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Report error Found 27 Enz. Inhib. hit(s) with all data for entry = 50035657
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rat)
Beecham Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM22372(4-[(2R,3S)-4-(3,4-dihydroxyphenyl)-2,3-dimethylbut...)
Affinity DataIC50:  140nMAssay Description:In vitro inhibition of RBL-1 5-lipoxygenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPolyunsaturated fatty acid 5-lipoxygenase(Rat)
Beecham Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50024851(7-Methyl-2-trifluoromethyl-1H-benzoimidazol-4-ol |...)
Affinity DataIC50:  250nMAssay Description:In vitro inhibition of RBL-1 5-lipoxygenase; Value ranges from 0.18-0.31More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPolyunsaturated fatty acid 5-lipoxygenase(Rat)
Beecham Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50000540(1-(3-Trifluoromethyl-phenyl)-4,5-dihydro-1H-pyrazo...)
Affinity DataIC50:  890nMAssay Description:In vitro inhibition of RBL-1 5-lipoxygenase; Value ranges from 0.72-1.07More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPolyunsaturated fatty acid 5-lipoxygenase(Rat)
Beecham Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50367452(CHEMBL1743607)
Affinity DataIC50:  1.00E+3nMAssay Description:In vitro inhibition of RBL-1 5-lipoxygenase; Value ranges from 0.3-1.6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPolyunsaturated fatty acid 5-lipoxygenase(Rat)
Beecham Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50024863(2-Benzyl-7-methyl-1H-benzoimidazol-4-ol | CHEMBL67...)
Affinity DataIC50:  1.20E+3nMAssay Description:In vitro inhibition of RBL-1 5-lipoxygenase; Value ranges from 0.4-2.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPolyunsaturated fatty acid 5-lipoxygenase(Rat)
Beecham Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50367457(CHEMBL1202795)
Affinity DataIC50:  1.20E+3nMAssay Description:In vitro inhibition of RBL-1 5-lipoxygenase; Value ranges from 1.0-1.5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPolyunsaturated fatty acid 5-lipoxygenase(Rat)
Beecham Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50367451(CHEMBL1202802)
Affinity DataIC50:  1.30E+3nMAssay Description:In vitro inhibition of RBL-1 5-lipoxygenase; Value ranges from 1.0-1.7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPolyunsaturated fatty acid 5-lipoxygenase(Rat)
Beecham Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50024850(2-Benzyl-5-tert-butyl-7-methyl-1H-benzoimidazol-4-...)
Affinity DataIC50:  1.30E+3nMAssay Description:In vitro inhibition of RBL-1 5-lipoxygenase; Value ranges from 1.1-1.6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPolyunsaturated fatty acid 5-lipoxygenase(Rat)
Beecham Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50367460(CHEMBL1202809)
Affinity DataIC50:  1.70E+3nMAssay Description:In vitro inhibition of RBL-1 5-lipoxygenase; Value ranges from 1.0-2.4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPolyunsaturated fatty acid 5-lipoxygenase(Rat)
Beecham Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50006811(2-(12-Hydroxy-5,10-dodecadiynyl)-3,5,6-trimethyl-p...)
Affinity DataIC50:  2.00E+3nMAssay Description:In vitro inhibition of RBL-1 5-lipoxygenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPolyunsaturated fatty acid 5-lipoxygenase(Rat)
Beecham Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50009004((phenidone)1-Phenyl-pyrazolidin-3-one | 1-Phenyl-p...)
Affinity DataIC50:  2.10E+3nMAssay Description:In vitro inhibition of RBL-1 5-lipoxygenase; Value ranges from 1.07-5.54More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPolyunsaturated fatty acid 5-lipoxygenase(Rat)
Beecham Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50367462(CHEMBL1202798)
Affinity DataIC50:  2.10E+3nMAssay Description:In vitro inhibition of RBL-1 5-lipoxygenase; Value ranges from 1.7-2.6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPolyunsaturated fatty acid 5-lipoxygenase(Rat)
Beecham Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50367454(CHEMBL1202796)
Affinity DataIC50:  2.10E+3nMAssay Description:In vitro inhibition of RBL-1 5-lipoxygenase; Value ranges from 1.3-2.8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPolyunsaturated fatty acid 5-lipoxygenase(Rat)
Beecham Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50367466(CHEMBL1202812)
Affinity DataIC50:  2.10E+3nMAssay Description:In vitro inhibition of RBL-1 5-lipoxygenase; Value ranges from 1.9-2.4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPolyunsaturated fatty acid 5-lipoxygenase(Rat)
Beecham Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50367456(CHEMBL1202797)
Affinity DataIC50:  2.20E+3nMAssay Description:In vitro inhibition of RBL-1 5-lipoxygenase; Value ranges from 1.4-3.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPolyunsaturated fatty acid 5-lipoxygenase(Rat)
Beecham Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50367463(CHEMBL1202811)
Affinity DataIC50:  2.20E+3nMAssay Description:In vitro inhibition of RBL-1 5-lipoxygenase; Value ranges from 0.9-4.0More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPolyunsaturated fatty acid 5-lipoxygenase(Rat)
Beecham Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50367455(CHEMBL1202805)
Affinity DataIC50:  2.30E+3nMAssay Description:In vitro inhibition of RBL-1 5-lipoxygenase; Value ranges from 1.8-2.8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPolyunsaturated fatty acid 5-lipoxygenase(Rat)
Beecham Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50024845(7-Methyl-2-(4-methyl-benzyl)-1H-benzoimidazol-4-ol...)
Affinity DataIC50:  2.54E+3nMAssay Description:In vitro inhibition of RBL-1 5-lipoxygenase; Value ranges from 2.46-2.63More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPolyunsaturated fatty acid 5-lipoxygenase(Rat)
Beecham Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50367459(CHEMBL1202810)
Affinity DataIC50:  3.00E+3nMAssay Description:In vitro inhibition of RBL-1 5-lipoxygenase; Value ranges from 2.3-.8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPolyunsaturated fatty acid 5-lipoxygenase(Rat)
Beecham Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50367458(CHEMBL1202806)
Affinity DataIC50:  3.30E+3nMAssay Description:In vitro inhibition of RBL-1 5-lipoxygenase; Value ranges from 1.8-5.7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPolyunsaturated fatty acid 5-lipoxygenase(Rat)
Beecham Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50367461(CHEMBL1202808)
Affinity DataIC50:  3.40E+3nMAssay Description:In vitro inhibition of RBL-1 5-lipoxygenase; Value ranges from 3.3-3.5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPolyunsaturated fatty acid 5-lipoxygenase(Rat)
Beecham Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50024854(7-Methyl-2-pyridin-3-ylmethyl-1H-benzoimidazol-4-o...)
Affinity DataIC50:  5.00E+3nMAssay Description:In vitro inhibition of RBL-1 5-lipoxygenase; Value ranges from 4.0-6.4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPolyunsaturated fatty acid 5-lipoxygenase(Rat)
Beecham Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50367465(CHEMBL1202800)
Affinity DataIC50:  5.20E+3nMAssay Description:In vitro inhibition of RBL-1 5-lipoxygenase; Value ranges from 3.8-7.1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPolyunsaturated fatty acid 5-lipoxygenase(Rat)
Beecham Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50367464(CHEMBL1202801)
Affinity DataIC50:  6.90E+3nMAssay Description:In vitro inhibition of RBL-1 5-lipoxygenase; Value ranges from 4.9-11.6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPolyunsaturated fatty acid 5-lipoxygenase(Rat)
Beecham Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50367453(CHEMBL1202799)
Affinity DataIC50:  9.70E+3nMAssay Description:In vitro inhibition of RBL-1 5-lipoxygenase; Value ranges from 7.5-11.8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPolyunsaturated fatty acid 5-lipoxygenase(Rat)
Beecham Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50024844(2-Benzyl-1H-benzoimidazol-4-ol | CHEMBL306680)
Affinity DataIC50:  2.00E+4nMAssay Description:In vitro inhibition of RBL-1 5-lipoxygenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPolyunsaturated fatty acid 5-lipoxygenase(Rat)
Beecham Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50024858(2-(4-Methoxy-benzyl)-1H-benzoimidazol-4-ol | CHEMB...)
Affinity DataIC50:  2.00E+4nMAssay Description:In vitro inhibition of RBL-1 5-lipoxygenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed