Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50019169
TargetOxysterols receptor LXR-beta(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM19993(CHEMBL62136 | [3H]T0901317 | T 0901317 | N-[4-(1,1...)
Affinity DataEC50:  220nMAssay Description:Agonist activity at LXRbeta (unknown origin) transfected in HEK293T cells incubated for 20 hrs by luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetOxysterols receptor LXR-alpha(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM19993(CHEMBL62136 | [3H]T0901317 | T 0901317 | N-[4-(1,1...)
Affinity DataEC50:  250nMAssay Description:Agonist activity at LXRalpha (unknown origin) transfected in HEK293T cells incubated for 20 hrs by luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetOxysterols receptor LXR-beta(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50616101(CHEMBL5431163)
Affinity DataEC50:  300nMAssay Description:Agonist activity at LXRbeta (unknown origin) transfected in HEK293T cells incubated for 20 hrs by luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50616101(CHEMBL5431163)
Affinity DataEC50:  810nMAssay Description:Agonist activity at LXRalpha (unknown origin) transfected in HEK293T cells incubated for 20 hrs by luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed