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Report error Found 56 Enz. Inhib. hit(s) with all data for entry = 50020128
Target5'-nucleotidase(Human)
Federal University of Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM554453(US11332492, Example 2)
Affinity DataIC50: 0.0500nMAssay Description:Inhibition of human CD73More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5'-nucleotidase(Human)
Federal University of Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM554453(US11332492, Example 2)
Affinity DataIC50: 0.0510nMAssay Description:Inhibition of human CD73 expressed in A-375 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5'-nucleotidase(Human)
Federal University of Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50527135(CHEMBL4452072)
Affinity DataKi:  0.318nMAssay Description:Binding affinity to human recombinant CD73 assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
Target5'-nucleotidase(Human)
Federal University of Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50546335(CHEMBL4755577)
Affinity DataKi:  2.20nMAssay Description:Binding affinity to human recombinant CD73 assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
Target5'-nucleotidase(Human)
Federal University of Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50626488(CHEMBL5402552)
Affinity DataKi:  5nMAssay Description:Binding affinity to C-terminal His6-tagged human recombinant CD73 in HEK293 cells assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5'-nucleotidase(Human)
Federal University of Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50271162(CHEMBL4127683)
Affinity DataIC50: 15nMAssay Description:Inhibition of human recombinant CD73More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5'-nucleotidase(Human)
Federal University of Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50626463(CHEMBL5405024)
Affinity DataIC50: 160nMAssay Description:Inhibition of human N-terminal Ecto-5'-nucleotidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5'-nucleotidase(Human)
Federal University of Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50626476(CHEMBL5396784)
Affinity DataIC50: 180nMAssay Description:Inhibition of human N-terminal Ecto-5'-nucleotidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5'-nucleotidase(Human)
Federal University of Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50626487(CHEMBL5421717)
Affinity DataKi:  185nMAssay Description:Binding affinity to recombinant human CD73 expressed in Sf9 cells preincubated for 25 mins and measured after 30 mins by liquid scintillation methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5'-nucleotidase(Mouse)
Federal University of Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM223080((E)-N'-(1-(3-(4-fluorophenyl)-5-phenyl-4,5-dih...)
Affinity DataIC50: 190nMAssay Description:Inhibition of mouse Ecto-5'-nucleotidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5'-nucleotidase(Mouse)
Federal University of Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50626492(CHEMBL3211645)
Affinity DataIC50: 210nMAssay Description:Inhibition of mouse Ecto-5'-nucleotidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5'-nucleotidase(Mouse)
Federal University of Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50626490(CHEMBL5410323)
Affinity DataIC50: 230nMAssay Description:Inhibition of mouse Ecto-5'-nucleotidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5'-nucleotidase(Human)
Federal University of Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50626469(CHEMBL5428233)
Affinity DataIC50: 250nMAssay Description:Inhibition of human N-terminal Ecto-5'-nucleotidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Human)
Federal University of Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50626489(CHEMBL5399001)
Affinity DataIC50: 250nMAssay Description:Inhibition of human TNAPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5'-nucleotidase(Human)
Federal University of Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50626475(CHEMBL5410463)
Affinity DataIC50: 280nMAssay Description:Inhibition of human N-terminal Ecto-5'-nucleotidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5'-nucleotidase(Human)
Federal University of Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50626462(CHEMBL5430511)
Affinity DataIC50: 280nMAssay Description:Inhibition of human N-terminal Ecto-5'-nucleotidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5'-nucleotidase(Human)
Federal University of Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50626470(CHEMBL1438157)
Affinity DataIC50: 290nMAssay Description:Inhibition of human N-terminal Ecto-5'-nucleotidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5'-nucleotidase(Human)
Federal University of Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50626494(CHEMBL5411508)
Affinity DataIC50: 290nMAssay Description:Inhibition of human recombinant Ecto-5'-nucleotidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5'-nucleotidase(Human)
Federal University of Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50626471(CHEMBL5398467)
Affinity DataIC50: 320nMAssay Description:Inhibition of human N-terminal Ecto-5'-nucleotidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5'-nucleotidase(Human)
Federal University of Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50561938(CHEMBL4746633)
Affinity DataIC50: 320nMAssay Description:Inhibition of human Ecto-5'-nucleotidase preincubated for 10 mins and measured after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5'-nucleotidase(Human)
Federal University of Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50626472(CHEMBL5406398)
Affinity DataIC50: 320nMAssay Description:Inhibition of human N-terminal Ecto-5'-nucleotidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5'-nucleotidase(Human)
Federal University of Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50626473(CHEMBL5420104)
Affinity DataIC50: 320nMAssay Description:Inhibition of human N-terminal Ecto-5'-nucleotidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5'-nucleotidase(Human)
Federal University of Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50626474(CHEMBL5417269)
Affinity DataIC50: 320nMAssay Description:Inhibition of human N-terminal Ecto-5'-nucleotidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5'-nucleotidase(Human)
Federal University of Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50179358(CHEMBL1206141)
Affinity DataKi:  451nMAssay Description:Binding affinity to recombinant human CD73 expressed in Sf9 cells preincubated for 25 mins and measured after 30 mins by liquid scintillation methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5'-nucleotidase(Human)
Federal University of Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50626503(CHEMBL5409919)
Affinity DataKi:  460nMAssay Description:Binding affinity to human recombinant Ecto-5'-nucleotidase assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5'-nucleotidase(Human)
Federal University of Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50626504(CHEMBL5438974)
Affinity DataKi:  460nMAssay Description:Binding affinity to human recombinant Ecto-5'-nucleotidase assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5'-nucleotidase(Human)
Federal University of Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50626495(CHEMBL5438317)
Affinity DataKi:  530nMAssay Description:Binding affinity to human recombinant Ecto-5'-nucleotidase assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5'-nucleotidase(Human)
Federal University of Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50626496(CHEMBL5403331)
Affinity DataKi:  530nMAssay Description:Binding affinity to human recombinant Ecto-5'-nucleotidase assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5'-nucleotidase(Human)
Federal University of Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50626499(CHEMBL1436168)
Affinity DataKi:  530nMAssay Description:Binding affinity to human recombinant Ecto-5'-nucleotidase assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5'-nucleotidase(Human)
Federal University of Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50626500(CHEMBL5432792)
Affinity DataKi:  530nMAssay Description:Binding affinity to human recombinant Ecto-5'-nucleotidase assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5'-nucleotidase(Human)
Federal University of Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50626497(CHEMBL5406328)
Affinity DataKi:  530nMAssay Description:Binding affinity to human recombinant Ecto-5'-nucleotidase assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5'-nucleotidase(Human)
Federal University of Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50626498(CHEMBL5405002)
Affinity DataKi:  530nMAssay Description:Binding affinity to human recombinant Ecto-5'-nucleotidase assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5'-nucleotidase(Human)
Federal University of Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50626501(TCMDC-123486 | GNF-Pf-4694 | MMV665943 | SJ0001107...)
Affinity DataKi:  530nMAssay Description:Binding affinity to human recombinant Ecto-5'-nucleotidase assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5'-nucleotidase(Human)
Federal University of Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50626502(CHEMBL5421860)
Affinity DataKi:  530nMAssay Description:Binding affinity to human recombinant Ecto-5'-nucleotidase assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5'-nucleotidase(Rat)
Federal University of Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50626464(CHEMBL5406908)
Affinity DataIC50: 640nMAssay Description:Inhibition of rat Ecto-5'-nucleotidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5'-nucleotidase(Mouse)
Federal University of Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50626491(CHEMBL3192470)
Affinity DataIC50: 680nMAssay Description:Inhibition of mouse Ecto-5'-nucleotidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5'-nucleotidase(Human)
Federal University of Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50626486(CHEMBL5437993)
Affinity DataKi:  831nMAssay Description:Binding affinity to recombinant human CD73 expressed in Sf9 cells preincubated for 25 mins and measured after 30 mins by liquid scintillation methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5'-nucleotidase(Human)
Federal University of Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50626485(CHEMBL5403535)
Affinity DataIC50: 860nMAssay Description:Inhibition of recombinant CD73 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5'-nucleotidase(Human)
Federal University of Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50626465(CHEMBL5436365)
Affinity DataIC50: 1.13E+3nMAssay Description:Inhibition of human N-terminal Ecto-5'-nucleotidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5'-nucleotidase(Human)
Federal University of Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50626478(CHEMBL5404987)
Affinity DataIC50: 1.14E+3nMAssay Description:Inhibition of human N-terminal Ecto-5'-nucleotidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5'-nucleotidase(Human)
Federal University of Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50626466(CHEMBL5403114)
Affinity DataIC50: 1.19E+3nMAssay Description:Inhibition of human N-terminal Ecto-5'-nucleotidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5'-nucleotidase(Human)
Federal University of Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50626467(CHEMBL5418144)
Affinity DataIC50: 1.72E+3nMAssay Description:Inhibition of human N-terminal Ecto-5'-nucleotidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5'-nucleotidase(Human)
Federal University of Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50626468(CHEMBL5402282)
Affinity DataIC50: 1.78E+3nMAssay Description:Inhibition of human N-terminal Ecto-5'-nucleotidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5'-nucleotidase(Mouse)
Federal University of Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50626478(CHEMBL5404987)
Affinity DataIC50: 1.93E+3nMAssay Description:Inhibition of mouse Ecto-5'-nucleotidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5'-nucleotidase(Human)
Federal University of Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50626477(CHEMBL5439958)
Affinity DataIC50: 2.69E+3nMAssay Description:Inhibition of human N-terminal Ecto-5'-nucleotidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5'-nucleotidase(Human)
Federal University of Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50353724(CHEMBL149463)
Affinity DataIC50: 4.66E+3nMAssay Description:Inhibition of human recombinant Ecto-5'-nucleotidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5'-nucleotidase(Human)
Federal University of Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50626484(CHEMBL5415729)
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of recombinant CD73 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5'-nucleotidase(Human)
Federal University of Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50626493(CHEMBL5436167)
Affinity DataIC50: 6.20E+3nMAssay Description:Inhibition of human recombinant Ecto-5'-nucleotidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5'-nucleotidase(Human)
Federal University of Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50626480(CHEMBL5425035)
Affinity DataIC50: 6.72E+3nMAssay Description:Inhibition of human recombinant CD73More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5'-nucleotidase(Mouse)
Federal University of Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM192657(N’-(4-methoxyphenylmethylene)benzohydrazide (...)
Affinity DataIC50: 1.38E+4nMAssay Description:Inhibition of mouse Ecto-5'-nucleotidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
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