Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50019860
TargetGlutaminase kidney isoform, mitochondrial(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM109086(US8604016, 670 | US9938267, Cmpd ID 670 | US107935...)
Affinity DataIC50: 20nMAssay Description:Inhibition of human recombinant GLS1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetGlutaminase kidney isoform, mitochondrial(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50623848(CHEMBL4556013)
Affinity DataIC50: 100nMAssay Description:Inhibition of N-terminal His-tagged GLS1 (unknown origin) expressed in Escherichia coli BL21 (DE3) preincubated for 20 mins and measured after 2 hrsMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50385299(CHEMBL2035464 | US8592468, EbSe16)
Affinity DataIC50: 200nMAssay Description:Inhibition of C-terminal His-tagged human recombinant KGA transformed in Escherichia coli BL21 DE3 at pH 7.4 incubated for 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50623849(CHEMBL5404634)
Affinity DataIC50: 6.10E+3nMAssay Description:Inhibition of full length C terminal His-tagged human KGA expressed in Escherichia coli BL-21 DE3More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50623850(CHEMBL5423249)
Affinity DataIC50: 6.80E+3nMAssay Description:Inhibition of C-terminal His-tagged human recombinant KGA transformed in Escherichia coli BL21 DE3 at pH 7.4 incubated for 3 hrsMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed