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Found 14 Enz. Inhib. hit(s) with all data for entry = 50016581
TargetPlasmepsin X(Plasmodium falciparum (isolate 3D7))
Merck

Curated by ChEMBL
LigandPNGBDBM50595797(CHEMBL5171401)
Affinity DataIC50:  0.0300nMAssay Description:Inhibition of Plasmodium falciparum 3D7 HA-glms-tagged PMX using DABCYL-HSFIQEGKEE-EDANS as substrate measured after 2 hrs by FRET assayMore data for this Ligand-Target Pair
TargetPlasmepsin X(Plasmodium falciparum (isolate 3D7))
Merck

Curated by ChEMBL
LigandPNGBDBM50595792(CHEMBL5182418)
Affinity DataIC50:  0.0600nMAssay Description:Inhibition of Plasmodium falciparum 3D7 HA-glms-tagged PMX using DABCYL-HSFIQEGKEE-EDANS as substrate measured after 2 hrs by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPlasmepsin X(Plasmodium falciparum (isolate 3D7))
Merck

Curated by ChEMBL
LigandPNGBDBM50595793(CHEMBL5187792)
Affinity DataIC50:  0.0700nMAssay Description:Inhibition of Plasmodium falciparum 3D7 HA-glms-tagged PMX using DABCYL-HSFIQEGKEE-EDANS as substrate measured after 2 hrs by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPlasmepsin X(Plasmodium falciparum (isolate 3D7))
Merck

Curated by ChEMBL
LigandPNGBDBM50595794(CHEMBL5193119)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of Plasmodium falciparum 3D7 HA-glms-tagged PMX using DABCYL-HSFIQEGKEE-EDANS as substrate measured after 2 hrs by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPlasmepsin X(Plasmodium falciparum (isolate 3D7))
Merck

Curated by ChEMBL
LigandPNGBDBM50595796(CHEMBL5199100)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of Plasmodium falciparum 3D7 HA-glms-tagged PMX using DABCYL-HSFIQEGKEE-EDANS as substrate measured after 2 hrs by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPlasmepsin X(Plasmodium falciparum (isolate 3D7))
Merck

Curated by ChEMBL
LigandPNGBDBM50595795(CHEMBL5207556)
Affinity DataIC50:  0.600nMAssay Description:Inhibition of Plasmodium falciparum 3D7 HA-glms-tagged PMX using DABCYL-HSFIQEGKEE-EDANS as substrate measured after 2 hrs by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPlasmepsin IX(Plasmodium falciparum (isolate 3D7))
Merck

Curated by ChEMBL
LigandPNGBDBM50595797(CHEMBL5171401)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of Plasmodium falciparum 3D7 HA-glms-tagged PMIX using DABCYL-HSFIQEGKEE-EDANS as substrate measured after 2 hrs by FRET assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPlasmepsin X(Plasmodium falciparum (isolate 3D7))
Merck

Curated by ChEMBL
LigandPNGBDBM50595790(CHEMBL5197877)
Affinity DataIC50:  1.90nMAssay Description:Inhibition of Plasmodium falciparum 3D7 HA-glms-tagged PMX using DABCYL-HSFIQEGKEE-EDANS as substrate measured after 2 hrs by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails PubMed
TargetPlasmepsin IX(Plasmodium falciparum (isolate 3D7))
Merck

Curated by ChEMBL
LigandPNGBDBM50595793(CHEMBL5187792)
Affinity DataIC50:  2.20nMAssay Description:Inhibition of Plasmodium falciparum 3D7 HA-glms-tagged PMIX using DABCYL-HSFIQEGKEE-EDANS as substrate measured after 2 hrs by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPlasmepsin IX(Plasmodium falciparum (isolate 3D7))
Merck

Curated by ChEMBL
LigandPNGBDBM50595792(CHEMBL5182418)
Affinity DataIC50:  4.5nMAssay Description:Inhibition of Plasmodium falciparum 3D7 HA-glms-tagged PMIX using DABCYL-HSFIQEGKEE-EDANS as substrate measured after 2 hrs by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPlasmepsin X(Plasmodium falciparum (isolate 3D7))
Merck

Curated by ChEMBL
LigandPNGBDBM50595791(CHEMBL5178733)
Affinity DataIC50:  5.70nMAssay Description:Inhibition of Plasmodium falciparum 3D7 HA-glms-tagged PMX using DABCYL-HSFIQEGKEE-EDANS as substrate measured after 2 hrs by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPlasmepsin IX(Plasmodium falciparum (isolate 3D7))
Merck

Curated by ChEMBL
LigandPNGBDBM50595796(CHEMBL5199100)
Affinity DataIC50:  12nMAssay Description:Inhibition of Plasmodium falciparum 3D7 HA-glms-tagged PMIX using DABCYL-HSFIQEGKEE-EDANS as substrate measured after 2 hrs by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPlasmepsin IX(Plasmodium falciparum (isolate 3D7))
Merck

Curated by ChEMBL
LigandPNGBDBM50595794(CHEMBL5193119)
Affinity DataIC50:  24nMAssay Description:Inhibition of Plasmodium falciparum 3D7 HA-glms-tagged PMIX using DABCYL-HSFIQEGKEE-EDANS as substrate measured after 2 hrs by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPlasmepsin IX(Plasmodium falciparum (isolate 3D7))
Merck

Curated by ChEMBL
LigandPNGBDBM50595795(CHEMBL5207556)
Affinity DataIC50:  68nMAssay Description:Inhibition of Plasmodium falciparum 3D7 HA-glms-tagged PMIX using DABCYL-HSFIQEGKEE-EDANS as substrate measured after 2 hrs by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed