Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50015692
LigandPNGBDBM50004566(CHEMBL268431 | 9-chloro-2-(furan-2-yl)-[1,2,4]tria...)
Affinity DataIC50: 110nMAssay Description:Inhibition of PI3Kgamma (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetCasein kinase I isoform delta(Human)
Technical University Dortmund

Curated by ChEMBL
LigandPNGBDBM50588635(CHEMBL5186013)
Affinity DataIC50: 120nMAssay Description:Inhibition of CK1delta (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
Technical University Dortmund

Curated by ChEMBL
LigandPNGBDBM50004566(CHEMBL268431 | 9-chloro-2-(furan-2-yl)-[1,2,4]tria...)
Affinity DataIC50: 140nMAssay Description:Inhibition of DNA-PK (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetCasein kinase I isoform alpha(Human)
Technical University Dortmund

Curated by ChEMBL
LigandPNGBDBM50588635(CHEMBL5186013)
Affinity DataIC50: 220nMAssay Description:Inhibition of CK1alpha (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetCasein kinase I isoform delta(Human)
Technical University Dortmund

Curated by ChEMBL
LigandPNGBDBM50004566(CHEMBL268431 | 9-chloro-2-(furan-2-yl)-[1,2,4]tria...)
Affinity DataIC50: 240nMAssay Description:Inhibition of CK1delta (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetCasein kinase I isoform epsilon(Human)
Technical University Dortmund

Curated by ChEMBL
LigandPNGBDBM50588635(CHEMBL5186013)
Affinity DataIC50: 380nMAssay Description:Inhibition of CK1epsilon (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetCasein kinase I isoform delta(Human)
Technical University Dortmund

Curated by ChEMBL
LigandPNGBDBM50588636(CHEMBL5182545)
Affinity DataIC50: 430nMAssay Description:Inhibition of CK1delta (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetCasein kinase I isoform epsilon(Human)
Technical University Dortmund

Curated by ChEMBL
LigandPNGBDBM50004566(CHEMBL268431 | 9-chloro-2-(furan-2-yl)-[1,2,4]tria...)
Affinity DataIC50: 490nMAssay Description:Inhibition of CK1epsilon (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetCasein kinase I isoform alpha(Human)
Technical University Dortmund

Curated by ChEMBL
LigandPNGBDBM50004566(CHEMBL268431 | 9-chloro-2-(furan-2-yl)-[1,2,4]tria...)
Affinity DataIC50: 820nMAssay Description:Inhibition of CK1alpha (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
LigandPNGBDBM50004566(CHEMBL268431 | 9-chloro-2-(furan-2-yl)-[1,2,4]tria...)
Affinity DataIC50: 970nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
LigandPNGBDBM50004566(CHEMBL268431 | 9-chloro-2-(furan-2-yl)-[1,2,4]tria...)
Affinity DataIC50: 1.28E+3nMAssay Description:Inhibition of PI3Kalpha (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetCasein kinase I isoform epsilon(Human)
Technical University Dortmund

Curated by ChEMBL
LigandPNGBDBM50588636(CHEMBL5182545)
Affinity DataIC50: 2.07E+3nMAssay Description:Inhibition of CK1epsilon (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetCasein kinase I isoform alpha(Human)
Technical University Dortmund

Curated by ChEMBL
LigandPNGBDBM50588636(CHEMBL5182545)
Affinity DataIC50: 2.92E+3nMAssay Description:Inhibition of CK1alpha (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetCasein kinase I isoform delta(Human)
Technical University Dortmund

Curated by ChEMBL
LigandPNGBDBM50023492(5-Amino-2-furan-2-yl-[1,2,4]triazolo[1,5-c]quinazo...)
Affinity DataIC50: 3.64E+3nMAssay Description:Inhibition of CK1delta (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetCasein kinase I isoform alpha(Human)
Technical University Dortmund

Curated by ChEMBL
LigandPNGBDBM50023492(5-Amino-2-furan-2-yl-[1,2,4]triazolo[1,5-c]quinazo...)
Affinity DataIC50: 6.18E+3nMAssay Description:Inhibition of CK1alpha (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
LigandPNGBDBM50004566(CHEMBL268431 | 9-chloro-2-(furan-2-yl)-[1,2,4]tria...)
Affinity DataIC50: 8.48E+3nMAssay Description:Inhibition of PI3Kbeta (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetCasein kinase I isoform epsilon(Human)
Technical University Dortmund

Curated by ChEMBL
LigandPNGBDBM50023492(5-Amino-2-furan-2-yl-[1,2,4]triazolo[1,5-c]quinazo...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CK1epsilon (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed