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Found 4 Enz. Inhib. hit(s) with all data for entry = 50016028
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Riken Center For Biosystems Dynamics Research

Curated by ChEMBL
LigandPNGBDBM50591566(CHEMBL5177152)
Affinity DataIC50:  1.10E+3nMAssay Description:Antagonist activity at rat TRPV1 expressed in human HEK293 cells assessed as inhibition of capsaicin-induced influx by measuring intracellular calciu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Riken Center For Biosystems Dynamics Research

Curated by ChEMBL
LigandPNGBDBM50591565(CHEMBL5188412)
Affinity DataIC50:  1.30E+3nMAssay Description:Antagonist activity at rat TRPV1 expressed in human HEK293 cells assessed as inhibition of capsaicin-induced influx by measuring intracellular calciu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Riken Center For Biosystems Dynamics Research

Curated by ChEMBL
LigandPNGBDBM20488((2E)-3-(4-chlorophenyl)-N-(3-methoxyphenyl)prop-2-...)
Affinity DataIC50:  3.70E+3nMAssay Description:Antagonist activity at rat TRPV1 expressed in human HEK293 cells assessed as inhibition of capsaicin-induced influx by measuring intracellular calciu...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Riken Center For Biosystems Dynamics Research

Curated by ChEMBL
LigandPNGBDBM50591564(CHEMBL5179629)
Affinity DataIC50:  4.20E+3nMAssay Description:Antagonist activity at rat TRPV1 expressed in human HEK293 cells assessed as inhibition of capsaicin-induced influx by measuring intracellular calciu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed