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Found 21 Enz. Inhib. hit(s) with all data for entry = 50017482
TargetB-cell lymphoma 6 protein(Homo sapiens)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50602185(CHEMBL5184651)
Affinity DataIC50:  8.90nMAssay Description:Binding affinity to BCL6 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetB-cell lymphoma 6 protein(Homo sapiens)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50602183(CHEMBL5178494)
Affinity DataIC50:  10nMAssay Description:Inhibition of D2-SMRT peptide binding to human BCL6 BTB-POZ domain incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetB-cell lymphoma 6 protein(Homo sapiens)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50602183(CHEMBL5178494)
Affinity DataIC50:  25nMAssay Description:Displacement AF647-NCOR peptide from human BCL6 BTB-POZ domain incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetB-cell lymphoma 6 protein(Homo sapiens)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50602183(CHEMBL5178494)
Affinity DataIC50:  25nMAssay Description:Displacement AF647-BCOR peptide from human BCL6 BTB-POZ domain incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetB-cell lymphoma 6 protein(Homo sapiens)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50602186(CHEMBL5207356)
Affinity DataIC50:  120nMAssay Description:Binding affinity to BCL6 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetB-cell lymphoma 6 protein(Homo sapiens)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50266780(CHEMBL4077392)
Affinity DataIC50:  480nMAssay Description:Binding affinity to BCL6 BTB domain (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetB-cell lymphoma 6 protein(Homo sapiens)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50266780(CHEMBL4077392)
Affinity DataIC50:  8.60E+3nMAssay Description:Binding affinity to BCL6 BTB domain (unknown origin) by mammalian two hybrid assayMore data for this Ligand-Target Pair
TargetB-cell lymphoma 6 protein(Homo sapiens)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50602184(CHEMBL1721570)
Affinity DataIC50:  8.30E+5nMAssay Description:Binding affinity to BCL6 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetB-cell lymphoma 6 protein(Homo sapiens)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50602181(CHEMBL5195169)
Affinity DataKd:  1.29E+5nMAssay Description:Binding affinity to recombinant RED-NHS labelled BCL6 BTB domain (unknown origin) incubated for 10 mins by microscale thermophoresis analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetB-cell lymphoma 6 protein(Homo sapiens)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50602182(CHEMBL5202768)
Affinity DataKd:  7.00E+3nMAssay Description:Binding affinity to recombinant RED-NHS labelled BCL6 BTB domain (unknown origin) incubated for 10 mins by microscale thermophoresis analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetB-cell lymphoma 6 protein(Homo sapiens)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50266782(Amanozine | Amenozine)
Affinity DataKd:  1.20E+6nMAssay Description:Binding affinity to BCL6 BTB domain (unknown origin) by SPR analysisMore data for this Ligand-Target Pair
TargetB-cell lymphoma 6 protein(Homo sapiens)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50546199(CHEMBL4751268)
Affinity DataKd:  1.80E+4nMAssay Description:Binding affinity to BCL6 BTB domain (5 to 129 residues) (unknown origin) expressed in Escherichia coli using 5-TAMRA-RSEIISTAPSSWVVPGP as substrate i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetB-cell lymphoma 6 protein(Homo sapiens)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50546199(CHEMBL4751268)
Affinity DataKd:  2.00E+4nMAssay Description:Binding affinity to BCL6 BTB domain (5 to 129 residues) (unknown origin) expressed in Escherichia coli by SPR analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetB-cell lymphoma 6 protein(Homo sapiens)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50602179(CHEMBL5204980)
Affinity DataKd:  1.37E+3nMAssay Description:Inhibition of BCL6 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetB-cell lymphoma 6 protein(Homo sapiens)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50602180(CHEMBL5195604)
Affinity DataKd:  0.600nMAssay Description:Binding affinity to BCL6 BTB domain (unknown origin) by SPR analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetB-cell lymphoma 6 protein(Homo sapiens)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50602179(CHEMBL5204980)
Affinity DataKd:  1.61E+3nMAssay Description:Binding affinity to BCL6 BTB domain (unknown origin) by SPR analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetB-cell lymphoma 6 protein(Homo sapiens)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50266780(CHEMBL4077392)
Affinity DataKd:  78nMAssay Description:Binding affinity to BCL6 BTB domain (unknown origin) by SPR analysisMore data for this Ligand-Target Pair
TargetB-cell lymphoma 6 protein(Homo sapiens)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50602178(CHEMBL5186766)
Affinity DataKd:  1.02E+4nMAssay Description:Binding affinity to wild type full length BCL6 BTB domain having SMRT BBD motif sequence (unknown origin) transfected in human HEK293 cells by electr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetB-cell lymphoma 6 protein(Homo sapiens)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50602180(CHEMBL5195604)
Affinity DataKd:  1nMAssay Description:Inhibition of FLAG tagged human BCL6 (5 to 129 residues) by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetB-cell lymphoma 6 protein(Homo sapiens)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50602181(CHEMBL5195169)
Affinity DataKd:  1.38E+5nMAssay Description:Binding affinity to BCL6 BTB domain (unknown origin) by NMR analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetB-cell lymphoma 6 protein(Homo sapiens)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50366287(CHEMBL4175189)
Affinity DataKd:  3.20E+6nMAssay Description:Binding affinity to BCL6 BTB domain (unknown origin) by NMR analysisMore data for this Ligand-Target Pair