Compile Data Set for Download or QSAR
Report error Found 63 Enz. Inhib. hit(s) with all data for entry = 50019722
TargetCasein kinase I isoform delta(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300884BDBM50300884((E)-3-(2,4-Dimethoxy-phenyl)-N-(4-[5-(4-fluoro-phe...)
Affinity DataIC50: 4nMAssay Description:Inhibition of CK1delta (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCasein kinase I isoform delta(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50439431BDBM50439431(CHEMBL2420704)
Affinity DataIC50: 6.60nMAssay Description:Inhibition of CK1delta (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCasein kinase I isoform epsilon(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50364141BDBM50364141(CHEMBL1951415)
Affinity DataIC50: 8nMAssay Description:Inhibition of CK1epsilon (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCasein kinase I isoform delta(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50364141BDBM50364141(CHEMBL1951415)
Affinity DataIC50: 14nMAssay Description:Inhibition of CK1delta (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCasein kinase I isoform delta(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50622312BDBM50622312(CHEMBL5397065)
Affinity DataIC50: 18nMAssay Description:Inhibition of CK1delta (unknown origin) using Light-TopoIla(Thr1342) peptide as substrate incubated for 10 mins in presence of ATP by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCasein kinase I isoform epsilon(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50439431BDBM50439431(CHEMBL2420704)
Affinity DataIC50: 28nMAssay Description:Inhibition of CK1epsilon (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCasein kinase I isoform epsilon(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50622312BDBM50622312(CHEMBL5397065)
Affinity DataIC50: 30nMAssay Description:Inhibition of CK1epsilon (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCasein kinase I isoform epsilon(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50399656BDBM50399656(CHEMBL2069623 | US11633415, Compound PF4800567)
Affinity DataIC50: 32nMAssay Description:Inhibition of CK1epsilon (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetCasein kinase I isoform epsilon(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50622286BDBM50622286(CHEMBL5435232)
Affinity DataIC50: 33nMAssay Description:Inhibition of CK1epsilon (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCasein kinase I isoform epsilon(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50622296BDBM50622296(CHEMBL5413697)
Affinity DataIC50: 36nMAssay Description:Inhibition of CK1epsilon (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCasein kinase I isoform delta(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50622286BDBM50622286(CHEMBL5435232)
Affinity DataIC50: 42nMAssay Description:Inhibition of CK1delta (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCasein kinase I isoform delta(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454220BDBM50454220(CHEMBL4211454)
Affinity DataIC50: 44nMAssay Description:Inhibition of CK1delta (unknown origin) using Light-TopoIla(Thr1342) peptide as substrate incubated for 10 mins in presence of ATP by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCasein kinase I isoform epsilon(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50622288BDBM50622288(CHEMBL5424568)
Affinity DataIC50: 58nMAssay Description:Inhibition of CK1epsilon (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCasein kinase I isoform epsilon(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300884BDBM50300884((E)-3-(2,4-Dimethoxy-phenyl)-N-(4-[5-(4-fluoro-phe...)
Affinity DataIC50: 73nMAssay Description:Inhibition of CK1epsilon (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCasein kinase I isoform epsilon(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50622310BDBM50622310(CHEMBL5419193)
Affinity DataIC50: 88nMAssay Description:Inhibition of CK1epsilon (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCasein kinase I isoform epsilon(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50622308BDBM50622308(CHEMBL5435094)
Affinity DataIC50: 100nMAssay Description:Inhibition of CK1epsilon (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCasein kinase I isoform epsilon(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50622311BDBM50622311(CHEMBL5414012)
Affinity DataIC50: 110nMAssay Description:Inhibition of CK1epsilon (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCasein kinase I isoform epsilon(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50622289BDBM50622289(CHEMBL5428835)
Affinity DataIC50: 110nMAssay Description:Inhibition of CK1epsilon (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCasein kinase I isoform epsilon(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50622295BDBM50622295(CHEMBL5409996)
Affinity DataIC50: 180nMAssay Description:Inhibition of CK1epsilon (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCasein kinase I isoform epsilon(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50622287BDBM50622287(CHEMBL5398768)
Affinity DataIC50: 180nMAssay Description:Inhibition of CK1epsilon (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCasein kinase I isoform epsilon(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50622307BDBM50622307(CHEMBL5415170)
Affinity DataIC50: 200nMAssay Description:Inhibition of CK1epsilon (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCasein kinase I isoform delta(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50622310BDBM50622310(CHEMBL5419193)
Affinity DataIC50: 200nMAssay Description:Inhibition of CK1delta (unknown origin) using Light-TopoIla(Thr1342) peptide as substrate incubated for 10 mins in presence of ATP by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCasein kinase I isoform epsilon(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50622294BDBM50622294(CHEMBL5434512)
Affinity DataIC50: 220nMAssay Description:Inhibition of CK1epsilon (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCasein kinase I isoform epsilon(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50622303BDBM50622303(CHEMBL5440959)
Affinity DataIC50: 220nMAssay Description:Inhibition of CK1epsilon (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCasein kinase I isoform epsilon(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50622293BDBM50622293(CHEMBL5413238)
Affinity DataIC50: 230nMAssay Description:Inhibition of CK1epsilon (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCasein kinase I isoform epsilon(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50622309BDBM50622309(CHEMBL5438046)
Affinity DataIC50: 240nMAssay Description:Inhibition of CK1epsilon (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCasein kinase I isoform epsilon(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50622292BDBM50622292(CHEMBL5431532)
Affinity DataIC50: 250nMAssay Description:Inhibition of CK1epsilon (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCasein kinase I isoform epsilon(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454220BDBM50454220(CHEMBL4211454)
Affinity DataIC50: 260nMAssay Description:Inhibition of CK1epsilon (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCasein kinase I isoform epsilon(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50622300BDBM50622300(CHEMBL5407178)
Affinity DataIC50: 340nMAssay Description:Inhibition of CK1epsilon (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCasein kinase I isoform epsilon(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50622290BDBM50622290(CHEMBL5434162)
Affinity DataIC50: 390nMAssay Description:Inhibition of CK1epsilon (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCasein kinase I isoform delta(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50622296BDBM50622296(CHEMBL5413697)
Affinity DataIC50: 400nMAssay Description:Inhibition of CK1delta (unknown origin) using Light-TopoIla(Thr1342) peptide as substrate incubated for 10 mins in presence of ATP by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCasein kinase I isoform delta(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50622311BDBM50622311(CHEMBL5414012)
Affinity DataIC50: 420nMAssay Description:Inhibition of CK1delta (unknown origin) using Light-TopoIla(Thr1342) peptide as substrate incubated for 10 mins in presence of ATP by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCasein kinase I isoform delta(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50622308BDBM50622308(CHEMBL5435094)
Affinity DataIC50: 440nMAssay Description:Inhibition of CK1delta (unknown origin) using Light-TopoIla(Thr1342) peptide as substrate incubated for 10 mins in presence of ATP by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCasein kinase I isoform epsilon(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50622304BDBM50622304(CHEMBL5402454)
Affinity DataIC50: 460nMAssay Description:Inhibition of CK1epsilon (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCasein kinase I isoform epsilon(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50622306BDBM50622306(CHEMBL5395469)
Affinity DataIC50: 570nMAssay Description:Inhibition of CK1epsilon (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCasein kinase I isoform epsilon(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50622298BDBM50622298(CHEMBL5426950)
Affinity DataIC50: 690nMAssay Description:Inhibition of CK1epsilon (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCasein kinase I isoform delta(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50399656BDBM50399656(CHEMBL2069623 | US11633415, Compound PF4800567)
Affinity DataIC50: 711nMAssay Description:Inhibition of CK1delta (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetCasein kinase I isoform epsilon(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50622301BDBM50622301(CHEMBL5406394)
Affinity DataIC50: 740nMAssay Description:Inhibition of CK1epsilon (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCasein kinase I isoform epsilon(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50622291BDBM50622291(CHEMBL5438462)
Affinity DataIC50: 910nMAssay Description:Inhibition of CK1epsilon (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCasein kinase I isoform delta(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50622287BDBM50622287(CHEMBL5398768)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of CK1delta (unknown origin) using Light-TopoIla(Thr1342) peptide as substrate incubated for 10 mins in presence of ATP by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCasein kinase I isoform delta(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50622294BDBM50622294(CHEMBL5434512)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of CK1delta (unknown origin) using Light-TopoIla(Thr1342) peptide as substrate incubated for 10 mins in presence of ATP by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCasein kinase I isoform epsilon(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50622305BDBM50622305(CHEMBL5396131)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of CK1epsilon (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCasein kinase I isoform delta(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50622289BDBM50622289(CHEMBL5428835)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of CK1delta (unknown origin) using Light-TopoIla(Thr1342) peptide as substrate incubated for 10 mins in presence of ATP by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCasein kinase I isoform epsilon(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50622302BDBM50622302(CHEMBL5431478)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of CK1epsilon (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCasein kinase I isoform delta(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50622309BDBM50622309(CHEMBL5438046)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of CK1delta (unknown origin) using Light-TopoIla(Thr1342) peptide as substrate incubated for 10 mins in presence of ATP by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCasein kinase I isoform epsilon(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50622297BDBM50622297(CHEMBL5401196)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of CK1epsilon (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCasein kinase I isoform delta(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50622295BDBM50622295(CHEMBL5409996)
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of CK1delta (unknown origin) using Light-TopoIla(Thr1342) peptide as substrate incubated for 10 mins in presence of ATP by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCasein kinase I isoform epsilon(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50622299BDBM50622299(CHEMBL5436401)
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibition of CK1epsilon (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCasein kinase I isoform delta(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50622288BDBM50622288(CHEMBL5424568)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CK1delta (unknown origin) using Light-TopoIla(Thr1342) peptide as substrate incubated for 10 mins in presence of ATP by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCasein kinase I isoform delta(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50622291BDBM50622291(CHEMBL5438462)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CK1delta (unknown origin) using Light-TopoIla(Thr1342) peptide as substrate incubated for 10 mins in presence of ATP by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
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