Compile Data Set for Download or QSAR
Report error Found 22 Enz. Inhib. hit(s) with all data for entry = 50019288
TargetNeuraminidase(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Jawaharlal Nehru University

Curated by ChEMBL
LigandPNGBDBM50617615(CHEMBL5401545)
Affinity DataKi:  0.290nMAssay Description:Binding affinity to influenza A virus H1N1 (A/Norway/1758/07) neuraminidase using MUNANA as substrate assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Jawaharlal Nehru University

Curated by ChEMBL
LigandPNGBDBM50617614(CHEMBL5428414)
Affinity DataKi:  0.740nMAssay Description:Binding affinity to influenza A virus H1N1 (A/Norway/1758/07) neuraminidase using MUNANA as substrate assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Wilson-Smith/1933 H1N1...)
Jawaharlal Nehru University

Curated by ChEMBL
LigandPNGBDBM50330326((4S,5R,6R)-5-Acetylamino-4-guanidino-6-((1R,3R)-1,...)
Affinity DataIC50: 15nMAssay Description:Inhibition of influenza A virus neuraminidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Wilson-Smith/1933 H1N1...)
Jawaharlal Nehru University

Curated by ChEMBL
LigandPNGBDBM50009296(R-125489 | LANINAMIVIR)
Affinity DataIC50: 18nMAssay Description:Inhibition of influenza A virus neuraminidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Memphis/1/1971 H3N2))
Jawaharlal Nehru University

Curated by ChEMBL
LigandPNGBDBM50617625(CHEMBL5411684)
Affinity DataIC50: 19nMAssay Description:Inhibition of influenza A virus H3N2 (A/Moscow/10/99) neuraminidase using MUNANA as substrate preincubated for 30 mins followed by substrate addition...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Jawaharlal Nehru University

Curated by ChEMBL
LigandPNGBDBM50206333(CHEMBL3951068)
Affinity DataIC50: 20nMAssay Description:Inhibition of avian Influenza A virus SN 33 (H1N1) neuraminidase infected in dog MDCK cells using MU-NANA as substrate assessed as reduction in viral...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Memphis/1/1971 H3N2))
Jawaharlal Nehru University

Curated by ChEMBL
LigandPNGBDBM50206333(CHEMBL3951068)
Affinity DataIC50: 25nMAssay Description:Inhibition of avian Influenza A Taiwan 3446 2002(H3N2) neuraminidase infected in dog MDCK cells using MU-NANA as substrate assessed as reduction in v...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Wilson-Smith/1933 H1N1...)
Jawaharlal Nehru University

Curated by ChEMBL
LigandPNGBDBM50617619(CHEMBL1179074)
Affinity DataIC50: 36nMAssay Description:Inhibition of influenza A virus neuraminidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Wilson-Smith/1933 H1N1...)
Jawaharlal Nehru University

Curated by ChEMBL
LigandPNGBDBM50617620(CHEMBL1179072)
Affinity DataIC50: 45nMAssay Description:Inhibition of influenza A virus neuraminidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Memphis/1/1971 H3N2))
Jawaharlal Nehru University

Curated by ChEMBL
LigandPNGBDBM50617616(CHEMBL4459836)
Affinity DataIC50: 67nMAssay Description:Inhibition of avian Influenza A Taiwan 3446 2002(H3N2) neuraminidase infected in dog MDCK cells using MU-NANA as substrate assessed as reduction in v...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Wilson-Smith/1933 H1N1...)
Jawaharlal Nehru University

Curated by ChEMBL
LigandPNGBDBM50617617(CHEMBL1179048)
Affinity DataIC50: 73nMAssay Description:Inhibition of influenza A virus neuraminidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Jawaharlal Nehru University

Curated by ChEMBL
LigandPNGBDBM50617616(CHEMBL4459836)
Affinity DataIC50: 75nMAssay Description:Inhibition of avian Influenza A virus SN 33 (H1N1) neuraminidase infected in dog MDCK cells using MU-NANA as substrate assessed as reduction in viral...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Wilson-Smith/1933 H1N1...)
Jawaharlal Nehru University

Curated by ChEMBL
LigandPNGBDBM50617618(CHEMBL1183504)
Affinity DataIC50: 82nMAssay Description:Inhibition of influenza A virus neuraminidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Wilson-Smith/1933 H1N1...)
Jawaharlal Nehru University

Curated by ChEMBL
LigandPNGBDBM50617621(CHEMBL1183488)
Affinity DataIC50: 99nMAssay Description:Inhibition of influenza A virus neuraminidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Memphis/1/1971 H3N2))
Jawaharlal Nehru University

Curated by ChEMBL
LigandPNGBDBM50617625(CHEMBL5411684)
Affinity DataIC50: 790nMAssay Description:Inhibition of influenza A virus H3N2 (A/Moscow/10/99) harboring E119V mutant neuraminidase using MUNANA as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Memphis/1/1971 H3N2))
Jawaharlal Nehru University

Curated by ChEMBL
LigandPNGBDBM50617627(CHEMBL5419264)
Affinity DataIC50: 6.98E+3nMAssay Description:Inhibition of influenza A virus A/H3N2 neuraminidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNeuraminidase(Influenza A virus)
Jawaharlal Nehru University

Curated by ChEMBL
LigandPNGBDBM50617622(CHEMBL5411309)
Affinity DataIC50: 8.86E+3nMAssay Description:Inhibition of influenza A virus A/RI/5+/1957(H2N2) neuraminidase using 4-MU-Neu5Ac as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Memphis/1/1971 H3N2))
Jawaharlal Nehru University

Curated by ChEMBL
LigandPNGBDBM50617629(CHEMBL5429849)
Affinity DataIC50: 1.23E+4nMAssay Description:Inhibition of influenza A virus A/H3N2 neuraminidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Memphis/1/1971 H3N2))
Jawaharlal Nehru University

Curated by ChEMBL
LigandPNGBDBM50617628(CHEMBL5433667)
Affinity DataIC50: 2.70E+4nMAssay Description:Inhibition of influenza A virus A/H3N2 neuraminidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Memphis/1/1971 H3N2))
Jawaharlal Nehru University

Curated by ChEMBL
LigandPNGBDBM50617626(CHEMBL5407388)
Affinity DataIC50: 2.70E+4nMAssay Description:Inhibition of influenza A virus A/H3N2 neuraminidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNeuraminidase(Influenza A virus)
Jawaharlal Nehru University

Curated by ChEMBL
LigandPNGBDBM50617623(CHEMBL5401504)
Affinity DataIC50: 1.20E+5nMAssay Description:Inhibition of influenza A virus A/RI/5+/1957(H2N2) neuraminidase using 4-MU-Neu5Ac as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNeuraminidase(Influenza A virus)
Jawaharlal Nehru University

Curated by ChEMBL
LigandPNGBDBM50617624(CHEMBL5433388)
Affinity DataIC50: 3.16E+5nMAssay Description:Inhibition of influenza A virus A/RI/5+/1957(H2N2) neuraminidase using 4-MU-Neu5Ac as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed