Compile Data Set for Download or QSAR
Report error Found 30 Enz. Inhib. hit(s) with all data for entry = 50018935
TargetBromodomain-containing protein 4(Human)
University of Maryland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50466283BDBM50466283(CHEMBL4278881)
Affinity DataKd:  28nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) assessed as dissociation constant by DiscoveRx BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Maryland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50613957BDBM50613957(CHEMBL5270205)
Affinity DataKd:  35nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) assessed as dissociation constant by DiscoveRx BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Maryland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50613948BDBM50613948(CHEMBL5270456)
Affinity DataKd:  44nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) assessed as dissociation constant by DiscoveRx BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Maryland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50613954BDBM50613954(CHEMBL5268457)
Affinity DataKd:  53nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) assessed as dissociation constant by DiscoveRx BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Maryland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50613956BDBM50613956(CHEMBL5267716)
Affinity DataKd:  54nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) assessed as dissociation constant by DiscoveRx BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Maryland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50613959BDBM50613959(CHEMBL5271263)
Affinity DataKd:  55nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) assessed as dissociation constant by DiscoveRx BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Maryland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50613960BDBM50613960(CHEMBL5280349)
Affinity DataKd:  95nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) assessed as dissociation constant by DiscoveRx BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Maryland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50613961BDBM50613961(CHEMBL5282274)
Affinity DataKd:  130nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) assessed as dissociation constant by DiscoveRx BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Maryland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50613964BDBM50613964(CHEMBL5285703)
Affinity DataKd:  170nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) assessed as dissociation constant by DiscoveRx BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Maryland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50613963BDBM50613963(CHEMBL5282421)
Affinity DataKd:  210nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) assessed as dissociation constant by DiscoveRx BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Maryland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50613958BDBM50613958(CHEMBL5272731)
Affinity DataKd:  210nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) assessed as dissociation constant by DiscoveRx BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Maryland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50613966BDBM50613966(CHEMBL5287776)
Affinity DataKd:  220nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) assessed as dissociation constant by DiscoveRx BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Maryland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50613955BDBM50613955(CHEMBL5270005)
Affinity DataKd:  250nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) assessed as dissociation constant by DiscoveRx BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Maryland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50613965BDBM50613965(CHEMBL5268057)
Affinity DataKd:  370nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) assessed as dissociation constant by DiscoveRx BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Maryland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50613962BDBM50613962(CHEMBL5269795)
Affinity DataKd:  490nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) assessed as dissociation constant by DiscoveRx BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Maryland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50613967BDBM50613967(CHEMBL5285213)
Affinity DataKd:  570nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) assessed as dissociation constant by DiscoveRx BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Maryland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50613948BDBM50613948(CHEMBL5270456)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) by Alphascreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Maryland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50613951BDBM50613951(CHEMBL5277846)
Affinity DataKd:  1.30E+3nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) assessed as dissociation constant by DiscoveRx BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Maryland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50613951BDBM50613951(CHEMBL5277846)
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) by Alphascreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Maryland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50613952BDBM50613952(CHEMBL5280039)
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) by Alphascreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Maryland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50613953BDBM50613953(CHEMBL5280986)
Affinity DataKd:  3.40E+3nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) assessed as dissociation constant by DiscoveRx BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Maryland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50613949BDBM50613949(CHEMBL5276495)
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) by Alphascreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetCytochrome P450 2C9(Human)
University of Maryland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50613948BDBM50613948(CHEMBL5270456)
Affinity DataIC50: 6.77E+3nMAssay Description:Inhibition of CYP2C9 (unknown origin) by fluorescence based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Maryland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50613952BDBM50613952(CHEMBL5280039)
Affinity DataKd:  7.40E+3nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) assessed as dissociation constant by DiscoveRx BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Maryland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50613953BDBM50613953(CHEMBL5280986)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) by Alphascreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetCytochrome P450 2C19(Human)
University of Maryland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50613948BDBM50613948(CHEMBL5270456)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CYP2C19 (unknown origin) by fluorescence based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetCytochrome P450 1A2(Human)
University of Maryland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50613948BDBM50613948(CHEMBL5270456)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CYP1A2 (unknown origin) by fluorescence based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetCytochrome P450 2D6(Human)
University of Maryland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50613948BDBM50613948(CHEMBL5270456)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CYP2D6 (unknown origin) by fluorescence based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetCytochrome P450 3A4(Human)
University of Maryland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50613948BDBM50613948(CHEMBL5270456)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin) by fluorescence based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Maryland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50613950BDBM50613950(CHEMBL5280137)
Affinity DataIC50: 1.00E+7nMAssay Description:Inhibition of BRD4 bromodomain 1/2 (unknown origin) by Alphascreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed