor 7(Homo sapiens (Human))
Takasaki University Of Health And Welfare
Curated by ChEMBL
Takasaki University Of Health And Welfare
Curated by ChEMBL
Affinity DataIC50: 850nMAssay Description:Antagonist activity at P2X7 receptor in human RPMI-8226 cells assessed as inhibition of ATP-induced Ca2+ influx by fura-2 staining based assayMore data for this Ligand-Target Pair
TargetP2X purinoceptor 7(Homo sapiens (Human))
Takasaki University Of Health And Welfare
Curated by ChEMBL
Takasaki University Of Health And Welfare
Curated by ChEMBL
Affinity DataIC50: 950nMAssay Description:Antagonist activity at P2X7 receptor in human RPMI-8226 cells assessed as inhibition of ATP-induced Ca2+ influx by fura-2 staining based assayMore data for this Ligand-Target Pair
TargetP2X purinoceptor 7(Homo sapiens (Human))
Takasaki University Of Health And Welfare
Curated by ChEMBL
Takasaki University Of Health And Welfare
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Antagonist activity at P2X7 receptor in human RPMI-8226 cells assessed as inhibition of ATP-induced Ca2+ influx by fura-2 staining based assayMore data for this Ligand-Target Pair
TargetP2X purinoceptor 7(Homo sapiens (Human))
Takasaki University Of Health And Welfare
Curated by ChEMBL
Takasaki University Of Health And Welfare
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMAssay Description:Antagonist activity at P2X7 receptor in human RPMI-8226 cells assessed as inhibition of ATP-induced Ca2+ influx by fura-2 staining based assayMore data for this Ligand-Target Pair
TargetP2X purinoceptor 7(Homo sapiens (Human))
Takasaki University Of Health And Welfare
Curated by ChEMBL
Takasaki University Of Health And Welfare
Curated by ChEMBL
Affinity DataIC50: 2.30E+3nMAssay Description:Antagonist activity at P2X7 receptor in human RPMI-8226 cells assessed as inhibition of ATP-induced Ca2+ influx by fura-2 staining based assayMore data for this Ligand-Target Pair
TargetP2X purinoceptor 7(Homo sapiens (Human))
Takasaki University Of Health And Welfare
Curated by ChEMBL
Takasaki University Of Health And Welfare
Curated by ChEMBL
Affinity DataIC50: 2.40E+3nMAssay Description:Antagonist activity at P2X7 receptor in human RPMI-8226 cells assessed as inhibition of ATP-induced Ca2+ influx by fura-2 staining based assayMore data for this Ligand-Target Pair
TargetP2X purinoceptor 7(Homo sapiens (Human))
Takasaki University Of Health And Welfare
Curated by ChEMBL
Takasaki University Of Health And Welfare
Curated by ChEMBL
Affinity DataIC50: 3.20E+3nMAssay Description:Antagonist activity at P2X7 receptor in human RPMI-8226 cells assessed as inhibition of ATP-induced Ca2+ influx by fura-2 staining based assayMore data for this Ligand-Target Pair
TargetP2X purinoceptor 7(Homo sapiens (Human))
Takasaki University Of Health And Welfare
Curated by ChEMBL
Takasaki University Of Health And Welfare
Curated by ChEMBL
Affinity DataIC50: 3.40E+3nMAssay Description:Antagonist activity at P2X7 receptor in human RPMI-8226 cells assessed as inhibition of ATP-induced Ca2+ influx by fura-2 staining based assayMore data for this Ligand-Target Pair
TargetP2X purinoceptor 7(Homo sapiens (Human))
Takasaki University Of Health And Welfare
Curated by ChEMBL
Takasaki University Of Health And Welfare
Curated by ChEMBL
Affinity DataIC50: 3.80E+3nMAssay Description:Antagonist activity at P2X7 receptor in human RPMI-8226 cells assessed as inhibition of ATP-induced Ca2+ influx by fura-2 staining based assayMore data for this Ligand-Target Pair
TargetP2X purinoceptor 7(Homo sapiens (Human))
Takasaki University Of Health And Welfare
Curated by ChEMBL
Takasaki University Of Health And Welfare
Curated by ChEMBL
Affinity DataIC50: 4.50E+3nMAssay Description:Antagonist activity at P2X7 receptor in human RPMI-8226 cells assessed as inhibition of ATP-induced Ca2+ influx by fura-2 staining based assayMore data for this Ligand-Target Pair
TargetP2X purinoceptor 7(Homo sapiens (Human))
Takasaki University Of Health And Welfare
Curated by ChEMBL
Takasaki University Of Health And Welfare
Curated by ChEMBL
Affinity DataIC50: 5.20E+3nMAssay Description:Antagonist activity at P2X7 receptor in human RPMI-8226 cells assessed as inhibition of ATP-induced Ca2+ influx by fura-2 staining based assayMore data for this Ligand-Target Pair
TargetP2X purinoceptor 7(Homo sapiens (Human))
Takasaki University Of Health And Welfare
Curated by ChEMBL
Takasaki University Of Health And Welfare
Curated by ChEMBL
Affinity DataIC50: 5.30E+3nMAssay Description:Antagonist activity at P2X7 receptor in human RPMI-8226 cells assessed as inhibition of ATP-induced Ca2+ influx by fura-2 staining based assayMore data for this Ligand-Target Pair
TargetP2X purinoceptor 7(Homo sapiens (Human))
Takasaki University Of Health And Welfare
Curated by ChEMBL
Takasaki University Of Health And Welfare
Curated by ChEMBL
Affinity DataIC50: 6.50E+3nMAssay Description:Antagonist activity at P2X7 receptor in human RPMI-8226 cells assessed as inhibition of ATP-induced Ca2+ influx by fura-2 staining based assayMore data for this Ligand-Target Pair
TargetP2X purinoceptor 7(Homo sapiens (Human))
Takasaki University Of Health And Welfare
Curated by ChEMBL
Takasaki University Of Health And Welfare
Curated by ChEMBL
Affinity DataIC50: 7.50E+3nMAssay Description:Antagonist activity at P2X7 receptor in human RPMI-8226 cells assessed as inhibition of ATP-induced Ca2+ influx by fura-2 staining based assayMore data for this Ligand-Target Pair
TargetP2X purinoceptor 7(Homo sapiens (Human))
Takasaki University Of Health And Welfare
Curated by ChEMBL
Takasaki University Of Health And Welfare
Curated by ChEMBL
Affinity DataIC50: 7.80E+3nMAssay Description:Antagonist activity at P2X7 receptor in human RPMI-8226 cells assessed as inhibition of ATP-induced Ca2+ influx by fura-2 staining based assayMore data for this Ligand-Target Pair
TargetP2X purinoceptor 7(Homo sapiens (Human))
Takasaki University Of Health And Welfare
Curated by ChEMBL
Takasaki University Of Health And Welfare
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at P2X7 receptor in human RPMI-8226 cells assessed as inhibition of ATP-induced Ca2+ influx by fura-2 staining based assayMore data for this Ligand-Target Pair
TargetP2X purinoceptor 7(Homo sapiens (Human))
Takasaki University Of Health And Welfare
Curated by ChEMBL
Takasaki University Of Health And Welfare
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at P2X7 receptor in human RPMI-8226 cells assessed as inhibition of ATP-induced Ca2+ influx by fura-2 staining based assayMore data for this Ligand-Target Pair
TargetP2X purinoceptor 7(Homo sapiens (Human))
Takasaki University Of Health And Welfare
Curated by ChEMBL
Takasaki University Of Health And Welfare
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at P2X7 receptor in human RPMI-8226 cells assessed as inhibition of ATP-induced Ca2+ influx by fura-2 staining based assayMore data for this Ligand-Target Pair
TargetP2X purinoceptor 7(Homo sapiens (Human))
Takasaki University Of Health And Welfare
Curated by ChEMBL
Takasaki University Of Health And Welfare
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at P2X7 receptor in human RPMI-8226 cells assessed as inhibition of ATP-induced Ca2+ influx by fura-2 staining based assayMore data for this Ligand-Target Pair
TargetP2X purinoceptor 7(Homo sapiens (Human))
Takasaki University Of Health And Welfare
Curated by ChEMBL
Takasaki University Of Health And Welfare
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at P2X7 receptor in human RPMI-8226 cells assessed as inhibition of ATP-induced Ca2+ influx by fura-2 staining based assayMore data for this Ligand-Target Pair
TargetP2X purinoceptor 7(Homo sapiens (Human))
Takasaki University Of Health And Welfare
Curated by ChEMBL
Takasaki University Of Health And Welfare
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at P2X7 receptor in human RPMI-8226 cells assessed as inhibition of ATP-induced Ca2+ influx by fura-2 staining based assayMore data for this Ligand-Target Pair
TargetP2X purinoceptor 7(Homo sapiens (Human))
Takasaki University Of Health And Welfare
Curated by ChEMBL
Takasaki University Of Health And Welfare
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at P2X7 receptor in human RPMI-8226 cells assessed as inhibition of ATP-induced Ca2+ influx by fura-2 staining based assayMore data for this Ligand-Target Pair