Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50019242
TargetMelanocortin receptor 4(Human)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50617059(CHEMBL5414451)
Affinity DataKi:  0.0600nMAssay Description:Displacement of sCy5-MT-I from human MC4R stably expressed in human HEK293 cells incubated for 2 hrs by Cheng-Prusoff equation based FACS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetMelanocortin receptor 4(Human)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50617058(CHEMBL5416095)
Affinity DataEC50:  0.980nMAssay Description:Agonist activity at human MC4R stably expressed in human Flp-In-293 cells assessed as cAMP accumulation incubated for 45 mins in presence of IBMX by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50617058(CHEMBL5416095)
Affinity DataEC50:  24nMAssay Description:Agonist activity at human MC1R stably expressed in human Flp-In-293 cells assessed as cAMP accumulation incubated for 45 mins in presence of IBMX by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed