Compile Data Set for Download or QSAR
Report error Found 39 Enz. Inhib. hit(s) with all data for entry = 50019215
TargetSerine/threonine-protein kinase 17B(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50239006(CHEMBL4060481)
Affinity DataKd:  8nMAssay Description:Binding affinity to DRAK2 (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase 17B(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50616760(CHEMBL5433785)
Affinity DataIC50: 10nMAssay Description:Inhibition of DRAK2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetDeath-associated protein kinase 3(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50616768(CHEMBL5407013)
Affinity DataKi: >10nMAssay Description:Inhibition of human recombinant GST-fused DAPK3 (1 to 320 residues) expressed in Escherichia coli BL21 (DE3) assessed as inhibition constant using MY...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase 17B(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50239006(CHEMBL4060481)
Affinity DataIC50: 29nMAssay Description:Inhibition of DRAK2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetDeath-associated protein kinase 1(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50239006(CHEMBL4060481)
Affinity DataKd:  54nMAssay Description:Binding affinity to DAPK1 (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase pim-3(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50616765(CHEMBL5425555)
Affinity DataKi:  72nMAssay Description:Inhibition of human full length-His6 tagged PIM3 (1 to 326 residues) expressed in Escherichia coli BL21 (DE3) assessed as inhibition constant using R...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetDeath-associated protein kinase 2(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM104065(HS38)
Affinity DataKd:  79nMAssay Description:Binding affinity to DAPK2 (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase 17A(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50616760(CHEMBL5433785)
Affinity DataIC50: 100nMAssay Description:Inhibition of DRAK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetDeath-associated protein kinase 3(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50616767(CHEMBL5410656)
Affinity DataKi:  119nMAssay Description:Inhibition of human recombinant GST-fused DAPK3 (1 to 320 residues) expressed in Escherichia coli BL21 (DE3) assessed as inhibition constant using MY...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetDeath-associated protein kinase 3(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50616766(CHEMBL5413882)
Affinity DataKi:  126nMAssay Description:Inhibition of human recombinant GST-fused DAPK3 (1 to 320 residues) expressed in Escherichia coli BL21 (DE3) assessed as inhibition constant using MY...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase pim-3(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM104065(HS38)
Affinity DataIC50: 200nMAssay Description:Inhibition of PIM3 (unknown origin) by (33P-ATP) filter-binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetDeath-associated protein kinase 1(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM104065(HS38)
Affinity DataIC50: 200nMAssay Description:Inhibition of DAPK1 (unknown origin) by (33P-ATP) filter-binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase pim-2(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM104065(HS38)
Affinity DataKi:  208nMAssay Description:Inhibition of human full length-His6 tagged PIM2 (1 to 311 residues) expressed in Escherichia coli BL21 (DE3) assessed as inhibition constant using R...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetDeath-associated protein kinase 1(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50616759(CHEMBL5407750)
Affinity DataIC50: 247nMAssay Description:Inhibition of DAPK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase 17B(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50616770(CHEMBL5401514)
Affinity DataKd:  250nMAssay Description:Binding affinity to DRAK2 (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetDeath-associated protein kinase 3(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM104065(HS38)
Affinity DataKi:  260nMAssay Description:Inhibition of human recombinant GST-fused DAPK3 (1 to 320 residues) expressed in Escherichia coli BL21 (DE3) assessed as inhibition constant using MY...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetDeath-associated protein kinase 3(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM104065(HS38)
Affinity DataKd:  280nMAssay Description:Binding affinity to DAPK3 (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetDeath-associated protein kinase 1(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM104065(HS38)
Affinity DataKd:  300nMAssay Description:Binding affinity to DAPK1 (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetDeath-associated protein kinase 3(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50616760(CHEMBL5433785)
Affinity DataIC50: 310nMAssay Description:Inhibition of DAPK3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetDeath-associated protein kinase 3(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50616765(CHEMBL5425555)
Affinity DataKi:  315nMAssay Description:Inhibition of human recombinant GST-fused DAPK3 (1 to 320 residues) expressed in Escherichia coli BL21 (DE3) assessed as inhibition constant using MY...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetDeath-associated protein kinase 1(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50616760(CHEMBL5433785)
Affinity DataIC50: 370nMAssay Description:Inhibition of DAPK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetDeath-associated protein kinase 1(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM67454(MLS002473304 | purpurin | 1,2,4-tris(oxidanyl)anth...)
Affinity DataIC50: 890nMAssay Description:Inhibition of DAPK1 (1 to 285 residues) (unknown origin) expressed in Escherichia coli using KKLNRTLSFAEPG as substrate in presence of ATP by fluoro-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetSerine/threonine-protein kinase pim-3(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50616767(CHEMBL5410656)
Affinity DataKi:  1.07E+3nMAssay Description:Inhibition of human full length-His6 tagged PIM3 (1 to 326 residues) expressed in Escherichia coli BL21 (DE3) assessed as inhibition constant using R...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50616765(CHEMBL5425555)
Affinity DataKi:  1.48E+3nMAssay Description:Inhibition of human full length-His6 tagged PIM1 (1 to 312 residues) expressed in Escherichia coli BL21 (DE3) assessed as inhibition constant using R...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase pim-3(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50616766(CHEMBL5413882)
Affinity DataKi:  2.50E+3nMAssay Description:Inhibition of human full length-His6 tagged PIM3 (1 to 326 residues) expressed in Escherichia coli BL21 (DE3) assessed as inhibition constant using R...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetDeath-associated protein kinase 1(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50616763(CHEMBL5412508)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of DAPK1 (unknown origin) in presence of 33P-ATP radiolabeled kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM104065(HS38)
Affinity DataKi:  2.94E+3nMAssay Description:Inhibition of human full length-His6 tagged PIM1 (1 to 312 residues) expressed in Escherichia coli BL21 (DE3) assessed as inhibition constant using R...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetDeath-associated protein kinase 1(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50206434(1,2-dihydroxyanthracene-9,10-dione | alizarin | 1,...)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of DAPK1 (1 to 285 residues) (unknown origin) expressed in Escherichia coli using KKLNRTLSFAEPG as substrate in presence of ATP by fluoro-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetDeath-associated protein kinase 1(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50616762(CHEMBL5426378)
Affinity DataIC50: 5.90E+3nMAssay Description:Inhibition of DAPK1 (unknown origin) in presence of 33P-ATP radiolabeled kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50616766(CHEMBL5413882)
Affinity DataKi:  6.31E+3nMAssay Description:Inhibition of human full length-His6 tagged PIM1 (1 to 312 residues) expressed in Escherichia coli BL21 (DE3) assessed as inhibition constant using R...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50616767(CHEMBL5410656)
Affinity DataKi:  6.48E+3nMAssay Description:Inhibition of human full length-His6 tagged PIM1 (1 to 312 residues) expressed in Escherichia coli BL21 (DE3) assessed as inhibition constant using R...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetDeath-associated protein kinase 1(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50616764(CHEMBL5028838)
Affinity DataIC50: 9.60E+3nMAssay Description:Inhibition of DAPK1 (1 to 285 residues) (unknown origin) expressed in Escherichia coli using KKLNRTLSFAEPG as substrate in presence of ATP by fluoro-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase 17B(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50616769(CHEMBL5400845)
Affinity DataIC50: 1.17E+4nMAssay Description:Inhibition of recombinant GST-tagged DRAK2 (unknown origin) by promega ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetDeath-associated protein kinase 1(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50616758(CHEMBL5398489)
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of DAPK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase pim-2(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50616765(CHEMBL5425555)
Affinity DataKi:  1.73E+4nMAssay Description:Inhibition of human full length-His6 tagged PIM2 (1 to 311 residues) expressed in Escherichia coli BL21 (DE3) assessed as inhibition constant using R...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetDeath-associated protein kinase 1(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50616761(CHEMBL5439149)
Affinity DataIC50: 2.30E+4nMAssay Description:Inhibition of DAPK1 (unknown origin) in presence of 33P-ATP radiolabeled kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase pim-3(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM104065(HS38)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human full length-His6 tagged PIM3 (1 to 326 residues) expressed in Escherichia coli BL21 (DE3) assessed as inhibition constant using R...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase pim-2(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50616766(CHEMBL5413882)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human full length-His6 tagged PIM2 (1 to 311 residues) expressed in Escherichia coli BL21 (DE3) assessed as inhibition constant using R...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase pim-2(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50616767(CHEMBL5410656)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human full length-His6 tagged PIM2 (1 to 311 residues) expressed in Escherichia coli BL21 (DE3) assessed as inhibition constant using R...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed