Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 50019834
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Xuzhou Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50396352BDBM50396352(CHEMBL2170062)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]-pentazocine from sigma1 receptor in guinea pig brain membrane at 1 uM by liquid scintillation counting analysis relative to cont...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Xuzhou Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50623542BDBM50623542(CHEMBL5440801)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]-pentazocine from sigma1 receptor in guinea pig brain membrane at 1 uM by liquid scintillation counting analysis relative to cont...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Xuzhou Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50623540BDBM50623540(CHEMBL5415318)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]-pentazocine from sigma1 receptor in guinea pig brain membrane at 1 uM by liquid scintillation counting analysis relative to cont...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
Xuzhou Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50623542BDBM50623542(CHEMBL5440801)
Affinity DataIC50: 19nMAssay Description:Antagonist activity at sigma1 receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Xuzhou Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50623539BDBM50623539(CHEMBL5415799)
Affinity DataKi:  27nMAssay Description:Displacement of [3H]-pentazocine from sigma1 receptor in guinea pig brain membrane at 1 uM by liquid scintillation counting analysis relative to cont...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Xuzhou Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50623541BDBM50623541(CHEMBL5405189)
Affinity DataKi:  33nMAssay Description:Displacement of [3H]-pentazocine from sigma1 receptor in guinea pig brain membrane at 1 uM by liquid scintillation counting analysis relative to cont...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Xuzhou Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50623536BDBM50623536(CHEMBL5394556)
Affinity DataKi:  35nMAssay Description:Displacement of [3H]-pentazocine from sigma1 receptor in guinea pig brain membrane at 1 uM by liquid scintillation counting analysis relative to cont...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Xuzhou Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50623542BDBM50623542(CHEMBL5440801)
Affinity DataKi:  37nMAssay Description:Displacement of [3H]-pentazocine from sigma1 receptor in guinea pig brain membrane assessed as inhibition constant in presence of phenytoin by liquid...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Xuzhou Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50623533BDBM50623533(CHEMBL5399552)
Affinity DataKi:  39nMAssay Description:Displacement of [3H]-pentazocine from sigma1 receptor in guinea pig brain membrane at 1 uM by liquid scintillation counting analysis relative to cont...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Xuzhou Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50623528BDBM50623528(CHEMBL5393921)
Affinity DataKi:  41nMAssay Description:Displacement of [3H]-pentazocine from sigma1 receptor in guinea pig brain membrane at 1 uM by liquid scintillation counting analysis relative to cont...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Xuzhou Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50623530BDBM50623530(CHEMBL5430839)
Affinity DataKi:  43nMAssay Description:Displacement of [3H]-pentazocine from sigma1 receptor in guinea pig brain membrane at 1 uM by liquid scintillation counting analysis relative to cont...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Xuzhou Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50623538BDBM50623538(CHEMBL5412845)
Affinity DataKi:  45nMAssay Description:Displacement of [3H]-pentazocine from sigma1 receptor in guinea pig brain membrane at 1 uM by liquid scintillation counting analysis relative to cont...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Xuzhou Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50623531BDBM50623531(CHEMBL5416549)
Affinity DataKi:  48nMAssay Description:Displacement of [3H]-pentazocine from sigma1 receptor in guinea pig brain membrane at 1 uM by liquid scintillation counting analysis relative to cont...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Xuzhou Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50623525BDBM50623525(CHEMBL5417570)
Affinity DataKi:  49nMAssay Description:Displacement of [3H]-pentazocine from sigma1 receptor in guinea pig brain membrane at 1 uM by liquid scintillation counting analysis relative to cont...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Xuzhou Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50623535BDBM50623535(CHEMBL5403544)
Affinity DataKi:  50nMAssay Description:Displacement of [3H]-pentazocine from sigma1 receptor in guinea pig brain membrane at 1 uM by liquid scintillation counting analysis relative to cont...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Xuzhou Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50623529BDBM50623529(CHEMBL5403914)
Affinity DataKi:  60nMAssay Description:Displacement of [3H]-pentazocine from sigma1 receptor in guinea pig brain membrane at 1 uM by liquid scintillation counting analysis relative to cont...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Xuzhou Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50623526BDBM50623526(CHEMBL5429201)
Affinity DataKi:  61nMAssay Description:Displacement of [3H]-pentazocine from sigma1 receptor in guinea pig brain membrane at 1 uM by liquid scintillation counting analysis relative to cont...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Xuzhou Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50623534BDBM50623534(CHEMBL5432392)
Affinity DataKi:  68nMAssay Description:Displacement of [3H]-pentazocine from sigma1 receptor in guinea pig brain membrane at 1 uM by liquid scintillation counting analysis relative to cont...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Xuzhou Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50623537BDBM50623537(CHEMBL5430052)
Affinity DataKi:  84nMAssay Description:Displacement of [3H]-pentazocine from sigma1 receptor in guinea pig brain membrane at 1 uM by liquid scintillation counting analysis relative to cont...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Xuzhou Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50623524BDBM50623524(CHEMBL5405596)
Affinity DataKi:  175nMAssay Description:Displacement of [3H]-pentazocine from sigma1 receptor in guinea pig brain membrane at 1 uM by liquid scintillation counting analysis relative to cont...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Xuzhou Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50623532BDBM50623532(CHEMBL5399495)
Affinity DataKi:  181nMAssay Description:Displacement of [3H]-pentazocine from sigma1 receptor in guinea pig brain membrane at 1 uM by liquid scintillation counting analysis relative to cont...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetSigma intracellular receptor 2(Human)
Xuzhou Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50623542BDBM50623542(CHEMBL5440801)
Affinity DataIC50: 227nMAssay Description:Antagonist activity at sigma2 receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Xuzhou Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50623527BDBM50623527(CHEMBL5396839)
Affinity DataKi:  393nMAssay Description:Displacement of [3H]-pentazocine from sigma1 receptor in guinea pig brain membrane at 1 uM by liquid scintillation counting analysis relative to cont...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed